日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Antifungal activity of oily core PEGylated PLGA nanocapsules loaded with Penicillium oxalicum fungal extract: in vitro, in vivo, and in silico study

负载草酸青霉菌提取物的油性核聚乙二醇化PLGA纳米胶囊的抗真菌活性:体外、体内和计算机模拟研究

Elekhnawy, Engy; Abdelkader, Dalia H; Eliwa, Duaa; Ibrahim, Sarah; Shaldam, Moataz A; Negm, Walaa A

Discovery of potent bisindole-based pyrazolopyridine derivatives as topoisomerase inhibitors: DNA damage induction and synergistic antileukemic activity

发现强效的基于双吲哚的吡唑并吡啶衍生物作为拓扑异构酶抑制剂:DNA损伤诱导和协同抗白血病活性

Eldehna, Wagdy M; Tawfik, Haytham O; Veselá, Denisa; Peřina, Miroslav; Negmeldin, Ahmed T; Elsayed, Zainab M; Majrashi, Taghreed A; Vojáčková, Veronika; Elbadawi, Mostafa M; Shaldam, Moataz A; Kryštof, Vladimír; Abdel-Aziz, Hatem A

Exploring the impact of the innovative compound 3-(3-(4-hydroxy-2-oxo-2H-chromen-3-yl)-5-(pyridin-3-yl)-1H-pyrazol-1-yl) indolin-2-one on accelerating wound recovery

探索创新化合物3-(3-(4-羟基-2-氧代-2H-色烯-3-基)-5-(吡啶-3-基)-1H-吡唑-1-基)吲哚啉-2-酮对加速伤口愈合的影响

Sabt, Ahmed; Abdelmegeed, Heba; Abdel-Razik, Abdel-Razik H; Thabit, Mohamed G; Balaha, Marwa; Shaldam, Moataz A; Reda, Ahmed M; Soliman, Ahmed A F; Abdelraof, Mohamed; Abdel Latif, Nehad A; Elghonemy, Mai M; Ahmed, Eman Y; Abdelrahman, Mohamed A; Batran, Rasha Z

Design, synthesis, and molecular modeling of novel thiazolopyridine-based inhibitors of enoyl acyl carrier protein reductase (InhA) as anti-Mycobacterium tuberculosis agents

设计、合成和分子建模新型噻唑并吡啶类烯酰酰基载体蛋白还原酶(InhA)抑制剂作为抗结核分枝杆菌药物

Sabt, Ahmed; Korycka-Machała, Małgorzata; Kassem, Asmaa F; Saleh, Abdulrahman M; Farag, Hanaa; Shaldam, Moataz A; Thabit, Mohamed G; Brzostek, Anna; Kuzioła, Magdalena; Dziadek, Bożena; Ibrahim, Hoda Atef Abdelsattar; Lei, Xinsheng; Dziadek, Jarosław; Abdelrahman, Mohamed A

Targeting Helicobacter pylori enzymes using Viscum album L. extract: in silico molecular docking and in vitro study

利用槲寄生提取物靶向幽门螺杆菌酶:计算机分子对接和体外研究

Cardos, Ioana Alexandra; Danila, Catalina; Yahya, Galal; Seleem, Noura M; Mosbah, Rasha A; Shaldam, Moataz A; Vicas, Simona Ioana; Metwally, Kamel; Cavalu, Simona Daniela

Mechanistic and Molecular Insights into Empagliflozin's Role in Ferroptosis and Inflammation Trajectories in Acetaminophen-Induced Hepatotoxicity.

从机制和分子层面深入了解恩格列净在对乙酰氨基酚诱导的肝毒性中铁死亡和炎症轨迹的作用

Alhaddad Aisha, Mosalam Esraa M, AboShabaan Hind S, Sallam Amany Said, Mahfouz Marwa M, Elhosary Enas, Mohammed Asmaa A, Metwally Ebtehal M, Shaldam Moataz A, Ghoneim Mai El-Sayed

Targeted synthesis of a trimethoxyphenyltetrahydropyrimidine analogue designed as a DNA intercalator: in silico, multi-spectroscopic, thermodynamic, and in vitro approaches

以DNA嵌入剂为设计目标的三甲氧基苯基四氢嘧啶类似物的靶向合成:计算机模拟、多光谱学、热力学和体外方法

Al-Karmalawy, Ahmed A; Elmaaty, Ayman Abo; Magdy, Galal; Radwan, Aya Saad; Alnajjar, Radwan; Shaldam, Moataz A; Al Khatib, Arwa Omar; Almujri, Salem Salman; Abdullah Alzahrani, Abdullah Yahya; Tawfik, Haytham O

Correction: Khayyat et al. Xylitol Inhibits Growth and Blocks Virulence in Serratia marcescens. Microorganisms 2021, 9, 1083

更正:Khayyat 等人,《木糖醇抑制粘质沙雷氏菌的生长并阻断其毒力》,《微生物》2021,9,1083

Khayyat, Ahdab N; Hegazy, Wael A H; Shaldam, Moataz A; Mosbah, Rasha; Almalki, Ahmad J; Ibrahim, Tarek S; Khayat, Maan T; Khafagy, El-Sayed; Soliman, Wafaa E; Abbas, Hisham A

Donepezil-based rational design of N-substituted quinazolinthioacetamide candidates as potential acetylcholine esterase inhibitors for the treatment of Alzheimer's disease: in vitro and in vivo studies

基于多奈哌齐的N-取代喹唑啉硫代乙酰胺类化合物的合理设计:作为治疗阿尔茨海默病的潜在乙酰胆碱酯酶抑制剂:体外和体内研究

Al-Karmalawy, Ahmed A; Mohamed, Ahmed F; Shalaby, Heba Nasr; Elmaaty, Ayman Abo; El-Shiekh, Riham A; Zeidan, Mohamed A; Alnajjar, Radwan; Alzahrani, Abdullah Yahya Abdullah; Al Mughram, Mohammed H; Shaldam, Moataz A; Tawfik, Haytham O

Benzenesulfonohydrazide-tethered non-fused and fused heterocycles as potential anti-mycobacterial agents targeting enoyl acyl carrier protein reductase (InhA) with antibiofilm activity

苯磺酰肼连接的非稠合和稠合杂环化合物作为潜在的抗分枝杆菌药物,靶向烯酰酰基载体蛋白还原酶(InhA),具有抗生物膜活性。

Al-Warhi, Tarfah; Sabt, Ahmed; Korycka-Machala, Małgorzata; Kassem, Asmaa F; Shaldam, Moataz A; Ibrahim, Hoda Atef Abdelsattar; Kawka, Malwina; Dziadek, Bożena; Kuzioła, Magdalena; Eldehna, Wagdy M; Dziadek, Jarosław