日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Whole-genome CRISPR-Cas9 knockout screens identify SHOC2 as a genetic dependency in NRAS-mutant melanoma

全基因组 CRISPR-Cas9 敲除筛选鉴定出 SHOC2 是 NRAS 突变型黑色素瘤的遗传依赖性基因

Gu, Andrea Y; Lee, Tet Woo; Khan, Aziza; Zhang, Xuenan; Hunter, Francis W; Singleton, Dean C; Jamieson, Stephen M F

CRISPR screens with trastuzumab emtansine in HER2-positive breast cancer cell lines reveal new insights into drug resistance

利用曲妥珠单抗-美坦新在HER2阳性乳腺癌细胞系中进行CRISPR筛选,揭示了耐药性的新机制。

Lipert, Barbara A; Siemens, Kyla N; Khan, Aziza; Airey, Rebecca; Dam, Gech Heng; Lu, Man; Flinterman, Marcella; Yong, Queenie; Lee, Tet Woo; Hunter, Francis W; Jamieson, Stephen M F

Growth hormone receptor antagonists, GHA2 and GHA3, with dual activity against the human and mouse receptor

生长激素受体拮抗剂GHA2和GHA3,对人和小鼠受体均具有活性。

Wang, Yue; Langley, Ries J; Harms, Julia; Portlock, Theo; Jamieson, Stephen M F; Perry, Jo K

The Chemistry of Anticancer Mononuclear and N-Bridged Dinuclear 8-Aminoquinoline Half-sandwich Metal Complexes

抗癌单核和N桥双核8-氨基喹啉半夹心金属配合物的化学性质

Steel, Tasha R; Stjärnhage, Julia; Riisom, Mie; Bloomfield, Hugh O; Herbert, Caitlin D; Jamieson, Stephen M F; Astin, Jonathan W; Söhnel, Tilo; Hartinger, Christian G

Identification of 6-Anilino Imidazo[4,5- c]pyridin-2-ones as Selective DNA-Dependent Protein Kinase Inhibitors and Their Application as Radiosensitizers

鉴定6-苯胺基咪唑并[4,5-c]吡啶-2-酮类化合物为选择性DNA依赖性蛋白激酶抑制剂及其在放射增敏剂中的应用

Cho R Hong,Lydia P Liew,Way W Wong,Benjamin D Dickson,Gary Cheng,Avik Shome,Rebecca Airey,Jagdish Jaiswal,Barbara Lipert,Stephen M F Jamieson,William R Wilson,Michael P Hay

Clinical relevance and therapeutic predictive ability of hypoxia biomarkers in head and neck cancer tumour models

缺氧生物标志物在头颈癌肿瘤模型中的临床意义和治疗预测能力

Lee, Tet Woo; Singleton, Dean C; Harms, Julia K; Lu, Man; McManaway, Sarah P; Lai, Amy; Tercel, Moana; Pruijn, Frederik B; Macann, Andrew M J; Hunter, Francis W; Wilson, William R; Jamieson, Stephen M F

Clonal dynamics limits detection of selection in tumour xenograft CRISPR/Cas9 screens

克隆动力学限制了肿瘤异种移植 CRISPR/Cas9 筛选中的选择检测

Tet Woo Lee, Francis W Hunter, Peter Tsai, Cristin G Print, William R Wilson, Stephen M F Jamieson

NIMG-70. MAGNETIC RESONANCE HYPOXIA IMAGING FOR RADIATION TREATMENT GUIDANCE IN GLIOBLASTOMA MULTIFORME - A DIAGNOSTIC/PROGNOSTIC CLINICAL IMAGING STUDY

NIMG-70. 磁共振低氧成像在多形性胶质母细胞瘤放射治疗指导中的应用——一项诊断/预后临床影像学研究

Harms, Julia K; Lee, Tet-Woo; Wang, Tao; Lai, Amy; Kee, Dennis; Chaplin, John M; McIvor, Nick P; Hunter, Francis W; Macann, Andrew M J; Wilson, William R; Jamieson, Stephen M F; Brighi, Caterina; Waddington, David; Keall, Paul; Booth, Jeremy; O'Brien, Kieran; Parkinson, Jonathon; Yim, Jackie; Bailey, Dale; Back, Michael; Drummond, James

Preclinical Activity and Pharmacokinetic/Pharmacodynamic Relationship for a Series of Novel Benzenesulfonamide Perforin Inhibitors

一系列新型苯磺酰胺类穿孔素抑制剂的临床前活性及药代动力学/药效学关系

Kate H Gartlan ,Jagdish K Jaiswal ,Matthew R Bull ,Hedieh Akhlaghi ,Vivien R Sutton ,Kylie A Alexander ,Karshing Chang ,Geoffrey R Hill ,Christian K Miller ,Patrick D O'Connor ,Jiney Jose ,Joseph A Trapani ,Susan A Charman ,Julie A Spicer ,Stephen M F Jamieson

Impact of the Metal Center and Leaving Group on the Anticancer Activity of Organometallic Complexes of Pyridine-2-carbothioamide

金属中心和离去基团对吡啶-2-硫代甲酰胺有机金属配合物抗癌活性的影响

Arshad, Jahanzaib; Tong, Kelvin K H; Movassaghi, Sanam; Söhnel, Tilo; Jamieson, Stephen M F; Hanif, Muhammad; Hartinger, Christian G