日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Pseudo-Natural Product Rhonin Targets RHOGDI

伪天然产物罗宁靶向RHOGDI

Akbarzadeh, Mohammad; Flegel, Jana; Patil, Sumersing; Shang, Erchang; Narayan, Rishikesh; Buchholzer, Marcel; Kazemein Jasemi, Neda S; Grigalunas, Michael; Krzyzanowski, Adrian; Abegg, Daniel; Shuster, Anton; Potowski, Marco; Karatas, Hacer; Karageorgis, George; Mosaddeghzadeh, Niloufar; Zischinsky, Mia-Lisa; Merten, Christian; Golz, Christopher; Brieger, Lucas; Strohmann, Carsten; Antonchick, Andrey P; Janning, Petra; Adibekian, Alexander; Goody, Roger S; Ahmadian, Mohammad Reza; Ziegler, Slava; Waldmann, Herbert

Pseudo Natural Products-Chemical Evolution of Natural Product Structure

拟天然产物——天然产物结构的化学演变

Karageorgis, George; Foley, Daniel J; Laraia, Luca; Brakmann, Susanne; Waldmann, Herbert

Natural product-informed exploration of chemical space to enable bioactive molecular discovery

以天然产物为指导的化学空间探索,助力生物活性分子的发现

Nelson, Adam; Karageorgis, George

Activity-Directed Synthesis: A Flexible Approach for Lead Generation

活性导向合成:一种灵活的先导化合物生成方法

Karageorgis, George; Liver, Samuel; Nelson, Adam

Dataset on the major and trace elements contents and contamination in the sediments of Saronikos Gulf and Elefsis Bay, Greece

希腊萨罗尼科斯湾和埃莱夫西斯湾沉积物中主要元素和微量元素含量及污染情况的数据集

Karageorgis, Aristomenis P; Botsou, Fotini; Kaberi, Helen; Iliakis, Stylianos

Synthesis of Indomorphan Pseudo-Natural Product Inhibitors of Glucose Transporters GLUT-1 and -3

合成吲哚吗啡类拟天然产物抑制剂,该抑制剂可抑制葡萄糖转运蛋白GLUT-1和GLUT-3

Ceballos, Javier; Schwalfenberg, Melanie; Karageorgis, George; Reckzeh, Elena S; Sievers, Sonja; Ostermann, Claude; Pahl, Axel; Sellstedt, Magnus; Nowacki, Jessica; Carnero Corrales, Marjorie A; Wilke, Julian; Laraia, Luca; Tschapalda, Kirsten; Metz, Malte; Sehr, Dominik A; Brand, Silke; Winklhofer, Konstanze; Janning, Petra; Ziegler, Slava; Waldmann, Herbert

A multi-center preclinical study of gadoxetate DCE-MRI in rats as a biomarker of drug induced inhibition of liver transporter function

一项多中心临床前研究,探讨钆塞酸动态对比增强磁共振成像(DCE-MRI)作为药物诱导的肝脏转运蛋白功能抑制生物标志物在大鼠中的应用。

Karageorgis, Anastassia; Lenhard, Stephen C; Yerby, Brittany; Forsgren, Mikael F; Liachenko, Serguei; Johansson, Edvin; Pilling, Mark A; Peterson, Richard A; Yang, Xi; Williams, Dominic P; Ungersma, Sharon E; Morgan, Ryan E; Brouwer, Kim L R; Jucker, Beat M; Hockings, Paul D

Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model

在人源化SCID小鼠模型中,系统性递送肿瘤靶向Bax衍生膜活性肽治疗黑色素瘤

Karageorgis, Anastassia; Claron, Michaël; Jugé, Romain; Aspord, Caroline; Thoreau, Fabien; Leloup, Claire; Kucharczak, Jérôme; Plumas, Joël; Henry, Maxime; Hurbin, Amandine; Verdié, Pascal; Martinez, Jean; Subra, Gilles; Dumy, Pascal; Boturyn, Didier; Aouacheria, Abdel; Coll, Jean-Luc

An MRI-based classification scheme to predict passive access of 5 to 50-nm large nanoparticles to tumors

基于 MRI 的分类方案,用于预测 5 至 50 纳米大纳米粒子被动进入肿瘤的情况

Anastassia Karageorgis, Sandrine Dufort, Lucie Sancey, Maxime Henry, Samuli Hirsjärvi, Catherine Passirani, Jean-Pierre Benoit, Julien Gravier, Isabelle Texier, Olivier Montigon, Mériem Benmerad, Valérie Siroux, Emmanuel L Barbier, Jean-Luc Coll

Activity-Directed Synthesis with Intermolecular Reactions: Development of a Fragment into a Range of Androgen Receptor Agonists

利用分子间反应进行活性导向合成:将片段开发成一系列雄激素受体激动剂

Karageorgis, George; Dow, Mark; Aimon, Anthony; Warriner, Stuart; Nelson, Adam