日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In silico docking yields small molecule negative allosteric modulators targeting the core of Frizzled 7

计算机模拟对接筛选出靶向Frizzled 7核心的小分子负变构调节剂。

Scharf, Magdalena M; Kinsolving, Julia; Grätz, Lukas; Voss, Jan Hendrik; Carrasco-Busturia, David; Forsberg, Björn; Kolb, Peter; Schulte, Gunnar

WNT-induced association of Frizzled and LRP6 is not sufficient for the initiation of WNT/β-catenin signaling.

WNT 诱导的 Frizzled 和 LRP6 的结合不足以启动 WNT/β-catenin 信号传导

Voss Jan Hendrik, Koszegi Zsombor, Yan Yining, Shorter Emily, Grätz Lukas, Lanner Johanna T, Calebiro Davide, Schulte Gunnar

Inactive structures of the vasopressin V2 receptor reveal distinct binding modes for Tolvaptan and Mambaquaretin toxin.

血管加压素 V2 受体的非活性结构揭示了托伐普坦和曼巴奎汀毒素的不同结合模式

Fouillen Aurélien, Bous Julien, Couvineau Pierre, Orcel Hélène, Mary Charline, Lafleur Lucie, Pierre Timothé, Mendre Christiane, Gilles Nicolas, Schulte Gunnar, Granier Sébastien, Mouillac Bernard

SAG1.3-derived Frizzled-targeting small-molecule compounds.

源自 SAG1.3 的 Frizzled 靶向小分子化合物。

Grätz Lukas, Turku Ainoleena, Kozielewicz Pawel, Bowin Carl-Fredrik, Scharf Magdalena M, Voss Jan H, Kinsolving Julia, Shekhani Rawan, Oliva-Vilarnau Nuria, Koolmeister Tobias, Körber Marlies, Lauschke Volker M, Löber Stefan, Gmeiner Peter, Schulte Gunnar

Complex G-protein signaling of the adhesion GPCR, ADGRA3.

粘附 GPCR ADGRA3 的复杂 G 蛋白信号传导

Bagger Sofie M, Schihada Hannes, Walser Anna L S, Drzazga Anna K, Grätz Lukas, Palmisano Tiago, Kuhn Christina K, Mavri Maša, Mølleskov-Jensen Ann-Sophie, Tall Gregory G, Schöneberg Torsten, Mathiasen Signe J, Javitch Jonathan A, Schulte Gunnar, Spiess Katja, Rosenkilde Mette M

Wnt-3a Induces Cytokine Release in Human Mast Cells

Wnt-3a诱导人肥大细胞释放细胞因子

Julia Tebroke ,Joris E Lieverse ,Jesper Säfholm ,Gunnar Schulte ,Gunnar Nilsson ,Elin Rönnberg

WNT signalling: mechanisms and therapeutic opportunities

WNT信号通路:机制和治疗机遇

Schulte, Gunnar; Bryja, Vitezslav

WNT Stimulation Dissociates a Frizzled 4 Inactive-State Complex with Gα12/13

WNT刺激使Frizzled 4非活性状态复合物与Gα12/13解离

Arthofer, Elisa; Hot, Belma; Petersen, Julian; Strakova, Katerina; Jäger, Stefan; Grundmann, Manuel; Kostenis, Evi; Gutkind, J Silvio; Schulte, Gunnar

WNT signaling in microglia and the glioma microenvironment

小胶质细胞和胶质瘤微环境中的WNT信号通路

Schulte, Gunnar

Molecular reorganization of endocannabinoid signalling in Alzheimer's disease

阿尔茨海默病中内源性大麻素信号传导的分子重组

Mulder, Jan; Zilberter, Misha; Pasquaré, Susana J; Alpár, Alán; Schulte, Gunnar; Ferreira, Samira G; Köfalvi, Attila; Martín-Moreno, Ana M; Keimpema, Erik; Tanila, Heikki; Watanabe, Masahiko; Mackie, Ken; Hortobágyi, Tibor; de Ceballos, Maria L; Harkany, Tibor