日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New scaffolds for type II JAK2 inhibitors overcome the acquired G993A resistance mutation

新型 II 型 JAK2 抑制剂支架克服了获得的 G993A 耐药突变

Matthew L Arwood ,Yao Liu ,Shannon K Harkins ,David M Weinstock ,Lei Yang ,Kristen E Stevenson ,Olivia D Plana ,Jingyun Dong ,Haley Cirka ,Kristen L Jones ,Anniina T Virtanen ,Dikshat G Gupta ,Amanda Ceas ,Brian Lawney ,Akinori Yoda ,Catharine Leahy ,Mingfeng Hao ,Zhixiang He ,Hwan Geun Choi ,Yaning Wang ,Olli Silvennoinen ,Stevan R Hubbard ,Tinghu Zhang ,Nathanael S Gray ,Loretta S Li

Human Polo-like Kinase Inhibitors as Antiplasmodials

人 Polo 样激酶抑制剂作为抗疟疾药物

Monica J Bohmer ,Jinhua Wang ,Eva S Istvan ,Madeline R Luth ,Jennifer E Collins ,Edward L Huttlin ,Lushun Wang ,Nimisha Mittal ,Mingfeng Hao ,Nicholas P Kwiatkowski ,Steven P Gygi ,Ratna Chakrabarti ,Xianming Deng ,Daniel E Goldberg ,Elizabeth A Winzeler ,Nathanael S Gray ,Debopam Chakrabarti

Development and Characterization of Selective FAK Inhibitors and PROTACs with In Vivo Activity

具有体内活性的选择性 FAK 抑制剂和 PROTAC 的开发和表征

Eriko Koide, Mikaela L Mohardt, Zainab M Doctor, Annan Yang, Mingfeng Hao, Katherine A Donovan, Christina C Kuismi, Alissa J Nelson, Kathryn Abell, Mike Aguiar, Jianwei Che, Matthew P Stokes, Tinghu Zhang, Andrew J Aguirre, Eric S Fischer, Nathanael S Gray, Baishan Jiang, Behnam Nabet

Mapping the Degradable Kinome Provides a Resource for Expedited Degrader Development

绘制可降解激酶组图谱为加速降解剂开发提供资源

Katherine A Donovan, Fleur M Ferguson, Jonathan W Bushman, Nicholas A Eleuteri, Debabrata Bhunia, SeongShick Ryu, Li Tan, Kun Shi, Hong Yue, Xiaoxi Liu, Dennis Dobrovolsky, Baishan Jiang, Jinhua Wang, Mingfeng Hao, Inchul You, Mingxing Teng, Yanke Liang, John Hatcher, Zhengnian Li, Theresa D Manz, B

NUAK2 is a critical YAP target in liver cancer

NUAK2 是肝癌中的关键 YAP 靶点

Wei-Chien Yuan, Brian Pepe-Mooney, Giorgio G Galli, Michael T Dill, Hai-Tsang Huang, Mingfeng Hao, Yumeng Wang, Han Liang, Raffaele A Calogero, Fernando D Camargo

Targeting MYC dependency in ovarian cancer through inhibition of CDK7 and CDK12/13

通过抑制 CDK7 和 CDK12/13 靶向卵巢癌中的 MYC 依赖性

Mei Zeng, Nicholas P Kwiatkowski, Tinghu Zhang, Behnam Nabet, Mousheng Xu, Yanke Liang, Chunshan Quan, Jinhua Wang, Mingfeng Hao, Sangeetha Palakurthi, Shan Zhou, Qing Zeng, Paul T Kirschmeier, Khyati Meghani, Alan L Leggett, Jun Qi, Geoffrey I Shapiro, Joyce F Liu, Ursula A Matulonis, Charles Y Lin

Covalent targeting of remote cysteine residues to develop CDK12 and CDK13 inhibitors

共价靶向远端半胱氨酸残基以开发 CDK12 和 CDK13 抑制剂

Tinghu Zhang, Nicholas Kwiatkowski, Calla M Olson, Sarah E Dixon-Clarke, Brian J Abraham, Ann K Greifenberg, Scott B Ficarro, Jonathan M Elkins, Yanke Liang, Nancy M Hannett, Theresa Manz, Mingfeng Hao, Bartlomiej Bartkowiak, Arno L Greenleaf, Jarrod A Marto, Matthias Geyer, Alex N Bullock, Richard