日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Intracellular and in vivo evaluation of imidazo[2,1-b]thiazole-5-carboxamide anti-tuberculosis compounds

咪唑并[2,1-b]噻唑-5-酰胺抗结核化合物的细胞内和体内评价

Garrett C Moraski, Nathalie Deboosère, Kate L Marshall, Heath A Weaver, Alexandre Vandeputte, Courtney Hastings, Lisa Woolhiser, Anne J Lenaerts, Priscille Brodin, Marvin J Miller

Development of a Novel Lead that Targets M. tuberculosis Polyketide Synthase 13

开发一种靶向结核分枝杆菌聚酮合酶13的新型先导化合物

Anup Aggarwal ,Maloy K Parai ,Nishant Shetty ,Deeann Wallis ,Lisa Woolhiser ,Courtney Hastings ,Noton K Dutta ,Stacy Galaviz ,Ramesh C Dhakal ,Rupesh Shrestha ,Shoko Wakabayashi ,Chris Walpole ,David Matthews ,David Floyd ,Paul Scullion ,Jennifer Riley ,Ola Epemolu ,Suzanne Norval ,Thomas Snavely ,Gregory T Robertson ,Eric J Rubin ,Thomas R Ioerger ,Frik A Sirgel ,Ruben van der Merwe ,Paul D van Helden ,Peter Keller ,Erik C Böttger ,Petros C Karakousis ,Anne J Lenaerts ,James C Sacchettini

Discovery of Novel Oral Protein Synthesis Inhibitors of Mycobacterium tuberculosis That Target Leucyl-tRNA Synthetase

发现针对亮氨酰-tRNA 合成酶的新型结核分枝杆菌口服蛋白质合成抑制剂

Andrés Palencia, Xianfeng Li, Wei Bu, Wai Choi, Charles Z Ding, Eric E Easom, Lisa Feng, Vincent Hernandez, Paul Houston, Liang Liu, Maliwan Meewan, Manisha Mohan, Fernando L Rock, Holly Sexton, Suoming Zhang, Yasheen Zhou, Baojie Wan, Yuehong Wang, Scott G Franzblau, Lisa Woolhiser, Veronica Gruppo