日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

N-Aryl-N-Lactosylamides as Potent and Highly Selective Inhibitors of Galectin-3 with Antifibrotic Activity

N-芳基-N-乳糖酰胺类化合物作为强效且高选择性的半乳糖凝集素-3抑制剂,具有抗纤维化活性

Zýka, Jakub; Kozák, Jaroslav; Vanekova, Lenka; Pimkova Polidarova, Marketa; Prouza, Vít; Habanová, Nina; Strmeň, Timotej; Zavřel, Martin; Pachl, Petr; Choutka, Jan; Grantz Saskova, Klara; Brazdova, Andrea; Parkan, Kamil; Pohl, Radek

Remaining Challenges in the Treatment of Relapsed Wilms Tumor: Children's Oncology Group and International Society of Paediatric Oncology Perspectives

复发性肾母细胞瘤治疗中仍存在的挑战:儿童肿瘤协作组和国际儿科肿瘤学会的观点

Sutton, Kathryn S; Walz, Amy L; Groenendijk, Alissa; Murphy, Andrew J; Pater, Luke; Janssens, Geert O; Brzezinski, Jack; Mullen, Elizabeth A; Spreafico, Filippo; Godzinski, Jan; van der Beek, Justine; Hwa Wijnen, Marc; van den Heuvel-Eibrink, Marry M; Pachl, Max; Graf, Norbert; Ehrlich, Peter F; Furtwangler, Rhoikos; Brok, Jesper; Geller, James

Current surgical approaches to pediatric renal tumors

目前儿童肾脏肿瘤的外科治疗方法

Glick, Richard D; Romao, Rodrigo L P; Pachl, Max; Kotagal, Meera; Buchanan, Amanda F; Murphy, Andrew J; Tracy, Elisabeth T; Pio, Luca; Cost, Nicholas G; Godzinski, Jan; Ehrlich, Peter F

Structural characterization of two prototypical repressors of SorC family reveals tetrameric assemblies on DNA and mechanism of function

SorC 家族两种原型阻遏物的结构表征揭示了 DNA 上的四聚体组装及其功能机制

Markéta Šoltysová, Jana Škerlová, Petr Pachl, Karel Škubník, Milan Fábry, Irena Sieglová, Martina Farolfi, Irina Grishkovskaya, Michal Babiak, Jiří Nováček, Libor Krásný, Pavlína Řezáčová

Targeted protein degradation using chimeric human E2 ubiquitin-conjugating enzymes

使用嵌合人类 E2 泛素结合酶进行靶向蛋白质降解

Jonathan D Taylor, Nathalie Barrett, Sergio Martinez Cuesta, Katelyn Cassidy, Fiona Pachl, James Dodgson, Radhika Patel, Tuula M Eriksson, Aidan Riley, Matthew Burrell, Christin Bauer, D Gareth Rees, Raffaello Cimbro, Andrew X Zhang, Ralph R Minter, James Hunt, Sandrine Legg

Evaluating Antimalarial Proteasome Inhibitors for Efficacy in Babesia Blood Stage Cultures

评估抗疟蛋白酶体抑制剂对巴贝斯虫血液阶段培养物的疗效

Luïse Robbertse, Pavla Fajtová, Pavla Šnebergerová, Marie Jalovecká, Viktoriya Levytska, Elany Barbosa da Silva, Vandna Sharma, Petr Pachl, Jehad Almaliti, Momen Al-Hindy, William H Gerwick, Evžen Bouřa, Anthony J O'Donoghue, Daniel Sojka

Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors

新型嘌呤核苷磷酸化酶抑制剂的设计、合成、生物学评价及晶体学研究

Jan Skácel, Stefan Djukic, Ondřej Baszczyňski, Filip Kalčic, Tadeáš Bílek, Karel Chalupský, Jaroslav Kozák, Alexandra Dvořáková, Eva Tloušt'ová, Zuzana Král'ová, Markéta Šmídková, Jan Voldřich, Michaela Rumlová, Petr Pachl, Jiří Brynda, Tereza Vučková, Milan Fábry, Jan Snášel, Iva Pichová, Pavlína Ř

Proteomics reveals antiviral host response and NETosis during acute COVID-19 in high-risk patients

蛋白质组学揭示高危患者急性 COVID-19 期间的抗病毒宿主反应和 NETosis

Bauer, Alina; Pachl, Elisabeth; Hellmuth, Johannes C; Kneidinger, Nikolaus; Heydarian, Motaharehsadat; Frankenberger, Marion; Stubbe, Hans C; Ryffel, Bernhard; Petrera, Agnese; Hauck, Stefanie M; Behr, Jürgen; Kaiser, Rainer; Scherer, Clemens; Deng, Li; Teupser, Daniel; Ahmidi, Narges; Muenchhoff, Maximilian; Schubert, Benjamin; Hilgendorff, Anne

mRNA display reveals a class of high-affinity bromodomain-binding motifs that are not found in the human proteome

mRNA 展示揭示了一类在人类蛋白质组中未发现的高亲和力溴结构域结合基序

Jason K K Low, Karishma Patel, Natasha Jones, Paul Solomon, Alexander Norman, Joshua W C Maxwell, Petr Pachl, Jacqueline M Matthews, Richard J Payne, Toby Passioura, Hiroaki Suga, Louise J Walport, Joel P Mackay

An evolutionary molecular adaptation of an unusual stefin from the liver fluke Fasciola hepatica redefines the cystatin superfamily

肝吸虫肝片吸虫中一种不寻常的胱抑素的进化分子适应性重新定义了胱抑素超家族

Michal Buša, Zuzana Matoušková, Pavla Bartošová-Sojková, Petr Pachl, Pavlína Řezáčová, Ramon Marc Eichenberger, Peter Deplazes, Martin Horn, Saša Štefanić, Michael Mareš