日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Extrahelical Binding Site for a 1 H-Imidazo[4,5-c]quinolin-4-amine A3 Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7

H-咪唑并[4,5-c]喹啉-4-胺 A3 腺苷受体正变构调节剂在螺旋 8 和跨膜域 1 和 7 的远端部分的螺旋外结合位点

Courtney L Fisher, Matteo Pavan, Veronica Salmaso, Robert F Keyes, Tina C Wan, Balaram Pradhan, Zhan-Guo Gao, Brian C Smith, Kenneth A Jacobson, John A Auchampach

A deep learning approach to investigate the filtration bleb functionality after glaucoma surgery: a preliminary study

利用深度学习方法研究青光眼手术后滤过泡功能:一项初步研究

Mastropasqua, Leonardo; Agnifili, Luca; Brescia, Lorenza; Figus, Michele; Posarelli, Chiara; Oddone, Francesco; Giammaria, Sara; Sacchi, Matteo; Pavan, Marco; Innocenti, Dante Degli; Olivotto, Valentina; Sensi, Stefano L; Mastropasqua, Rodolfo

SARS-CoV-2 3CLpro mutations selected in a VSV-based system confer resistance to nirmatrelvir, ensitrelvir, and GC376

在基于 VSV 的系统中筛选出的 SARS-CoV-2 3CLpro 突变导致对尼玛瑞韦、恩西瑞韦和 GC376 产生耐药性

Emmanuel Heilmann, Francesco Costacurta, Seyed Arad Moghadasi, Chengjin Ye, Matteo Pavan, Davide Bassani, Andre Volland, Claudia Ascher, Alexander Kurt Hermann Weiss, David Bante, Reuben S Harris, Stefano Moro, Bernhard Rupp, Luis Martinez-Sobrido, Dorothee von Laer

Streptogramin A derivatives as mitochondrial translation inhibitors to suppress glioblastoma stem cell growth

链霉菌素 A 衍生物作为线粒体翻译抑制剂抑制胶质母细胞瘤干细胞生长

Denise Sighel, Giulia Battistini, Emanuele Filiberto Rosatti, Jacopo Vigna, Matteo Pavan, Romina Belli, Daniele Peroni, Federica Alessandrini, Sara Longhi, Michael Pancher, Joanna Rorbach, Stefano Moro, Alessandro Quattrone, Ines Mancini

Discovery of the 3-Amino-1,2,4-triazine-Based Library as Selective PDK1 Inhibitors with Therapeutic Potential in Highly Aggressive Pancreatic Ductal Adenocarcinoma

发现 3-氨基-1,2,4-三嗪类化合物库作为选择性 PDK1 抑制剂,具有治疗高侵袭性胰腺导管腺癌的潜力

Daniela Carbone, Michele De Franco, Camilla Pecoraro, Davide Bassani, Matteo Pavan, Stella Cascioferro, Barbara Parrino, Girolamo Cirrincione, Stefano Dall'Acqua, Stefano Moro, Valentina Gandin, Patrizia Diana

"Dual Anta-Inhibitors" of the A2A Adenosine Receptor and Casein Kinase CK1delta: Synthesis, Biological Evaluation, and Molecular Modeling Studies

A2A 腺苷受体和酪蛋白激酶 CK1delta 的“双重拮抗剂”:合成、生物学评价和分子建模研究

Andrea Spinaci, Michela Buccioni, Daniela Catarzi, Chang Cui, Vittoria Colotta, Diego Dal Ben, Eleonora Cescon, Beatrice Francucci, Ilenia Grieco, Catia Lambertucci, Gabriella Marucci, Davide Bassani, Matteo Pavan, Flavia Varano, Stephanie Federico, Giampiero Spalluto, Stefano Moro, Rosaria Volpini

Reconstructing reactivity in dynamic host-guest systems at atomistic resolution: amide hydrolysis under confinement in the cavity of a coordination cage

以原子级分辨率重构动态主客体体系中的反应性:配位笼空腔限域下的酰胺水解

Delle Piane, Massimo; Pesce, Luca; Cioni, Matteo; Pavan, Giovanni M

Into the Dynamics of a Supramolecular Polymer at Submolecular Resolution

亚分子分辨率下超分子聚合物的动力学研究

Bochicchio, Davide; Salvalaglio, Matteo; Pavan, Giovanni M

Gadolinium MRI contrast agents based on triazine dendrimers: relaxivity and in vivo pharmacokinetics

基于三嗪树状聚合物的钆磁共振造影剂:弛豫率和体内药代动力学

Lim, Jongdoo; Turkbey, Baris; Bernardo, Marcelino; Bryant, L Henry Jr; Garzoni, Matteo; Pavan, Giovanni M; Nakajima, Takahito; Choyke, Peter L; Simanek, Eric E; Kobayashi, Hisataka