日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5'-Terminal Oligopyrimidine Motif-Containing mRNA

磺酰邻氨基苯甲酸类似物通过下调由含5'末端寡嘧啶基序的mRNA编码的核糖体蛋白的表达,表现出泛血清型抗登革热活性。

Gwee, Chin Piaw; Felicetti, Tommaso; Chan, Kitti Wing Ki; Tan, Min Jie Alvin; Bin Mohd Mazlan, Muhammad Danial; Milite, Ciro; Pepe, Giacomo; Sarnari, Chiara; Ng, Xiao Dan; Phoo, Wint Wint; Tan, Jasmine Hwee Yee; Mah, Marcus G; Watanabe, Satoru; Huang, Jing Xiu; Massari, Serena; Tabarrini, Oriana; Sabatini, Stefano; Campiglia, Pietro; Sbardella, Gianluca; Smith, Gavin J D; Alonso, Sylvie; Sun, Alfred Xuyang; Sobota, Radoslaw M; Vasudevan, Subhash G; Manfroni, Giuseppe

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3-c][1,2]benzothiazine 5,5-Dioxide Derivatives

NorA 外排泵抑制剂:扩展吡唑并[4,3-c][1,2]苯并噻嗪 5,5-二氧化物衍生物的构效关系知识

Cernicchi, Giada; Di Gregorio, Alessandra; Felicetti, Tommaso; Rampacci, Elisa; Casari, Giulia; Armeni, Tatiana; Romaldi, Brenda; Zefaj, Ermelinda; Passamonti, Fabrizio; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Vignaroli, Carla; Sabatini, Stefano

Broad-Spectrum Antiviral Activity of Pyridobenzothiazolone Analogues Against Respiratory Viruses.

吡啶并苯并噻唑啉酮类似物对呼吸道病毒的广谱抗病毒活性

Feyles Elisa, Felicetti Tommaso, Arduino Irene, Rittà Massimo, Civra Andrea, Muratori Luisa, Raimondo Stefania, Lembo David, Manfroni Giuseppe, Donalisio Manuela

New Pyridobenothiazolone Derivatives Display Nanomolar Pan-Serotype Anti-Dengue Virus Activity.

新型吡啶并噻唑啉酮衍生物显示出纳摩尔级泛血清型抗登革病毒活性

Felicetti Tommaso, Gwee Chin Piaw, Chan Kitti Wing Ki, Pepe Giacomo, Milite Ciro, Campiglia Pietro, Watanabe Satoru, Mazlan Muhammad Danial Bin Mohd, Sabatini Stefano, Massari Serena, Tabarrini Oriana, Sbardella Gianluca, Vasudevan Subhash G, Manfroni Giuseppe

Small Molecule Drugs Targeting Viral Polymerases

靶向病毒聚合酶的小分子药物

Palazzotti, Deborah; Sguilla, Martina; Manfroni, Giuseppe; Cecchetti, Violetta; Astolfi, Andrea; Barreca, Maria Letizia

Synthetically accessible de novo design using reaction vectors: Application to PARP1 inhibitors

利用反应载体进行合成可及的从头设计:应用于PARP1抑制剂

Ghiandoni, Gian Marco; Flanagan, Stuart R; Bodkin, Michael J; Nizi, Maria Giulia; Galera-Prat, Albert; Brai, Annalaura; Chen, Beining; Wallace, James E A; Hristozov, Dimitar; Webster, James; Manfroni, Giuseppe; Lehtiö, Lari; Tabarrini, Oriana; Gillet, Valerie J

Modulating microRNA Processing: Enoxacin, the Progenitor of a New Class of Drugs

调控microRNA加工:依诺沙星,一类新型药物的先驱

Felicetti, Tommaso; Cecchetti, Violetta; Manfroni, Giuseppe

Comprehensive response to Usutu virus following first isolation in blood donors in the Friuli Venezia Giulia region of Italy: Development of recombinant NS1-based serology and sensitivity to antiviral drugs

意大利弗留利-威尼斯朱利亚大区首次从献血者中分离出乌苏图病毒后,采取了全面的应对措施:开发基于重组NS1的血清学检测方法及抗病毒药物敏感性检测

Caracciolo, Ilaria; Mora-Cardenas, Erick; Aloise, Chiara; Carletti, Tea; Segat, Ludovica; Burali, Maria Sole; Chiarvesio, Alexsia; Totis, Vivianna; Avšič-Županc, Tatjana; Mastrangelo, Eloise; Manfroni, Giuseppe; D'Agaro, Pierlanfranco; Marcello, Alessandro

Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli

2-苯基喹啉外排抑制剂PQQ4R对大肠杆菌的作用机制

Machado, Diana; Fernandes, Laura; Costa, Sofia S; Cannalire, Rolando; Manfroni, Giuseppe; Tabarrini, Oriana; Couto, Isabel; Sabatini, Stefano; Viveiros, Miguel