日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Lead Optimization: Synthesis and Biological Evaluation of Griseofulvin Derivatives as Novel SIRT6 Activators

先导化合物优化:灰黄霉素衍生物作为新型SIRT6激活剂的合成及生物学评价

Zorko, Tilen; Kogovšek, Jan; Ciber, Luka; Ostojić, Ivana; Maraš, Nenad; Novinec, Marko; Štefane, Bogdan

Cooperativity in Escherichia coli L-Threonine Dehydrogenase and Its Inhibition by an Antibacterial N-Pyridylpyrazolone Derivative

大肠杆菌L-苏氨酸脱氢酶的协同作用及其被抗菌N-吡啶基吡唑酮衍生物抑制

Obaha, Ana; Mikulič Vernik, Nika; Mlinar, Karmen; Tušek, Marcel; Stojkovska Docevska, Milena; Petek, Nejc; Svete, Jurij; Novinec, Marko

Synthesis of Bioconjugation Reagents for Use in Covalent Cross-Linking of Proteins by Azide-Alkyne Cycloaddition

利用叠氮-炔环加成反应合成用于蛋白质共价交联的生物偶联试剂

Suhorepec, Nadja; Ciber, Luka; Grošelj, Uroš; Petek, Nejc; Štefane, Bogdan; Novinec, Marko; Svete, Jurij

New achievements in orbital angular momentum beam characterization using a Hartmann wavefront sensor and the Kirkpatrick-Baez active optical system KAOS

利用哈特曼波前传感器和柯克帕特里克-贝兹主动光学系统KAOS在轨道角动量光束表征方面取得的新成果

Novinec, Luka; Pancaldi, Matteo; Capotondi, Flavio; De Ninno, Giovanni; Guzzi, Francesco; Kourousias, George; Pedersoli, Emanuele; Ressel, Barbara; Rösner, Benedikt; Simoncig, Alberto; Zangrando, Marco; Manfredda, Michele

Activity-based probes trap early active intermediates during metacaspase activation

基于活性的探针在半胱天冬酶活化过程中捕获早期活性中间体

Vida Štrancar, Katarina P van Midden, Daniel Krahn, Kyoko Morimoto, Marko Novinec, Christiane Funk, Simon Stael, Christopher J Schofield, Marina Klemenčič, Renier A L van der Hoorn

Structural polymorphism of coiled-coils from the stalk domain of SARS-CoV-2 spike protein

SARS-CoV-2刺突蛋白茎部结构域卷曲螺旋的结构多态性

Živič, Zala; Strmšek, Žiga; Novinec, Marko; Lah, Jurij; Hadži, San

Regioselective Synthesis of 5- and 3-Hydroxy- N-Aryl-1 H-Pyrazole-4-Carboxylates and Their Evaluation as Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase

5- 和 3-羟基-N-芳基-1 H-吡唑-4-羧酸的区域选择性合成及其作为恶性疟原虫二氢乳清酸脱氢酶抑制剂的评价

Luka Vah, Tadej Medved, Uroš Grošelj, Marina Klemenčič, Črtomir Podlipnik, Bogdan Štefane, Jernej Wagger, Marko Novinec, Jurij Svete

Kinetic Characterization of Cerium and Gallium Ions as Inhibitors of Cysteine Cathepsins L, K, and S

铈和镓离子作为半胱氨酸蛋白酶 L、K 和 S 抑制剂的动力学表征

Marko Novinec, Primož Bembič, Milica Janković, Marija Kisilak, Jakob Kljun, Iztok Turel

Inhibition of Human Cathepsins B and L by Caffeic Acid and Its Derivatives

咖啡酸及其衍生物对人类组织蛋白酶B和L的抑制

Liza Ulčakar, Marko Novinec

Cathepsin K cleavage of SDF-1α inhibits its chemotactic activity towards glioblastoma stem-like cells

组织蛋白酶 K 切割 SDF-1α 可抑制其对胶质母细胞瘤干细胞样细胞的趋化活性

Vashendriya V V Hira, Urška Verbovšek, Barbara Breznik, Matic Srdič, Marko Novinec, Hala Kakar, Jill Wormer, Britt Van der Swaan, Brigita Lenarčič, Luiz Juliano, Shwetal Mehta, Cornelis J F Van Noorden, Tamara T Lah