日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Highly Potent Noncovalent Inhibitors of SARS-CoV-2 Main Protease through Computer-Aided Drug Design

利用计算机辅助药物设计发现SARS-CoV-2主蛋白酶的高效非共价抑制剂

Okabe, Atsutoshi; Carney, Daniel W; Tawada, Michiko; Akther, Thamina; Aida, Jumpei; Takagi, Terufumi; Dougan, Douglas R; Leffler, Abba E; Bell, Jeffrey A; Frye, Leah; Hickey, Eugene R; Komandla, Mallareddy; Tao, Will; Selimkhanov, Jangir; Yonemori, Kazuko; Chang, Edcon; Saikatendu, Kumar; Ochida, Atsuko

Fluorescence based live cell imaging identifies exon 14 skipped hepatocyte growth factor receptor (MET) degraders

基于荧光的活细胞成像技术可识别外显子14跳跃的肝细胞生长因子受体(MET)降解酶。

Mallareddy, Jayapal Reddy; Yang, Lin; Lin, Wan-Hsin; Feathers, Ryan; Ayers-Ringler, Jennifer; Tolosa, Ezequiel; Kizhake, Amritha G; Kizhake, Smitha; Kubica, Sydney P; Boghean, Lidia; Alvarez, Sophie; Naldrett, Michael J; Singh, Sarbjit; Rana, Sandeep; Zahid, Muhammad; Schaefer-Klein, Janet; Roden, Anja; Kosari, Farhad; Anastasiadis, Panos Z; Borad, Mitesh; Natarajan, Amarnath; Mansfield, Aaron S

Leveraging Artificial Intelligence for the Diagnosis of Systemic Sclerosis Associated Pulmonary Arterial Hypertension: Opportunities, Challenges, and Future Perspectives

利用人工智能诊断系统性硬化症相关肺动脉高压:机遇、挑战与未来展望

Jain, Samiksha; Kaur, Avneet; Qadeer, Abdul; Ghosh, Victor; Thota, Shivani; Banala, Mallareddy; Lee, Jieun; Yerrapragada, Gayathri; Elangovan, Poonguzhali; Shariff, Mohammed Naveed; Natarajan, Thangeswaran; Janarthanan, Jayarajasekaran; Jayapradhaban Kala, Jayavinamika; Richard, Samuel; Vommi, Saai Poornima; Karuppiah, Shiva Sankari; Muthyala, Anjani; Iyer, Vivek N; Helgeson, Scott A; Mitra, Dipankar; Arunachalam, Shivaram P

DHODH inhibition enhances the efficacy of immune checkpoint blockade by increasing cancer cell antigen presentation

DHODH抑制剂通过增加癌细胞抗原呈递来增强免疫检查点阻断的疗效。

Mullen, Nicholas J; Shukla, Surendra K; Thakur, Ravi; Kollala, Sai Sundeep; Wang, Dezhen; Chaika, Nina; Santana, Juan F; Miklavcic, William R; LaBreck, Drew A; Mallareddy, Jayapal Reddy; Price, David H; Natarajan, Amarnath; Mehla, Kamiya; Sykes, David B; Hollingsworth, Michael A; Singh, Pankaj K

Proteolysis targeting chimera (PROTAC)-driven antibody internalization of oncogenic cell surface receptors

蛋白水解靶向嵌合体(PROTAC)驱动的致癌细胞表面受体抗体内化

Ezequiel J Tolosa ,Lin Yang ,Jennifer Ayers-Ringler ,Shinichiro Suzuki ,Jayapal Reddy Mallareddy ,Janet Schaefer-Klein ,Mitesh Borad ,Farhad Kosari ,Amarnath Natarajan ,Aaron S Mansfield

Novel Spirocyclic Dimer, SpiD3, Targets Chronic Lymphocytic Leukemia Survival Pathways with Potent Preclinical Effects

新型螺环二聚体 SpiD3 靶向慢性淋巴细胞白血病生存途径,具有强效临床前效应

Alexandria P Eiken, Audrey L Smith, Sydney A Skupa, Elizabeth Schmitz, Sandeep Rana, Sarbjit Singh, Siddhartha Kumar, Jayapal Reddy Mallareddy, Aguirre A de Cubas, Akshay Krishna, Achyuth Kalluchi, M Jordan Rowley, Christopher R D'Angelo, Matthew A Lunning, R Gregory Bociek, Julie M Vose, Amarnath N

Central Corneal Thickness and Endothelial Cell Changes in Diabetics and Age-Matched Non-diabetics in a Tertiary Care Hospital in Central India

印度中部一家三级医院糖尿病患者和年龄匹配的非糖尿病患者的中央角膜厚度和内皮细胞变化

Daigavane, Sachin; Mallareddy, Vijaya

Nanoparticle-Mediated Cell Delivery: Advancements in Corneal Endothelial Regeneration

纳米颗粒介导的细胞递送:角膜内皮再生技术的进展

Mallareddy, Vijaya; Daigavane, Sachin

Enhancing Prenatal Group Medical Visits with Mindfulness Skills: A Pragmatic Trial with Latina and BIPOC Pregnant Women Experiencing Multiple Forms of Structural Inequity

利用正念技巧提升产前团体医疗就诊体验:一项针对面临多种结构性不平等的拉丁裔和有色人种孕妇的实用性试验

Duncan, Larissa G; Zhang, Na; Santana, Trilce; Cook, Joseph G; Castro-Smyth, Lisabeth; Hutchison, Margaret S; Huynh, Tuyen; Mallareddy, Deena; Jurkiewicz, Laurie; Bardacke, Nancy

The Novel Anti-Cancer Agent, SpiD3, Is Cytotoxic in CLL Cells Resistant to Ibrutinib or Venetoclax

新型抗癌药物 SpiD3 对对伊布替尼或维奈克拉具有耐药性的 CLL 细胞具有细胞毒性

Alexandria P Eiken, Elizabeth Schmitz, Erin M Drengler, Audrey L Smith, Sydney A Skupa, Kabhilan Mohan, Sandeep Rana, Sarbjit Singh, Jayapal Reddy Mallareddy, Grinu Mathew, Amarnath Natarajan, Dalia El-Gamal