日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Low-level whole-brain radiation enhances theranostic potential of single-domain antibody fragments for human epidermal growth factor receptor type 2 (HER2)-positive brain metastases

低剂量全脑放射治疗可增强单域抗体片段对人表皮生长因子受体2型(HER2)阳性脑转移瘤的诊疗潜力

Procissi, Daniele; Jannetti, Stephen A; Zannikou, Markella; Zhou, Zhengyuan; McDougald, Darryl; Kanojia, Deepak; Zhang, Hui; Burdett, Kirsten; Vaidyanathan, Ganesan; Zalutsky, Michael R; Balyasnikova, Irina V

Synthesis and preliminary evaluation of (211)At-labeled inhibitors of prostate-specific membrane antigen for targeted alpha particle therapy of prostate cancer

合成并初步评价(211)At标记的前列腺特异性膜抗原抑制剂在前列腺癌靶向α粒子治疗中的应用

Vaidyanathan, Ganesan; Mease, Ronnie C; Minn, Il; Choi, Jaeyeon; Chen, Ying; Shallal, Hassan; Kang, Choong Mo; McDougald, Darryl; Kumar, Vivek; Pomper, Martin G; Zalutsky, Michael R

Labeling Single Domain Antibody Fragments with Fluorine-18 Using 2,3,5,6-Tetrafluorophenyl 6-[(18)F]Fluoronicotinate Resulting in High Tumor-to-Kidney Ratios

利用 2,3,5,6-四氟苯基 6-[(18)F]氟烟酸酯对单域抗体片段进行氟-18 标记,可获得较高的肿瘤/肾脏比率

Zhou, Zhengyuan; McDougald, Darryl; Devoogdt, Nick; Zalutsky, Michael R; Vaidyanathan, Ganesan

Fluorine-18 Labeling of the HER2-Targeting Single-Domain Antibody 2Rs15d Using a Residualizing Label and Preclinical Evaluation

利用残留标记对靶向 HER2 的单域抗体 2Rs15d 进行氟-18 标记及其临床前评估

Zhou, Zhengyuan; Vaidyanathan, Ganesan; McDougald, Darryl; Kang, Choong Mo; Balyasnikova, Irina; Devoogdt, Nick; Ta, Angeline N; McNaughton, Brian R; Zalutsky, Michael R

Preclinical Evaluation of 18F-Labeled Anti-HER2 Nanobody Conjugates for Imaging HER2 Receptor Expression by Immuno-PET

利用免疫PET成像技术对18F标记的抗HER2纳米抗体偶联物进行HER2受体表达成像的临床前评估

Vaidyanathan, Ganesan; McDougald, Darryl; Choi, Jaeyeon; Koumarianou, Eftychia; Weitzel, Douglas; Osada, Takuya; Lyerly, H Kim; Zalutsky, Michael R

Synthesis and evaluation of 4-[18F]fluoropropoxy-3-iodobenzylguanidine ([18F]FPOIBG): A novel 18F-labeled analogue of MIBG

4-[18F]氟丙氧基-3-碘苄胍 ([18F]FPOIBG) 的合成与评价:一种新型的 18F 标记的 MIBG 类似物

Vaidyanathan, Ganesan; McDougald, Darryl; Koumarianou, Eftychia; Choi, Jaeyeon; Hens, Marc; Zalutsky, Michael R

N-Succinimidyl guanidinomethyl iodobenzoate protein radiohalogenation agents: influence of isomeric substitution on radiolabeling and target cell residualization

N-琥珀酰亚胺基胍基甲基碘苯甲酸酯蛋白放射性卤化剂:异构体取代对放射性标记和靶细胞残留的影响

Choi, Jaeyeon; Vaidyanathan, Ganesan; Koumarianou, Eftychia; McDougald, Darryl; Pruszynski, Marek; Osada, Takuya; Lahoutte, Tony; Lyerly, H Kim; Zalutsky, Michael R

Radioiodinated O(6)-Benzylguanine derivatives containing an azido function.

含有叠氮基团的放射性碘标记的 O(6)-苄基鸟嘌呤衍生物

Vaidyanathan Ganesan, White Benjamin, Affleck Donna J, McDougald Darryl, Zalutsky Michael R

An alternative and expedient synthesis of radioiodinated 4-iodophenylalanine

放射性碘标记的4-碘苯丙氨酸的一种替代且简便的合成方法

Vaidyanathan, Ganesan; McDougald, Darryl; Grasfeder, Linda; Zalutsky, Michael R; Chin, Bennett

Targeting aldehyde dehydrogenase: a potential approach for cell labeling

靶向醛脱氢酶:一种潜在的细胞标记方法

Vaidyanathan, Ganesan; Song, Haijing; Affleck, Donna; McDougald, Darryl L; Storms, Robert W; Zalutsky, Michael R; Chin, Bennett B