日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A novel DNA sequence-selective, guanine mono-alkylating ADC payload suitable for solid tumour treatment

一种新型的DNA序列选择性鸟嘌呤单烷基化抗体药物偶联物(ADC)有效载荷,适用于实体瘤治疗。

Andriollo, Paolo; di Mascio, Daniella; Jackson, Paul J M; Hasan, Md Mahbub; Pysz-Hosey, Ilona; Procopiou, George; Fox, Keith R; Rahman, Khondaker Miraz; Thurston, David E

Detection of Virulence-Associated Genes among Brucella melitensis and Brucella abortus Clinical Isolates in Greece, 2001-2022

2001-2022年希腊布鲁氏菌(羊布鲁氏菌和牛布鲁氏菌)临床分离株毒力相关基因的检测

Papaparaskevas, Joseph; Procopiou, Alexandra; Routsias, John; Vrioni, Georgia; Tsakris, Athanasios

A Perspective on the Influence of National Corporate Governance Institutions and Government's Political Ideology on the Speed to Lockdown as a Means of Protection Against Covid-19

国家公司治理制度和政府政治意识形态对采取封锁措施速度以应对新冠肺炎疫情的影响分析

Chow, Dawn Yi Lin; Petrou, Andreas; Procopiou, Andreas

DNA sequence-selective G-A cross-linking ADC payloads for use in solid tumour therapies

DNA 序列选择性 GA 交联 ADC 有效载荷用于实体肿瘤治疗

George Procopiou, Paul J M Jackson, Daniella di Mascio, Jennifer L Auer, Chris Pepper, Khondaker Miraz Rahman, Keith R Fox, David E Thurston

Oncocytic Adrenocortical Neoplasm with Concomitant Papillary Thyroid Cancer

伴有乳头状甲状腺癌的嗜酸性肾上腺皮质肿瘤

Podetta, Michele; Pusztaszeri, Marc; Toso, Christian; Procopiou, Michel; Triponez, Frédéric; Sadowski, Samira Mercedes

Short and efficient syntheses of protoberberine alkaloids using palladium-catalyzed enolate arylation

利用钯催化烯醇化物芳基化反应高效简便地合成原小檗碱生物碱

Gatland, Alice E; Pilgrim, Ben S; Procopiou, Panayiotis A; Donohoe, Timothy J

Synthetic Studies Towards the Core Structure of Nakadomarin A by a Thioamide-Based Strategy

基于硫酰胺策略的合成研究:Nakadomarin A核心结构的构建

Chavda, Jai K; Procopiou, Panayiotis A; Horton, Peter N; Coles, Simon J; Porter, Michael J

Modular isoquinoline synthesis using catalytic enolate arylation and in situ functionalization

利用催化烯醇化芳基化和原位官能化进行模块化异喹啉合成

Pilgrim, Ben S; Gatland, Alice E; McTernan, Charlie T; Procopiou, Panayiotis A; Donohoe, Timothy J

Lead optimisation of the N1 substituent of a novel series of indazole arylsulfonamides as CCR4 antagonists and identification of a candidate for clinical investigation

对一系列新型吲唑芳基磺酰胺的 N1 取代基进行优化,将其作为 CCR4 拮抗剂,并确定临床研究候选药物

Panayiotis A Procopiou, Alison J Ford, Rebecca H Graves, David A Hall, Simon T Hodgson, Yannick M L Lacroix, Deborah Needham, Robert J Slack

Heavier Group‐2‐Element Catalyzed Hydroamination of Carbodiimides

较重的第2族元素催化碳二亚胺的氢胺化反应

Xie, Wensheng; Zhang, Genpei; Guo, Zhenhu; Huang, Hongye; Ye, Jielin; Gao, Xiaohan; Yue, Kai; Wei, Yen; Zhao, Lingyun; Lachs, Jennifer R; Barrett, Anthony G M; Crimmin, Mark R; Kociok‐Köhn, Gabriele; Hill, Michael S; Mahon, Mary F; Procopiou, Panayiotis A