日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting cell cycle and apoptotic pathways with newly synthesized diselenide-linked imidazolone analogues with strong CDK6-targeting potential

利用新合成的具有强 CDK6 靶向潜力的二硒化物连接的咪唑酮类似物靶向细胞周期和凋亡通路

Abdel-Motaal, Marwa; Shaaban, Saad; Hawas, Samia S; Elsharif, Asma M; Sharaky, Marwa; Alatawi, Fatema S; Eissa, Mohamed E; Al Khatib, Arwa Omar; Abd El-Lateef, Hany M; Asem, Medhat; Al-Karmalawy, Ahmed A

Hybrid benzylidene thiazolidine-2,4-diones as potent apoptosis-inducing anticancer agents: design-driven optimization, cytotoxic profiling, and mechanistic validation in prostate cancer

杂合亚苄基噻唑烷-2,4-二酮类化合物作为强效的凋亡诱导型抗癌药物:基于设计的优化、细胞毒性分析以及在前列腺癌中的机制验证

Shaaban, Saad; Hawas, Samia S; Sharaky, Marwa; Ba-Ghazal, Hussein; Elmaaty, Ayman Abo; Alomari, Khadra B; Alaasar, Mohamed; Elsharif, Asma M; Alatawi, Fatema S; Mohamed, Mohamed Alaa; Al Khatib, Arwa Omar; Al-Karmalawy, Ahmed A

Organoselenium-based Schiff bases and amidic acid derivatives as promising anticancer agents targeting breast cancer by downregulating BCL-2: design, synthesis, and biological evaluation

基于有机硒的席夫碱和酰胺酸衍生物作为靶向乳腺癌、通过下调BCL-2表达的潜在抗癌药物:设计、合成和生物学评价

Shaaban, Saad; Hawas, Samia S; Elsharif, Asma M; Sharaky, Marwa; Ba-Ghazal, Hussein; Alaasar, Mohamed; Alatawi, Fatema S; Alomari, Khadra B; Eissa, Mohamed E; Al Khatib, Arwa Omar; Alnajjar, Radwan; Al-Karmalawy, Ahmed A

In silico and in vitro study of the proapoptotic, autophagic and antitumor effects of cirsimaritin and humulene in hepatocellular carcinoma.

利用计算机模拟和体外实验研究了西西马汀和葎草烯在肝细胞癌中的促凋亡、自噬和抗肿瘤作用。

Ismail Abo-Elfadl Huda M, Megahd Huda E, Sharaky Marwa, Alshazly Omar, Mohamed Mamdouh F A, El-Rhman Amira Abd

Design, Synthesis, and Characterization of Novel Pyrazole Cross-Linked Chitosan Derivatives Modified with Zinc Oxide Nanoparticles for Boosting Their Anticancer Activity

设计、合成和表征新型吡唑交联壳聚糖衍生物,并用氧化锌纳米粒子修饰以增强其抗癌活性

Almutairi, Hanan D; Abdel-Motaal, Marwa; Sharaky, Marwa; Mohamed, Nadia A

New tetrahydroisoquinolines bearing nitrophenyl group targeting HSP90 and RET enzymes: synthesis, characterization and biological evaluation

靶向 HSP90 和 RET 酶的含硝基苯基的新型四氢异喹啉:合成、表征及生物学评价

Etify A Bakhite, Reda Hassanien, Nasser Farhan, Eman M Sayed, Marwa Sharaky

Folate-based binuclear Mn(II) chelates with 2,2'-bipyridine/1,10-phenanthroline as targeted anticancer agents for colon cancer cells.

以叶酸为基础的双核Mn(II)螯合物与2,2'-联吡啶/1,10-菲咯啉作为结肠癌细胞的靶向抗癌剂

Ragab Mona S, Soliman Marwa H, Sharaky Marwa M, Saad Abdelrahman, Shehata Mohamed R, Shoukry Mohamed M, Ragheb Mohamed A

Dual EGFR and telomerase inhibitory potential of new triazole tethered Schiff bases endowed with apoptosis: design, synthesis, and biological assessments

新型三唑连接的席夫碱具有双重 EGFR 和端粒酶抑制潜力,并能诱导细胞凋亡:设计、合成和生物学评价

Zeidan, Mohamed A; Ashour, Heba F; Yassen, Asmaa S A; Abo Elmaaty, Ayman; Farag, Ayman B; Sharaky, Marwa; Abdullah Alzahrani, Abdullah Yahya; Mughram, Mohammed H Al; Al-Karmalawy, Ahmed A

Isatin, a monoamine oxidase inhibitor, sensitizes resistant breast cancer cells to tamoxifen via MAO-A/HIF1α/MMPs modulation.

靛红是一种单胺氧化酶抑制剂,它通过 MAO-A/HIF1α/MMPs 调节使耐药乳腺癌细胞对他莫昔芬敏感。

Abdelwahed Fatma M, Ibrahim Marwa A, Sharaky Marwa, Effat Heba

Effect of palliative radiotherapy and cyclin-dependent kinase 4/6 inhibitor on breast cancer cell lines

姑息性放疗和细胞周期蛋白依赖性激酶 4/6 抑制剂对乳腺癌细胞系的影响

Sharaky, Marwa; El Kiki, Shereen M; Effat, Heba; Mansour, Heba H