日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multifunctional, Fluorene-Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease

一种多功能、基于芴的胆碱能和GABA能神经传递调节剂,作为阿尔茨海默病姑息治疗的新型候选药物

Panek, Dawid; Pasieka, Anna; Jończyk, Jakub; Gawlińska, Milena; Zaręba, Paula; Siwek, Agata; Wolak, Małgorzata; Mordyl, Barbara; Głuch-Lutwin, Monika; Latacz, Gniewomir; Brazzolotto, Xavier; Chantegreil, Fabien; Nachon, Florian; Zdarova Karasova, Jana; Pejchal, Jaroslav; Mzik, Martin; Sestak, Vit; Prchal, Lukas; Odvarkova, Jitka; Soukup, Ondrej; Korabecny, Jan; Sorf, Ales; Hamsikova, Marie; Zemanova, Lucie; Muckova, Lubica; Vánova, Nela; Dryja, Pola; Sałat, Kinga; Höfner, Georg; Wanner, Klaus; Więckowska, Anna; Malawska, Barbara

Revolutionizing tuberculosis treatment: Breakthroughs, challenges, and hope on the horizon

结核病治疗的革命性变革:突破、挑战与希望

Kufa, Martin; Finger, Vladimir; Kovar, Ondrej; Soukup, Ondrej; Torruellas, Carilyn; Roh, Jaroslav; Korabecny, Jan

Glutamate utilization fuels rapid production of mitochondrial ROS in dendritic cells and drives systemic inflammation during tularemia.

谷氨酸的利用促进树突状细胞中线粒体活性氧的快速产生,并在兔热病期间引发全身炎症

Fabrik Ivo, Spidlova Petra, Prchal Lukas, Fabrikova Daniela, Viduka Ina, Marecic Valentina, Filimonenko Vlada, Sleha Radek, Vajrychova Marie, Kupcik Rudolf, Soukup Ondrej, Rousar Tomas, Härtlova Anetta, Santic Marina, Stulik Jiri

Scaffold Hopping in Tuberculosis Drug Discovery: Principles, Applications, and Case Studies

结核病药物研发中的骨架跃迁:原理、应用和案例研究

Kovar, Ondrej; Kufa, Martin; Finger, Vladimir; Soukup, Ondrej; Kratky, Martin; Torruellas, Carilyn; Roh, Jaroslav; Korabecny, Jan

Nanodiamond mediated delivery of pyridinium oxime antidotes to central nervous system for potential treatment of exposure to nerve agents

利用纳米金刚石介导将吡啶肟解毒剂递送至中枢神经系统,有望用于治疗神经毒剂暴露。

Bondar, Denys; Smirnova, Olga; Nagappa, Nandish M; Heinmaa, Ivo; Soukup, Ondrej; Kobrlova, Tereza; Opravil, Jakub; Hrabinova, Martina; Jun, Daniel; Starkov, Pavel; Spuul, Pirjo; Kuča, Kamil; Mochalin, Vadym N; Karpichev, Yevgen

Memantine Administration Enhances Glutamatergic and GABAergic Pathways in the Human Hippocampus of Alzheimer's Disease Patients

美金刚给药可增强阿尔茨海默病患者海马体中的谷氨酸能和GABA能通路

Fabrik, Ivo; Kupcik, Rudolf; Fabrikova, Daniela; Chvojkova, Marketa; Holubova, Kristina; Hakenova, Kristina; Horak, Martin; Soukup, Jiri; Manethova, Monika; Rusina, Robert; Matej, Radoslav; Ryska, Ales; Soukup, Ondrej

The Effect of Tacrine on Functional Response of the Lower Oesophageal Sphincter Assessed by Endoscopic Luminal Impedance Planimetry in Experimental Pigs

他克林对实验猪下食管括约肌功能反应的影响——内镜腔阻抗容积描记法评估

Bures, Jan; Novak, Martin; Radochova, Vera; Kohoutova, Darina; Prchal, Lukas; Martinek, Jan; Mares, Jan; Cerny, Jaroslav; Suchanek, Stepan; Pejchal, Jaroslav; Voxova, Barbora; Urbanek, Petr; Zavoral, Miroslav; Soukup, Ondrej

Discovery of a 6-Aminobenzo[b]thiophene 1,1-Dioxide Derivative (K2071) with a Signal Transducer and Activator of Transcription 3 Inhibitory, Antimitotic, and Senotherapeutic Activities.

发现一种 6-氨基苯并[b]噻吩 1,1-二氧化物衍生物 (K2071),具有信号转导和转录激活因子 3 抑制、抗有丝分裂和衰老治疗活性

Oleksak Patrik, Rysanek David, Vancurova Marketa, Vasicova Pavla, Urbancokova Alexandra, Novak Josef, Maurencova Dominika, Kashmel Pavel, Houserova Jana, Mikyskova Romana, Novotny Ondrej, Reinis Milan, Juda Pavel, Hons Miroslav, Kroupova Jirina, Sedlak David, Sulimenko Tetyana, Draber Pavel, Chlubnova Marketa, Nepovimova Eugenie, Kuca Kamil, Lisa Miroslav, Andrys Rudolf, Kobrlova Tereza, Soukup Ondrej, Janousek Jiri, Prchal Lukas, Bartek Jiri, Musilek Kamil, Hodny Zdenek

A-agents, misleadingly known as "Novichoks": a narrative review

A型特工,被误导地称为“诺维乔克”:一篇叙述性综述

Opravil, Jakub; Pejchal, Jaroslav; Finger, Vladimir; Korabecny, Jan; Rozsypal, Tomas; Hrabinova, Martina; Muckova, Lubica; Hepnarova, Vendula; Konecny, Jan; Soukup, Ondrej; Jun, Daniel

Is It the Twilight of BACE1 Inhibitors?

BACE1抑制剂的末日到了吗?

Hrabinova, Martina; Pejchal, Jaroslav; Kucera, Tomas; Jun, Daniel; Schmidt, Monika; Soukup, Ondrej