日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cytochrome P450 2J2 is required for the natural compound austocystin D to elicit cancer cell toxicity

细胞色素 P450 2J2 是天然化合物 austocystin D 引发癌细胞毒性所必需的

Yukiko Kojima, Saki Fujieda, Liya Zhou, Masahiro Takikawa, Kouji Kuramochi, Toshiki Furuya, Ayaka Mizumoto, Noritaka Kagaya, Teppei Kawahara, Kazuo Shin-Ya, Shingo Dan, Akihiro Tomida, Fuyuki Ishikawa, Mahito Sadaie

Prediction of cell cycle distribution after drug exposure by high content imaging analysis using low-toxic DNA staining dye

使用低毒 DNA 染色染料通过高内涵成像分析预测药物暴露后的细胞周期分布

Kazuma Takeuchi, Yumiko Nishimura, Takayoshi Matsubara, Sho Isoyama, Asuka Suzuki, Masaaki Matsuura, Shingo Dan

Subtype-selective induction of apoptosis in translocation-related sarcoma cells induced by PUMA and BIM upon treatment with pan-PI3K inhibitors

泛 PI3K 抑制剂治疗后,PUMA 和 BIM 诱导的易位相关肉瘤细胞亚型选择性凋亡

Sho Isoyama, Naomi Tamaki, Yutaka Noguchi, Mutsumi Okamura, Yuki Yoshimatsu, Tadashi Kondo, Takeshi Suzuki, Shin-Ichi Yaguchi, Shingo Dan

Discovery of novel DNA-damaging agents through phenotypic screening for DNA double-strand break

通过 DNA 双链断裂表型筛选发现新型 DNA 损伤剂

Doudou Zhang, Takashi Shimokawa, Qianqian Guo, Shingo Dan, Yoshio Miki, Shigeaki Sunada

Structure-antitumor activity relationship of hybrid acetogenins focusing on connecting groups between heterocycles and the linker moiety

杂化乙酰辅酶A的结构-抗肿瘤活性关系,重点关注杂环和连接部分之间的连接基团

Kaito Ohta, Tetsuya Fushimi, Mutsumi Okamura, Akinobu Akatsuka, Shingo Dan, Hiroki Iwasaki, Masayuki Yamashita, Naoto Kojima

Spautin-1 inhibits mitochondrial complex I and leads to suppression of the unfolded protein response and cell survival during glucose starvation

Spautin-1 抑制线粒体复合物 I,导致葡萄糖饥饿期间未折叠蛋白反应和细胞存活受到抑制

Kazuhiro Kunimasa, Chika Ikeda-Ishikawa, Yuri Tani, Satomi Tsukahara, Junko Sakurai, Yuka Okamoto, Masaru Koido, Shingo Dan, Akihiro Tomida

Suppression of tumor metastasis by a RECK-activating small molecule

RECK 激活小分子抑制肿瘤转移

Yoko Yoshida, Kanako Yuki, Shingo Dan, Kanami Yamazaki, Makoto Noda

Cancer immunotherapy with PI3K and PD-1 dual-blockade via optimal modulation of T cell activation signal

通过优化调节 T 细胞活化信号,实现 PI3K 和 PD-1 双重阻断的癌症免疫治疗

Sho Isoyama, Shigeyuki Mori, Daisuke Sugiyama, Yasuhiro Kojima, Yasuko Tada, Kohei Shitara, Kunihiko Hinohara, Shingo Dan, Hiroyoshi Nishikawa

Mitochondrial complex I inhibitors suppress tumor growth through concomitant acidification of the intra- and extracellular environment

线粒体复合物 I 抑制剂通过同时酸化细胞内和细胞外环境来抑制肿瘤生长。

Junjiro Yoshida ,Tomokazu Ohishi ,Hikaru Abe ,Shun-Ichi Ohba ,Hiroyuki Inoue ,Ihomi Usami ,Masahide Amemiya ,Raphael Oriez ,Chiharu Sakashita ,Shingo Dan ,Minoru Sugawara ,Tokuichi Kawaguchi ,Junko Ueno ,Yuko Asano ,Ami Ikeda ,Manabu Takamatsu ,Gulanbar Amori ,Yasumitsu Kondoh ,Kaori Honda ,Hiroyuki Osada ,Tetsuo Noda ,Takumi Watanabe ,Takao Shimizu ,Masakatsu Shibasaki ,Manabu Kawada

Lamellarin 14, a derivative of marine alkaloids, inhibits the T790M/C797S mutant epidermal growth factor receptor

层状蛋白 14 是一种海洋生物碱衍生物,可抑制 T790M/C797S 突变表皮生长因子受体

Naoyuki Nishiya, Yusuke Oku, Chie Ishikawa, Tsutomu Fukuda, Shingo Dan, Tetsuo Mashima, Masaru Ushijima, Yoko Furukawa, Yuka Sasaki, Keishi Otsu, Tomoko Sakyo, Masanori Abe, Honami Yonezawa, Fumito Ishibashi, Masaaki Matsuura, Akihiro Tomida, Hiroyuki Seimiya, Takao Yamori, Masatomo Iwao, Yoshimasa