日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

AI-driven discovery of synergistic drug combinations against pancreatic cancer.

利用人工智能发现对抗胰腺癌的协同药物组合

Pourmousa Mohsen, Jain Sankalp, Barnaeva Elena, Jin Wengong, Hochuli Joshua, Itkin Zina, Maxfield Travis, Melo-Filho Cleber, Thieme Andrew, Wilson Kelli, Klumpp-Thomas Carleen, Michael Sam, Southall Noel, Jaakkola Tommi, Muratov Eugene N, Barzilay Regina, Tropsha Alexander, Ferrer Marc, Zakharov Alexey V

Dona Flor and her two husbands: Discovery of novel HDAC6/AKT2 inhibitors for myeloid cancer treatment

唐娜·弗洛尔和她的两位丈夫:发现用于治疗髓系癌症的新型HDAC6/AKT2抑制剂

Waitman, Karoline B; Martin, Holli-Joi; Carlos, Jorge A E G; Braga, Rodolpho C; Souza, Vinícius A M; Melo-Filho, Cleber C; Hilscher, Sebastian; Toledo, Mônica F Z J; Tavares, Maurício T; Costa-Lotufo, Letícia V; Machado-Neto, João A; Schutkowski, Mike; Sippl, Wolfgang; Kronenberger, Thales; Alves, Vinicius M; Parise-Filho, Roberto; Muratov, Eugene N

On the importance of data curation for knowledge mining in antiviral research

数据整理对于抗病毒研究知识挖掘的重要性

Martin, Holli-Joi; Melo-Filho, Cleber C; Zakharov, Alexey V; Muratov, Eugene; Tropsha, Alexander

Conserved Filovirus Proteins as Targets of Broad-Spectrum Antivirals

保守的丝状病毒蛋白作为广谱抗病毒药物的靶点

Scotti, Marcus Tullius; Kelestemur, Enes; Martin, Holli-Joi; Novy, Brandon; Melo-Filho, Cleber C; de Menezes, Renata Priscila Barros; Herrera-Acevedo, Chonny; Tropsha, Alexander; Muratov, Eugene N

Modeling interactions between Heparan sulfate and proteins based on the Heparan sulfate microarray analysis

基于硫酸乙酰肝素微阵列分析构建硫酸乙酰肝素与蛋白质相互作用模型

Melo-Filho, Cleber C; Su, Guowei; Liu, Kevin; Muratov, Eugene N; Tropsha, Alexander; Liu, Jian

Conserved coronavirus proteins as targets of broad-spectrum antivirals

冠状病毒的保守蛋白作为广谱抗病毒药物的靶点

Melo-Filho, Cleber C; Bobrowski, Tesia; Martin, Holli-Joi; Sessions, Zoe; Popov, Konstantin I; Moorman, Nathaniel J; Baric, Ralph S; Muratov, Eugene N; Tropsha, Alexander

Small Molecule Antiviral Compound Collection (SMACC): a database to support the discovery of broad-spectrum antiviral drug molecules

小分子抗病毒化合物库(SMACC):一个支持发现广谱抗病毒药物分子的数据库

Martin, Holli-Joi; Melo-Filho, Cleber C; Korn, Daniel; Eastman, Richard T; Rai, Ganesha; Simeonov, Anton; Zakharov, Alexey V; Muratov, Eugene; Tropsha, Alexander

Learning from history: do not flatten the curve of antiviral research!

从历史中吸取教训:不要让抗病毒研究的曲线变平!

Bobrowski, Tesia; Melo-Filho, Cleber C; Korn, Daniel; Alves, Vinicius M; Popov, Konstantin I; Auerbach, Scott; Schmitt, Charles; Moorman, Nathaniel J; Muratov, Eugene N; Tropsha, Alexander

QSAR-Based Virtual Screening: Advances and Applications in Drug Discovery

基于QSAR的虚拟筛选:药物发现的进展与应用

Neves, Bruno J; Braga, Rodolpho C; Melo-Filho, Cleber C; Moreira-Filho, José Teófilo; Muratov, Eugene N; Andrade, Carolina Horta

Computer-aided discovery of two novel chalcone-like compounds active and selective against Leishmania infantum

利用计算机辅助发现两种对婴儿利什曼原虫具有活性和选择性的新型查尔酮类化合物

Gomes, Marcelo N; Alcântara, Laura M; Neves, Bruno J; Melo-Filho, Cleber C; Freitas-Junior, Lucio H; Moraes, Carolina B; Ma, Rui; Franzblau, Scott G; Muratov, Eugene; Andrade, Carolina Horta