日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BRD4 PROTAC degrader ARV-825 inhibits T-cell acute lymphoblastic leukemia by targeting 'Undruggable' Myc-pathway genes

BRD4 PROTAC 降解剂 ARV-825 通过靶向“不可治疗”的 Myc 通路基因来抑制 T 细胞急性淋巴细胞白血病

Shuiyan Wu #, You Jiang #, Yi Hong #, Xinran Chu, Zimu Zhang, Yanfang Tao, Ziwei Fan, Zhenjiang Bai, Xiaolu Li, Yanling Chen, Zhiheng Li, Xin Ding, Haitao Lv, Xiaoli Du, Su Lin Lim, Yongping Zhang, Saihu Huang, Jun Lu, Jian Pan, Shaoyan Hu0

PROTAC Bromodomain Inhibitor ARV-825 Displays Anti-Tumor Activity in Neuroblastoma by Repressing Expression of MYCN or c-Myc

PROTAC 溴结构域抑制剂 ARV-825 通过抑制 MYCN 或 c-Myc 的表达在神经母细胞瘤中表现出抗肿瘤活性

Zhiheng Li, Su Lin Lim, Yanfang Tao, Xiaolu Li, Yi Xie, Chun Yang, Zimu Zhang, You Jiang, Xianbing Zhang, Xu Cao, Hairong Wang, Guanghui Qian, Yi Wu, Mei Li, Fang Fang, Ying Liu, Mingcui Fu, Xin Ding, Zhenghong Zhu, Haitao Lv, Jun Lu, Sheng Xiao, Shaoyan Hu, Jian Pan

Multiple myeloma: Combination therapy of BET proteolysis targeting chimeric molecule with CDK9 inhibitor

多发性骨髓瘤:BET蛋白水解靶向嵌合分子与CDK9抑制剂联合治疗

Su-Lin Lim, Liang Xu, Bing-Chen Han, Pavithra Shyamsunder, Wee-Joo Chng, H Phillip Koeffler

Proteolysis targeting chimeric molecules as therapy for multiple myeloma: efficacy, biomarker and drug combinations

蛋白水解靶向嵌合分子治疗多发性骨髓瘤:疗效、生物标志物和药物组合

Su Lin Lim, Alisa Damnernsawad, Pavithra Shyamsunder, Wee Joo Chng, Bing Chen Han, Liang Xu, Jian Pan, Dakle Pushkar Pravin, Serhan Alkan, Jeffrey W Tyner, H Phillip Koeffler

Mutational Landscape of Pediatric Acute Lymphoblastic Leukemia

儿童急性淋巴细胞白血病的突变概况

Ling-Wen Ding #, Qiao-Yang Sun #, Kar-Tong Tan #, Wenwen Chien, Anand Mayakonda, Allen Eng Juh Yeoh, Norihiko Kawamata, Yasunobu Nagata, Jin-Fen Xiao, Xin-Yi Loh, De-Chen Lin, Manoj Garg, Yan-Yi Jiang, Liang Xu, Su-Lin Lim, Li-Zhen Liu, Vikas Madan, Masashi Sanada, Lucia Torres Fernández, S S Hema P

SETDB1 accelerates tumourigenesis by regulating the WNT signalling pathway

SETDB1通过调控WNT信号通路加速肿瘤发生

Qiao-Yang Sun, Ling-Wen Ding, Jin-Fen Xiao, Wenwen Chien, Su-Lin Lim, Norimichi Hattori, Lee Goodglick, David Chia, Vei Mah, Mohammad Alavi, Sara R Kim, Ngan B Doan, Jonathan W Said, Xin-Yi Loh, Liang Xu, Li-Zhen Liu, Henry Yang, Takahide Hayano, Shuo Shi, Dong Xie, De-Chen Lin, H Phillip Koeffler