日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Optimization of Pyridone α-Ketoamides as Inhibitors of the SARS-CoV-2 Main Protease

基于结构的吡啶酮α-酮酰胺类化合物作为SARS-CoV-2主蛋白酶抑制剂的优化

Akula, Ravi Kumar; El Kilani, Haifa; Metzen, Alina; Röske, Judith; Zhang, Kaixuan; Göhl, Matthias; Arisetti, Nanaji; Marsh, Graham P; Maple, Hannah J; Cooper, Mark S; Karadogan, Burhan; Jochmans, Dirk; Neyts, Johan; Rox, Katharina; Hilgenfeld, Rolf; Brönstrup, Mark

Structure-Guided Design of ISOX-DUAL-Based Degraders Targeting BRD4 and CBP/EP300: A Case of Degrader Collapse.

基于 ISOX-DUAL 的结构导向降解剂设计:针对 BRD4 和 CBP/EP300 的降解剂崩溃案例

Edmonds Anthony K, Balourdas Dimitrios-Ilias, Marsh Graham P, Felix Robert, Brasher Bradley, Cooper Jeff, Graber-Feesl Cari, Kollareddy Madhu, Malik Karim, Stewart Helen, Chevassut Timothy J T, Lineham Ella, Morley Simon, Fedorov Oleg, Bennett James, Rajasekaran Mohan B, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Joerger Andreas C, Maple Hannah J, Spencer John

Development of p300-targeting degraders with enhanced selectivity and onset of degradation.

开发具有增强选择性和更快降解速度的p300靶向降解剂

Marsh Graham P, Cooper Mark S, Goggins Sean, Reynolds Stephen J, Wheeler Dean F, Cresser-Brown Joel O, Arnold Robert E, Babcock Emily G, Hughes Gareth, Bosnakovski Darko, Kyba Michael, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Maple Hannah J

Chirality: a key parameter in chemical probes

手性:化学探针的关键参数

McGown, Andrew; Nafie, Jordan; Otayfah, Mohammed; Hassell-Hart, Storm; Tizzard, Graham J; Coles, Simon J; Banks, Rebecca; Marsh, Graham P; Maple, Hannah J; Kostakis, George E; Proietti Silvestri, Ilaria; Colbon, Paul; Spencer, John

Developing degraders: principles and perspectives on design and chemical space

降解剂的开发:设计和化学空间的原则和视角

Maple, Hannah J; Clayden, Nat; Baron, Anne; Stacey, Callum; Felix, Robert