日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Publisher Correction: Mutant p53 protein accumulation is selectively targetable by proximity-inducing drugs

出版商更正:突变型p53蛋白的积累可被邻近诱导药物选择性靶向。

Sadagopan, Ananthan; Carson, Maximilian; Zamurs, Eriks J; Garaffo, Nicholas; Chang, Heng-Jui; Schreiber, Stuart L; Meyerson, Matthew; Gibson, William J

Mutant p53 protein accumulation is selectively targetable by proximity-inducing drugs

突变型p53蛋白的积累可被邻近诱导药物选择性地靶向。

Sadagopan, Ananthan; Carson, Maximilian; Zamurs, Eriks J; Garaffo, Nicholas; Chang, Heng-Jui; Schreiber, Stuart L; Meyerson, Matthew; Gibson, William J

Highly specific intracellular ubiquitination of a small molecule.

小分子的高度特异性细胞内泛素化。

Li Weicheng, Garcia-Rivera Enrique M, Mitchell Dylan C, Chick Joel M, Maetani Micah, Bhadoria Rohit, Knapp John M, Misu Ryosuke, Matthews Geoffrey M, Shirasaki Ryosuke, de Matos Simoes Ricardo, Viswanathan Vasanthi, Pulice John L, Rees Matthew G, Roth Jennifer A, Gygi Steven P, Mitsiades Constantine S, Kadoch Cigall, Schreiber Stuart L, Ostrem Jonathan M L

The Ulcerative Colitis-Associated Gene NXPE1 Catalyzes Glycan Modifications on Colonic Mucin.

溃疡性结肠炎相关基因 NXPE1 催化结肠粘蛋白的糖基化修饰

Humeidi Ranad, Oshiro-Rapley Noriko, Gu Xiebin, An Joon Soo, Ananthakrishnan Ashwin N, Creasey Elizabeth A, Daly Mark J, Schreiber Stuart L, Graham Daniel B, Seyedsayamdost Mohammad R, Xavier Ramnik J

Development of an FKBP12-recruiting chemical-induced proximity DNA-encoded library and its application to discover an autophagy potentiator.

开发 FKBP12 募集化学诱导邻近 DNA 编码文库及其在发现自噬增强剂中的应用

Tan Zher Yin, Adade Joel K A, Gu Xiebin, Hecht Cody J S, Salcius Michael, Tong Bingqi, Liu Shuang, Hwang Seungmin, Zécri Frédéric J, Graham Daniel B, Schreiber Stuart L, Xavier Ramnik J

Systematic in vitro evolution in Plasmodium falciparum reveals key determinants of drug resistance.

恶性疟原虫体外系统进化揭示了耐药性的关键决定因素

Luth Madeline R, Godinez-Macias Karla P, Chen Daisy, Okombo John, Thathy Vandana, Cheng Xiu, Daggupati Sindhu, Davies Heledd, Dhingra Satish K, Economy Jan M, Edgar Rebecca C S, Gomez-Lorenzo Maria G, Istvan Eva S, Jado Juan Carlos, LaMonte Gregory M, Melillo Bruno, Mok Sachel, Narwal Sunil K, Ndiaye Tolla, Ottilie Sabine, Palomo Diaz Sara, Park Heekuk, Peña Stella, Rocamora Frances, Sakata-Kato Tomoyo, Small-Saunders Jennifer L, Summers Robert L, Tumwebaze Patrick K, Vanaerschot Manu, Xia Guoqin, Yeo Tomas, You Ashley, Gamo Francisco-Javier, Goldberg Daniel E, Lee Marcus C S, McNamara Case W, Ndiaye Daouda, Rosenthal Philip J, Schreiber Stuart L, Serra Gloria, De Siqueira-Neto Jair Lage, Skinner-Adams Tina S, Uhlemann Anne-Catrin, Kato Nobutaka, Lukens Amanda K, Wirth Dyann F, Fidock David A, Winzeler Elizabeth A

Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders

螺环丙烯酰胺立体探针的蛋白质组学配体结合能力图谱鉴定共价ERCC3降解剂

Liu, Zhonglin; Remsberg, Jarrett R; Li, Haoxin; Njomen, Evert; DeMeester, Kristen E; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M; Schreiber, Stuart L; Melillo, Bruno; Cravatt, Benjamin F

Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes.

扩展可配体结合蛋白质组的化学工具:基于多样性的合成的光反应立体探针

Ogasawara Daisuke, Konrad David B, Tan Zher Yin, Carey Kimberly L, Luo Jessica, Won Sang Joon, Li Haoxin, Carter Trever R, DeMeester Kristen E, Njomen Evert, Schreiber Stuart L, Xavier Ramnik J, Melillo Bruno, Cravatt Benjamin F

Bicyclic Pyrrolidine Inhibitors of Toxoplasma gondii Phenylalanine t-RNA Synthetase with Antiparasitic Potency In Vitro and Brain Exposure

体外和脑暴露中具有抗寄生虫效力的弓形虫苯丙氨酸tRNA合成酶双环吡咯烷抑制剂

Ence, Chloe C; Uddin, Taher; Borrel, Julien; Mittal, Payal; Xie, Han; Zoller, Jochen; Sharma, Amit; Comer, Eamon; Schreiber, Stuart L; Melillo, Bruno; Sibley, L David; Chatterjee, Arnab K

Bicyclic pyrrolidine inhibitors of Toxoplasma gondii phenylalanine t-RNA synthetase with antiparasitic potency in vitro and brain exposure

体外和脑暴露实验表明,双环吡咯烷类弓形虫苯丙氨酸tRNA合成酶抑制剂具有抗寄生虫活性。

Ence, Chloe C; Uddin, Taher; Borrel, Julien; Mittal, Payal; Xie, Han; Zoller, Jochen; Sharma, Amit; Comer, Eamon; Schreiber, Stuart L; Melillo, Bruno; Sibley, L David; Chatterjee, Arnab K