日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Polyfunctionalized N-Arylsulfonyl Indoles: Identification of (E)-N-Hydroxy-3-{3-[(5-(3-(piperidin-1-yl)propoxy]-1H-indol-1-yl)sulfonyl]phenyl}acrylamide (MTP150) for the Epigenetic-Based Therapy of Parkinson's Disease

多功能化N-芳基磺酰基吲哚:(E)-N-羟基-3-{3-[(5-(3-(哌啶-1-基)丙氧基]-1H-吲哚-1-基)磺酰基]苯基}丙烯酰胺 (MTP150) 的鉴定及其在帕金森病表观遗传治疗中的应用

Toledano-Pinedo, Mireia; Porro-Pérez, Alicia; Schäker-Hübner, Linda; Diez-Iriepa, Daniel; Iriepa, Isabel; Siwek, Agata; Wolak, Małgorzata; Satała, Grzegorz; Bojarski, Andrzej J; Doroz-Płonka, Agata; Handzlik, Jadwiga; Godyń, Justyna; Dallemagne, Patrick; Rochais, Christophe; Davis, Audrey; Since, Marc; Pérez, Belén; Bellver-Sanchis, Aina; Irisarri, Alba; Pallàs, Mercè; Solana-Manrique, Cristina; López-Muñoz, Francisco; Ismaili, Lhassane; Griñán-Ferré, Christian; Paricio, Nuria; K Hansen, Finn; Więckowska, Anna; Marco-Contelles, José

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease

利用多组分合成法制备多靶点喹唑啉类化合物,调节胆碱酯酶、氧化应激和淀粉样蛋白聚集活性,用于治疗阿尔茨海默病

Chakhari, Saida; Marco-Contelles, José; Iriepa, Isabel; Carreiras, Maria do Carmo; Chabchoub, Fakher; Ismaili, Lhassane; Refouvelet, Bernard

Nrf2 Activation and Antioxidant Properties of Chromone-Containing MTDLs for Alzheimer's Disease Treatment

含色酮的MTDLs的Nrf2激活和抗氧化特性及其在阿尔茨海默病治疗中的应用

Simakov, Alexey; Chhor, Stecy; Ismaili, Lhassane; Martin, Hélène

Design and Synthesis of Multi-Functional Ligands through Hantzsch Reaction: Targeting Ca(2+) Channels, Activating Nrf2 and Possessing Cathepsin S Inhibitory, and Antioxidant Properties

利用Hantzsch反应设计合成多功能配体:靶向Ca²⁺通道、激活Nrf2、抑制组织蛋白酶S并具有抗氧化特性

Pachón-Angona, Irene; Bernard, Paul J; Simakov, Alexey; Maj, Maciej; Jozwiak, Krzysztof; Novotna, Anna; Lemke, Carina; Gütschow, Michael; Martin, Helene; Oset-Gasque, María-Jesús; Contelles, José-Marco; Ismaili, Lhassane

Photoluminescence lifetime stability studies of β-diketonate europium complexes based phenanthroline derivatives in poly(methyl methacrylate) films

β-二酮铕配合物(基于菲咯啉衍生物)在聚甲基丙烯酸甲酯薄膜中的光致发光寿命稳定性研究

Essahili, Othmane; Ouafi, Mouad; Ilsouk, Mohamed; Lakbita, Omar; Duhayon, Carine; Mahi, Lhassane; Moudam, Omar

The Proof-of-Concept of MBA121, a Tacrine-Ferulic Acid Hybrid, for Alzheimer's Disease Therapy.

MBA121(一种他克林-阿魏酸混合物)用于治疗阿尔茨海默病的概念验证

Rodríguez-Ruiz Emelina R, Herrero-Labrador Raquel, Fernández-Fernández Ana P, Serrano-Masa Julia, Martínez-Montero José A, González-Nieto Daniel, Hana-Vaish Mayuri, Benchekroun Mohamed, Ismaili Lhassane, Marco-Contelles José, Martínez-Murillo Ricardo

Biginelli Reaction Synthesis of Novel Multitarget-Directed Ligands with Ca2+ Channel Blocking Ability, Cholinesterase Inhibition, Antioxidant Capacity, and Nrf2 Activation

Biginelli 反应合成具有 Ca2+ 通道阻断能力、胆碱酯酶抑制能力、抗氧化能力和 Nrf2 激活能力的新型多靶点配体

Rim Malek, Alexey Simakov, Audrey Davis, Maciej Maj, Paul J Bernard, Artur Wnorowski, Helene Martin, José Marco-Contelles, Fakher Chabchoub, Patrick Dallemagne, Christophe Rochais, Krzysztof Jozwiak, Lhassane Ismaili

Editorial: Advances in drug discovery for anti-Alzheimer's agents

社论:抗阿尔茨海默病药物研发进展

Ismaili, Lhassane

Ferulic acid derivatives block coronaviruses HCoV-229E and SARS-CoV-2 replication in vitro

阿魏酸衍生物在体外可抑制冠状病毒HCoV-229E和SARS-CoV-2的复制

Pasquereau, Sébastien; Galais, Mathilde; Bellefroid, Maxime; Pachón Angona, Irene; Morot-Bizot, Stéphanie; Ismaili, Lhassane; Van Lint, Carine; Herbein, Georges

Triazolopyridopyrimidine: A New Scaffold for Dual-Target Small Molecules for Alzheimer's Disease Therapy

三唑并吡啶并嘧啶:一种用于阿尔茨海默病治疗的双靶点小分子新型支架

Zribi, Lazhar; Pachòn-Angona, Irene; Bautista-Aguilera, Òscar M; Diez-Iriepa, Daniel; Marco-Contelles, José; Ismaili, Lhassane; Iriepa, Isabel; Chabchoub, Fakher