日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Age of Puberty Onset among Healthy Schoolgirls in North Karnataka: A Cross Sectional Study

北卡纳塔克邦健康女学生青春期开始年龄:一项横断面研究

Kotla, Sruthi; Ghatnatti, Vikrant; Narsannavar, Ashwini; Goroshi, Manjunath; Ganakumar, Vanishri; Paricharak, Pritish P; Venkateswarlu, Damacharlla

Data-driven approaches used for compound library design, hit triage and bioactivity modeling in high-throughput screening

高通量筛选中用于化合物库设计、先导化合物筛选和生物活性建模的数据驱动方法

Paricharak, Shardul; Méndez-Lucio, Oscar; Chavan Ravindranath, Aakash; Bender, Andreas; IJzerman, Adriaan P; van Westen, Gerard J P

Novel Adamantanyl-Based Thiadiazolyl Pyrazoles Targeting EGFR in Triple-Negative Breast Cancer

新型金刚烷基噻二唑吡唑类药物靶向治疗三阴性乳腺癌中的 EGFR

Anusha Sebastian, Vijay Pandey, Chakrabhavi Dhananjaya Mohan, Yi Ting Chia, Shobith Rangappa, Jessin Mathai, C P Baburajeev, Shardul Paricharak, Lewis H Mervin, Krishna C Bulusu, Julian E Fuchs, Andreas Bender, Shuhei Yamada, Basappa, Peter E Lobie, Kanchugarakoppal S Rangappa

Trisubstituted-Imidazoles Induce Apoptosis in Human Breast Cancer Cells by Targeting the Oncogenic PI3K/Akt/mTOR Signaling Pathway

三取代咪唑通过靶向致癌 PI3K/Akt/mTOR 信号通路诱导人类乳腺癌细胞凋亡

Chakrabhavi Dhananjaya Mohan, V Srinivasa, Shobith Rangappa, Lewis Mervin, Surender Mohan, Shardul Paricharak, Sefer Baday, Feng Li, Muthu K Shanmugam, Arunachalam Chinnathambi, M E Zayed, Sulaiman Ali Alharbi, Andreas Bender, Gautam Sethi, Basappa, Kanchugarakoppal S Rangappa

Proteochemometric modelling coupled to in silico target prediction: an integrated approach for the simultaneous prediction of polypharmacology and binding affinity/potency of small molecules

蛋白质化学计量学建模与计算机靶点预测相结合:一种用于同时预测小分子多药理学和结合亲和力/效力的综合方法

Paricharak, Shardul; Cortés-Ciriano, Isidro; IJzerman, Adriaan P; Malliavin, Thérèse E; Bender, Andreas

A Nano-MgO and Ionic Liquid-Catalyzed 'Green' Synthesis Protocol for the Development of Adamantyl-Imidazolo-Thiadiazoles as Anti-Tuberculosis Agents Targeting Sterol 14α-Demethylase (CYP51)

一种以纳米氧化镁和离子液体为催化剂的“绿色”合成方案,用于开发靶向甾醇14α-去甲基酶(CYP51)的金刚烷基咪唑并噻二唑类抗结核药物

Anusha, Sebastian; Cp, Baburajeev; Mohan, Chakrabhavi Dhananjaya; Mathai, Jessin; Rangappa, Shobith; Mohan, Surender; Chandra; Paricharak, Shardul; Mervin, Lewis; Fuchs, Julian E; M, Mahedra; Bender, Andreas; Basappa; Rangappa, Kanchugarakoppal S

Novel benzoxazine-based aglycones block glucose uptake in vivo by inhibiting glycosidases

新型苯并恶嗪类糖苷配基通过抑制糖苷酶来阻止体内葡萄糖的吸收

Hanumantharayappa Bharathkumar, Mahalingam S Sundaram, Swamy Jagadish, Shardul Paricharak, Mahadevappa Hemshekhar, Daniel Mason, Kempaiah Kemparaju, Kesturu S Girish, Basappa, Andreas Bender, Kanchugarakoppal S Rangappa

Histopathological study of skin adnexal tumours-institutional study in South India

皮肤附属器肿瘤的组织病理学研究——南印度机构研究

Sharma, Ankit; Paricharak, Deepak G; Nigam, Jitendra Singh; Rewri, Shivani; Soni, Priyanka Bhatia; Omhare, Anita; Sekar, Preethi