日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery and Characterization of Divarasib (GDC-6036), a Potent Covalent Inhibitor of KRAS G12C.

Divarasib (GDC-6036) 的发现和表征,一种强效的 KRAS G12C 共价抑制剂。

Endres Nicholas F, Do Steven, Mroue Rana, Terrett Jack A, Saabye Matt, Oh Angela, Hunsaker Thomas, Chan Emily, Tran John C, Nguyen Lan K, Lian Qihui, Ma Taylur P, Garner Thomas, Gerosa Luca, Beresini Maureen, Boudreau Aaron, Bronner Sarah M, Cyr Patrick, Ishisoko Noriko, Izrayelit Yevgeniy, Jiang Fan, Kellar Terry, La Hank, Labadie Sharada, Lardy Matthew, Liu Liling, Liu Wendy, Miller Sarah, Rudolph Joachim, Plise Emile, Sellers Benjamin D, Shao Cheng, Wang Weiru, Wang Yanguang, Wei Wentao, Wong Susan, Yu Christine, Yu Kebing, Yuen Po-Wai, Zang Richard, Zhang Chenghong, Zhou Yuhui, Zhu Xiaoyu, Quinn John G, Ye Xin, Kiefer James R, Mao Jialin, Evangelista Marie, Merchant Mark, Landry Matthew L, Malhotra Sushant, Purkey Hans E

The potential of H5N1 viruses to adapt to bovine cells varies throughout evolution

H5N1病毒适应牛细胞的能力在进化过程中不断变化

Turnbull, Matthew L; Zakaria, Mohammad Khalid; Upfold, Nicole S; Bakshi, Siddharth; Magill, Callum; Das, Udeet Ranjan; Clarke, Andrew T; Mojsiejczuk, Laura; Herder, Vanessa; Dee, Kieran; Liu, Nancy; Folwarczna, Monika; Ilia, Georgios; Furnon, Wilhelm; Schultz, Verena; Chen, Hanting; Devlin, Ryan; McCowan, Jack; Young, Alex L; Po, Wai-Wai; Smollett, Katherine; Yaseen, Muhammad Ahsan; Ross, Rebecca; Bhide, Avanti; van Kekem, Bianca; Fouchier, Ron A M; da Silva Filipe, Ana; Iqbal, Munir; Roberts, Ed; Hughes, Joseph; Werling, Dirk; Murcia, Pablo R; Palmarini, Massimo

Enhanced Specificity in Colorimetric LAMP Assay for Sarocladium kiliense Detection Using a Combination of Two Additives

两种添加剂组合提高比色LAMP检测中Sarocladium kiliense的特异性

Wong, Yu-Ning; Hau, Pak-Ting; Chau, Eddie Chung-Ting; Ng, Laam-Ching; Murillo, Michaela; Fung, Joshua; Po, Wai-Wai; Yu, Ray Chun-Wai; Kam, Melody Kai-Ting; Tam, Emily Wan-Ting; Tsang, Chi-Ching; Chow, Franklin Wang-Ngai

Post-injury administration of NAAG peptidase inhibitor prodrug, PGI-02776, in experimental TBI

在实验性创伤性脑损伤中,损伤后给予NAAG肽酶抑制剂前药PGI-02776

Feng, Jun-Feng; Van, Ken C; Gurkoff, Gene G; Kopriva, Christina; Olszewski, Rafal T; Song, Minsoo; Sun, Shifeng; Xu, Man; Neale, Joseph H; Yuen, Po-Wai; Lowe, David A; Zhou, Jia; Lyeth, Bruce G

Chemistry and pharmacology of nicotinic ligands based on 6-[5-(azetidin-2-ylmethoxy)pyridin-3-yl]hex-5-yn-1-ol (AMOP-H-OH) for possible use in depression

基于 6-[5-(氮杂环丁烷-2-基甲氧基)吡啶-3-基]己-5-炔-1-醇 (AMOP-H-OH) 的尼古丁配体的化学和药理学研究及其在抑郁症治疗中的潜在应用

Kozikowski, Alan P; Eaton, J Brek; Bajjuri, Krishna Mohan; Chellappan, Sheela K; Chen, Yihua; Karadi, Sudhakar; He, Rong; Caldarone, Barbara; Manzano, Michael; Yuen, Po-Wai; Lukas, Ronald J