日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MTA-cooperative PRMT5 inhibitors from cofactor-directed DNA-encoded library screens.

通过辅因子导向的DNA编码文库筛选得到的MTA协同PRMT5抑制剂

Andersson Jan, Cowland Sanne, Vestergaard Mikkel, Yang Yajing, Liu Siyuan, Fang Xie, Mukund Susmith, Ghimire-Rijal Sudipa, Carter Chris, Chung Grace, Jacso Tomas, Sarvary Ian, Hughes Paul E, Gouliaev Alex, Payton Marc, Belmontes Brian, Caenepeel Sean, Franch Thomas, Glad Sanne, Husemoen Birgitte, Nielsen Søren Jensby

From DNA-Encoded Library Screening to AM-9747: An MTA-Cooperative PRMT5 Inhibitor with Potent Oral In Vivo Efficacy.

从 DNA 编码文库筛选到 AM-9747:一种具有强效口服体内疗效的 MTA 协同 PRMT5 抑制剂

Sarvary Ian, Vestergaard Mikkel, Moretti Loris, Andersson Jan, Peiró Cadahía Jorge, Cowland Sanne, Flagstad Thomas, Franch Thomas, Gouliaev Alex, Husemoen Gitte, Jacso Tomas, Kronborg Titi, Kuropatnicka Aleksandra, Nadali Anna, Madsen Mads, Nielsen So Ren, Pii David, Ryborg So Ren, Soede Camillia, Allen Jennifer R, Bourbeau Matthew, Li Kexue, Liu Qingyian, Lo Mei-Chu, Madoux Franck, Mardirossian Narbe, Moriguchi Jodi, Ngo Rachel, Peng Chi-Chi, Pettus Liping, Tamayo Nuria, Wang Paul, Kapoor Rajiv, Belmontes Brian, Caenepeel Sean, Hughes Paul, Liu Siyuan, Slemmons Katherine K, Yang Yajing, Xie Fang, Ghimire-Rijal Sudipa, Mukund Susmith, Glad Sanne

Unveiling Hidden Risks: Intentional Molecular Screening for Sexually Transmitted Infections and Vaginosis Pathogens in Patients Who Have Been Exclusively Tested for Human Papillomavirus Genotyping

揭示隐藏的风险:对已接受过人乳头瘤病毒基因分型检测的患者进行性传播感染和阴道病病原体的分子筛查

Fabiola Hernández-Rosas, Manuel Rey-Barrera, Flavio Hernández-Barajas, Claudia Rangel-Soto, Mariana Socorro García-González, Shumeyker Susmith Franco-González, Mercedes Piedad de León-Bautista

Potassium channels Kv1.3 and KCa3.1 cooperatively and compensatorily regulate antigen-specific memory T cell functions

钾通道 Kv1.3 和 KCa3.1 协同和补偿性调节抗原特异性记忆 T 细胞功能

Eugene Y Chiang, Tianbo Li, Surinder Jeet, Ivan Peng, Juan Zhang, Wyne P Lee, Jason DeVoss, Patrick Caplazi, Jun Chen, Søren Warming, David H Hackos, Susmith Mukund, Christopher M Koth, Jane L Grogan

Phosphorylation and linear ubiquitin direct A20 inhibition of inflammation

磷酸化和线性泛素直接抑制 A20 炎症

Ingrid E Wertz, Kim Newton, Dhaya Seshasayee, Saritha Kusam, Cynthia Lam, Juan Zhang, Nataliya Popovych, Elizabeth Helgason, Allyn Schoeffler, Surinder Jeet, Nandhini Ramamoorthi, Lorna Kategaya, Robert J Newman, Keisuke Horikawa, Debra Dugger, Wendy Sandoval, Susmith Mukund, Anuradha Zindal, Flaviu

IL-12 secreting tumor-targeted chimeric antigen receptor T cells eradicate ovarian tumors in vivo

分泌IL-12的肿瘤靶向嵌合抗原受体T细胞可在体内根除卵巢肿瘤。

Koneru, Mythili; Purdon, Terence J; Spriggs, David; Koneru, Susmith; Brentjens, Renier J

Histone deacetylase (HDAC) inhibitor kinetic rate constants correlate with cellular histone acetylation but not transcription and cell viability

组蛋白去乙酰化酶(HDAC)抑制剂的动力学速率常数与细胞组蛋白乙酰化相关,但与转录和细胞活力无关。

Benjamin E L Lauffer ,Robert Mintzer, Rina Fong, Susmith Mukund, Christine Tam, Inna Zilberleyb, Birgit Flicke, Allegra Ritscher, Grazyna Fedorowicz, Roxanne Vallero, Daniel F Ortwine, Janet Gunzner, Zora Modrusan, Lars Neumann, Christopher M Koth, Patrick J Lupardus, Joshua S Kaminker, Christopher E Heise, Pascal Steiner

Mechanism of displacement of a catalytically essential loop from the active site of mammalian fructose-1,6-bisphosphatase

哺乳动物果糖-1,6-二磷酸酶活性位点催化必需环的置换机制

Gao, Yang; Iancu, Cristina V; Mukind, Susmith; Choe, Jun-Yong; Honzatko, Richard B

Affinities between the binding partners of the HIV-1 integrase dimer-lens epithelium-derived growth factor (IN dimer-LEDGF) complex

HIV-1 整合酶二聚体-晶状体上皮衍生生长因子 (IN 二聚体-LEDGF) 复合物结合伙伴之间的亲和力

Manuel Tsiang, Gregg S Jones, Magdeleine Hung, Susmith Mukund, Bin Han, Xiaohong Liu, Kerim Babaoglu, Eric Lansdon, Xiaowu Chen, Jacob Todd, Terrence Cai, Nikos Pagratis, Roman Sakowicz, Romas Geleziunas