日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MELLODDY: Cross-pharma Federated Learning at Unprecedented Scale Unlocks Benefits in QSAR without Compromising Proprietary Information

MELLODDY:前所未有的跨制药公司联邦学习规模释放了QSAR的优势,且不泄露专有信息

Heyndrickx, Wouter; Mervin, Lewis; Morawietz, Tobias; Sturm, Noé; Friedrich, Lukas; Zalewski, Adam; Pentina, Anastasia; Humbeck, Lina; Oldenhof, Martijn; Niwayama, Ritsuya; Schmidtke, Peter; Fechner, Nikolas; Simm, Jaak; Arany, Adam; Drizard, Nicolas; Jabal, Rama; Afanasyeva, Arina; Loeb, Regis; Verma, Shlok; Harnqvist, Simon; Holmes, Matthew; Pejo, Balazs; Telenczuk, Maria; Holway, Nicholas; Dieckmann, Arne; Rieke, Nicola; Zumsande, Friederike; Clevert, Djork-Arné; Krug, Michael; Luscombe, Christopher; Green, Darren; Ertl, Peter; Antal, Peter; Marcus, David; Do Huu, Nicolas; Fuji, Hideyoshi; Pickett, Stephen; Acs, Gergely; Boniface, Eric; Beck, Bernd; Sun, Yax; Gohier, Arnaud; Rippmann, Friedrich; Engkvist, Ola; Göller, Andreas H; Moreau, Yves; Galtier, Mathieu N; Schuffenhauer, Ansgar; Ceulemans, Hugo

Discovery of New Binders for DCAF1, an Emerging Ligase Target in the Targeted Protein Degradation Field

在靶向蛋白降解领域,发现了一种新兴的连接酶靶点——DCAF1 的新型结合剂。

Vulpetti, Anna; Holzer, Philipp; Schmiedeberg, Niko; Imbach-Weese, Patricia; Pissot-Soldermann, Carole; Hollingworth, Gregory J; Radimerski, Thomas; Thoma, Claudio R; Stachyra, Therese-Marie; Wojtynek, Matthias; Maschlej, Magdalena; Chau, Suzanne; Schuffenhauer, Ansgar; Fernández, César; Schröder, Martin; Renatus, Martin

Retrospective evaluation of early thrombosis in transjugular intrahepatic portosystemic polytetrafluoroethylene-coated shunts under 2-day postinterventional heparinization

回顾性评估经颈静脉肝内门体分流术(TIPS)聚四氟乙烯涂层分流术后2天肝素化治疗中早期血栓形成的情况

Goessmann, Holger; Schuffenhauer, Verna; Kandulski, Arne; Weigand, Kilian; Jung, Ernst-Michael; Uller, Wibke; Scharf, Gregor; Stroszczynski, Cristian; Verloh, Niklas

Gene-signature-derived IC50s/EC50s reflect the potency of causative upstream targets and downstream phenotypes

基因特征衍生的 IC50/EC50 反映了致病上游靶点和下游表型的效力

Steffen Renner, Christian Bergsdorf, Rochdi Bouhelal, Magdalena Koziczak-Holbro, Andrea Marco Amati, Valerie Techer-Etienne, Ludivine Flotte, Nicole Reymann, Karen Kapur, Sebastian Hoersch, Edward James Oakeley, Ansgar Schuffenhauer, Hanspeter Gubler, Eugen Lounkine, Pierre Farmer

A Multi-Pumping Flow System for In Situ Measurements of Dissolved Manganese in Aquatic Systems

用于原位测量水生系统中溶解锰的多泵流量系统

Meyer, David; Prien, Ralf D; Dellwig, Olaf; Waniek, Joanna J; Schuffenhauer, Ingo; Donath, Jan; Krüger, Siegfried; Pallentin, Malte; Schulz-Bull, Detlef E

Estimation of synthetic accessibility score of drug-like molecules based on molecular complexity and fragment contributions

基于分子复杂性和片段贡献的类药分子合成可及性评分估算

Ertl, Peter; Schuffenhauer, Ansgar

BIOS: Similarity-based design of natural product derived compound collections

BIOS:基于相似性的天然产物衍生化合物库设计

Reddy, D V Subba; Wetzel, S; Renner, S; Nören-Müller, A; Schuffenhauer, A; Ertl, P; Waldmann, Herbert

Charting biologically relevant chemical space: a structural classification of natural products (SCONP)

绘制生物学相关化学空间图:天然产物的结构分类(SCONP)

Koch, Marcus A; Schuffenhauer, Ansgar; Scheck, Michael; Wetzel, Stefan; Casaulta, Marco; Odermatt, Alex; Ertl, Peter; Waldmann, Herbert

An optimized probe set for the detection of small interchromosomal aberrations by use of 24-color FISH

一种用于通过24色FISH检测小型染色体间畸变的优化探针组

Azofeifa, J; Fauth, C; Kraus, J; Maierhofer, C; Langer, S; Bolzer, A; Reichman, J; Schuffenhauer, S; Speicher, M R

Parental origin and mechanisms of formation of cytogenetically recognisable de novo direct and inverted duplications

亲本来源和细胞遗传学上可识别的新生直接和反向重复的形成机制

Kotzot, D; Martinez, M J; Bagci, G; Basaran, S; Baumer, A; Binkert, F; Brecevic, L; Castellan, C; Chrzanowska, K; Dutly, F; Gutkowska, A; Karaüzüm, S B; Krajewska-Walasek, M; Luleci, G; Miny, P; Riegel, M; Schuffenhauer, S; Seidel, H; Schinzel, A