Imlunestrant Is an Oral, Brain-Penetrant Selective Estrogen Receptor Degrader with Potent Antitumor Activity in ESR1 Wild-Type and Mutant Breast Cancer
Imlunestrant 是一种口服、脑渗透性选择性雌激素受体降解剂,对 ESR1 野生型和突变型乳腺癌具有强效抗肿瘤活性
期刊:Cancer Research
影响因子:12.5
doi:10.1158/0008-5472.CAN-24-2608
Shripad V Bhagwat #, Cecilia Mur #, Matthew Vandekopple #, Baohui Zhao, Weihua Shen, Carlos Marugán, Andrew Capen, Lisa Kindler, Jennifer R Stephens, Lysiane Huber, Mark A Castanares, David Garcia-Tapia, Jeff D Cohen, Jolie Bastian, Brian Mattioni, Eunice Yuen, Thomas K Baker, Vivian Rodriguez Cruz,