日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An engineered trafficking biosensor reveals a role for DNAJC13 in DOR downregulation.

工程化运输生物传感器揭示了 DNAJC13 在 DOR 下调中的作用

Novy Brandon, Dagunts Aleksandra, Weishaar Tatum, Holland Emily E, Adoff Hayden, Hutchinson Emily, De Maria Monica, Kampmann Martin, Tsvetanova Nikoleta G, Lobingier Braden T

A Hit Prioritization Strategy for Compound Library Screening Using LiP-MS and Molecular Dynamics Simulations Applied to KRas G12D Inhibitors

基于LiP-MS和分子动力学模拟的化合物库筛选先导化合物优先级排序策略及其在KRas G12D抑制剂中的应用

Absar, Foroughsadat; Novy, Brandon; Nagy, Edith; Petrotchenko, Evgeniy V; Popov, Konstantin I; Cross, Jason B; Thapar, Roopa; Borchers, Christoph H

Characterization of the KRas G12D-inhibitor interactions by differential HDX-MS and molecular dynamics simulations

利用差分氢氘交换质谱和分子动力学模拟表征KRas G12D-抑制剂相互作用

Petrotchenko, Evgeniy V; Novy, Brandon; Nagy, Edith; Popov, Konstantin I; Cross, Jason B; Thapar, Roopa; Borchers, Christoph H

DNAJC13 localization to endosomes is opposed by its J domain and its disordered C-terminus.

DNAJC13 定位于内体受到其 J 结构域和无序 C 末端的阻碍

Adoff Hayden, Novy Brandon, Holland Emily, Lobingier Braden T

Open-Source DNA-Encoded Library informatics Package for Design, Decoding, and Analysis: DELi

用于设计、解码和分析的开源DNA编码文库信息学软件包:DELi

Wellnitz, James; Novy, Brandon; Maxfield, Travis; Lin, Shu-Hang; Zhilinskaya, Ivanna; Axtman, Matthew; Leisner, Tina; Merten, Eric; Norris-Drouin, Jacqueline L; Hardy, Brian P; Pearce, Kenneth H; Popov, Konstantin I

Expansion of DNA-Encoded Library Hits Using Generative Chemistry and Ultra-Large Compound Catalogs

利用生成化学和超大型化合物目录扩展DNA编码化合物库

Novy, Brandon; Lin, Shu-Hang; Shell, Devan J; Maxfield, Travis; Merten, Eric M; Wellnitz, James; Guduru, Shiva K R; Hardy, P Brian; Pearce, Kenneth H; Popov, Konstantin I

Conserved Filovirus Proteins as Targets of Broad-Spectrum Antivirals

保守的丝状病毒蛋白作为广谱抗病毒药物的靶点

Scotti, Marcus Tullius; Kelestemur, Enes; Martin, Holli-Joi; Novy, Brandon; Melo-Filho, Cleber C; de Menezes, Renata Priscila Barros; Herrera-Acevedo, Chonny; Tropsha, Alexander; Muratov, Eugene N

DNAJC13 localization to endosomes is opposed by its J domain and its disordered C-terminal tail.

DNAJC13 定位于内体受到其 J 结构域和无序 C 端尾部的阻碍

Adoff Hayden, Novy Brandon, Holland Emily, Lobingier Braden T