日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Library docking for Cannabinoid-2 Receptor ligands

大麻素-2受体配体的库对接

Rachman, Moira M; Iliopoulos-Tsoutsouvas, Christos; Sacco, Michael D; Xu, Xinyu; Wu, Cheng-Guo; Santos, Emma; Glenn, Isabella S; Paris, Lu; Cahill, Michelle K; Ganapathy, Suthakar; Tummino, Tia A; Moroz, Yurii S; Radchenko, Dmytro S; Okorie, Meri; Tawfik, Vivianne; Irwin, John J; Makriyannis, Alexandros; Skiniotis, Georgios; Shoichet, Brian K

Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects.

针对副作用较小的 1 型大麻素受体激动剂的虚拟库对接

Tummino Tia A, Iliopoulos-Tsoutsouvas Christos, Braz Joao M, O'Brien Evan S, Stein Reed M, Craik Veronica, Tran Ngan K, Ganapathy Suthakar, Liu Fangyu, Shiimura Yuki, Tong Fei, Ho Thanh C, Radchenko Dmytro S, Moroz Yurii S, Rosado Sian Rodriguez, Bhardwaj Karnika, Benitez Jorge, Liu Yongfeng, Kandasamy Herthana, Normand Claire, Semache Meriem, Sabbagh Laurent, Glenn Isabella, Irwin John J, Kumar Kaavya Krishna, Makriyannis Alexandros, Basbaum Allan I, Shoichet Brian K

Systematic Engineering of TROP2-Targeted CAR T-Cell Therapy Overcomes Resistance Pathways in Solid Tumors

系统性改造TROP2靶向CAR T细胞疗法可克服实体瘤的耐药通路

Elliott J Brea,Simon Baldacci,Neil Savage,Francesco Facchinetti,Conor Hinchey,Sachiv Chakravarti,Alexis Mottram,Kenneth Ngo,Ha Vo,Brittaney A Leeper,Bishma Tuladhar,Suthakar Ganapathy,Elena V Ivanova,Aisha Saldanha,Marie-Anais Locquet,Abdulmajeed Salamah,Malcolm Holterhus,Evelyn B Mesler,Martina De Vizio,Carla Stornante,Marco Campisi,Navin R Mahadevan,Tran C Thai,Timothy J Haggerty,Zehua Li,Cui Nie,Changjing Deng,Xiaoxiao Wang,Louis L Liu,Thanh U Barbie,Prafulla C Gokhale,Cloud P Paweletz,Anusuya Ramasubramanian,Pasi A Jänne,David A Barbie,Eric L Smith

Novel Tetraolefinic Chain Phenyl Substituted Endocannabinoid Probes.

新型四烯烃链苯基取代内源性大麻素探针。

Georgiadis Markos-Orestis, Ji Lipin, Tong Fei, Dang Vuong Q, Ferreira Luana Assis, Faragher Alexandra, Tran Ngan, Sadybekov Anastasiia V, Ganapathy Suthakar, Zvonok Nikolai, Katritch Vsevolod, Hohmann Andrea G, Bohn Laura M, Makriyannis Alexandros, Nikas Spyros P

RSONAR: Data-Driven Evaluation of Dual-Use Star Tracker for Stratospheric Space Situational Awareness (SSA)

RSONAR:用于平流层空间态势感知(SSA)的双用途星敏感器的数据驱动评估

Suthakar, Vithurshan; Porto, Ian; Myhre, Marissa; Sanvido, Aiden Alexander; Clark, Ryan; Lee, Regina S K

The USP1 Inhibitor KSQ-4279 Overcomes PARP Inhibitor Resistance in Homologous Recombination-Deficient Tumors

USP1 抑制剂 KSQ-4279 克服了同源重组缺陷肿瘤中的 PARP 抑制剂耐药性

Louise Cadzow, Jehrod Brenneman, Erica Tobin, Pamela Sullivan, Sumeet Nayak, Janid A Ali, Sol Shenker, Jim Griffith, Michael McGuire, Paula Grasberger, Yuji Mishina, Morgan Murray, Anne E Dodson, Hugh Gannon, Elsa Krall, Jeff Hixon, Edmond Chipumuro, Kerstin Sinkevicius, Prafulla C Gokhale, Suthakar

CAR memory-like NK cells targeting the membrane proximal domain of mesothelin demonstrate promising activity in ovarian cancer

靶向间皮素膜近端结构域的 CAR 记忆样 NK 细胞在卵巢癌中表现出良好的活性

Mubin Tarannum, Khanhlinh Dinh, Juliana Vergara, Grace Birch, Yasmin Z Abdulhamid, Isabel E Kaplan, Oyku Ay, Andreia Maia, Owen Beaver, Michal Sheffer, Roman Shapiro, Alaa Kassim Ali, Han Dong, James Dongjoo Ham, Eden Bobilev, Sydney James, Amy B Cameron, Quang-De Nguyen, Suthakar Ganapathy, Chayapa

Improving agricultural spraying with multi-rotor drones: a technical study on operational parameter optimization

利用多旋翼无人机改进农业喷洒:作业参数优化技术研究

Yallappa, D; Kavitha, R; Surendrakumar, A; Suthakar, B; Mohan Kumar, A P; Kannan, Balaji; Kalarani, M K

ABRpresto: An algorithm for automatic thresholding of the Auditory Brainstem Response using resampled cross-correlation across subaverages

ABRpresto:一种利用子平均值间的重采样互相关进行听觉脑干反应自动阈值化的算法

Shaheen, Luke A; Buran, Brad N; Suthakar, Kirupa; Koehler, Seth D; Chung, Yoojin

Experience-dependent flexibility in a molecularly diverse central-to-peripheral auditory feedback system

分子多样化的中枢到外周听觉反馈系统中依赖经验的灵活性

Michelle M Frank, Austen A Sitko, Kirupa Suthakar, Lester Torres Cadenas, Mackenzie Hunt, Mary Caroline Yuk, Catherine J C Weisz, Lisa V Goodrich