日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hydrogen Sulfide (H(2)S)-Donating Formyl Peptide Receptor 2 (FPR2) Agonists: Design, Synthesis, and Biological Evaluation in Primary Mouse Microglia Culture.

硫化氢 (H(2)S) 供体甲酰肽受体 2 (FPR2) 激动剂:设计、合成和在原代小鼠小胶质细胞培养中的生物学评价

Brunetti Leonardo, Francavilla Fabio, Niso Mauro, Frydrych Jakub Kosma, Trojan Ewa, Schepetkin Igor A, Kirpotina Liliya N, Grygier Beata, Łukowicz Krzysztof, Quinn Mark T, Basta-Kaim Agnieszka, Lacivita Enza, Leopoldo Marcello

Tricyclic Isatin Derivatives as Anti-Inflammatory Compounds with High Kinase Binding Affinity

三环靛红衍生物作为具有高激酶结合亲和力的抗炎化合物

Uvarov, Alexander V; Schepetkin, Igor A; Quinn, Mark T; Khlebnikov, Andrei I

c-Jun N-Terminal Kinase (JNK) Inhibitor IQ-1S as a Suppressor of Tumor Spheroid Growth

c-Jun N 端激酶 (JNK) 抑制剂 IQ-1S 作为肿瘤球体生长的抑制因子

Afrimzon, Elena; Deutsch, Mordechai; Sobolev, Maria; Zurgil, Naomi; Khlebnikov, Andrei I; Buldakov, Mikhail A; Schepetkin, Igor A

Regulation of Blood-Brain Barrier Permeability via JNK Signaling Pathway: Mechanisms and Potential Therapeutic Strategies for Ischemic Stroke, Alzheimer's Disease and Brain Tumors

JNK信号通路调控血脑屏障通透性:缺血性卒中、阿尔茨海默病和脑肿瘤的机制及潜在治疗策略

Plotnikov, Mark B; Anishchenko, Anna M; Khlebnikov, Andrei I; Schepetkin, Igor A

Activity-Based Profiling of Papain-like Cysteine Proteases During Late-Stage Leaf Senescence in Barley

大麦叶片衰老后期木瓜蛋白酶样半胱氨酸蛋白酶的活性分析

Schepetkin, Igor A; Fischer, Andreas M

Design, Synthesis, and Biological Evaluation of Novel Heteroaryl, Squaramide, and Indolcarboxamide Derivatives as Formyl Peptide Receptor 2 Agonists to Target Neuroinflammation

设计、合成和生物学评价新型杂芳基、方酰胺和吲哚甲酰胺衍生物作为甲酰肽受体2激动剂靶向治疗神经炎症

Francavilla, Fabio; Vitone, Daniele; Schepetkin, Igor A; Kirpotina, Lilya N; Carrieri, Antonio; Brunetti, Leonardo; Ghafir El Idrissi, Imane; Perrone, Maria Grazia; Frydrych, Jakub Kosma; Trojan, Ewa; Quinn, Mark T; Basta-Kaim, Agnieszka; Lacivita, Enza; Leopoldo, Marcello

Evaluation of Nitric Oxide-Donating Properties of 11H-indeno[1,2-b]quinoxalin-11-one Oxime (IQ-1) by Electron Paramagnetic Resonance Spectroscopy

利用电子顺磁共振波谱法评价11H-茚并[1,2-b]喹喔啉-11-酮肟(IQ-1)的氧化氮供体性质

Andrianov, Viacheslav V; Schepetkin, Igor A; Bazan, Leah V; Gainutdinov, Khalil L; Kovrizhina, Anastasia R; Atochin, Dmitriy N; Khlebnikov, Andrei I

Phytochemical Composition and Biological Activity of the Essential Oil from Ericameria nauseosa Collected in Southwestern Montana, United States

美国蒙大拿州西南部采集的埃里克梅利亚·纳塞奥萨(Ericameria nauseosa)精油的植物化学成分和生物活性

Schepetkin, Igor A; Özek, Gulmira; Özek, Temel; Kirpotina, Liliya N; Khlebnikov, Andrei I; Ayçiçek, Kevser; Lavin, Matthew; Quinn, Mark T

Cathepsin B- and L-like Protease Activities Are Induced During Developmental Barley Leaf Senescence.

大麦叶片发育衰老过程中,组织蛋白酶 B 和 L 样蛋白酶活性被诱导

Schepetkin Igor A, Fischer Andreas M

Neuroprotective Effects of Tryptanthrin-6-Oxime in a Rat Model of Transient Focal Cerebral Ischemia

色胺酮-6-肟在大鼠短暂性局灶性脑缺血模型中的神经保护作用

Plotnikov, Mark B; Chernysheva, Galina A; Smol'yakova, Vera I; Aliev, Oleg I; Anishchenko, Anna M; Ulyakhina, Olga A; Trofimova, Eugene S; Ligacheva, Anastasia A; Anfinogenova, Nina D; Osipenko, Anton N; Kovrizhina, Anastasia R; Khlebnikov, Andrei I; Schepetkin, Igor A; Drozd, Anastasia G; Plotnikov, Evgenii V; Atochin, Dmitriy N; Quinn, Mark T