日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Role of donor regulatory T-cell adoptive immunotherapy in B-cell immunity after hematopoietic cell transplantation

供体调节性T细胞过继免疫疗法在造血干细胞移植后B细胞免疫中的作用

Piccinelli, Sara; Limongello, Roberto; Viglione, Valerio; Hohxa, Eni; Zei, Tiziana; Ostini, Roberta Iacucci; Bigerna, Barbara; Tabarrini, Alessia; Sembenico, Rebecca; Tricarico, Sara; Zorutti, Francesco; Martelli, Maria Paola; Carotti, Alessandra; Martelli, Massimo Fabrizio; Velardi, Andrea; Ruggeri, Loredana; Mancusi, Antonella; Pierini, Antonio

Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5'-Terminal Oligopyrimidine Motif-Containing mRNA

磺酰邻氨基苯甲酸类似物通过下调由含5'末端寡嘧啶基序的mRNA编码的核糖体蛋白的表达,表现出泛血清型抗登革热活性。

Gwee, Chin Piaw; Felicetti, Tommaso; Chan, Kitti Wing Ki; Tan, Min Jie Alvin; Bin Mohd Mazlan, Muhammad Danial; Milite, Ciro; Pepe, Giacomo; Sarnari, Chiara; Ng, Xiao Dan; Phoo, Wint Wint; Tan, Jasmine Hwee Yee; Mah, Marcus G; Watanabe, Satoru; Huang, Jing Xiu; Massari, Serena; Tabarrini, Oriana; Sabatini, Stefano; Campiglia, Pietro; Sbardella, Gianluca; Smith, Gavin J D; Alonso, Sylvie; Sun, Alfred Xuyang; Sobota, Radoslaw M; Vasudevan, Subhash G; Manfroni, Giuseppe

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3-c][1,2]benzothiazine 5,5-Dioxide Derivatives

NorA 外排泵抑制剂:扩展吡唑并[4,3-c][1,2]苯并噻嗪 5,5-二氧化物衍生物的构效关系知识

Cernicchi, Giada; Di Gregorio, Alessandra; Felicetti, Tommaso; Rampacci, Elisa; Casari, Giulia; Armeni, Tatiana; Romaldi, Brenda; Zefaj, Ermelinda; Passamonti, Fabrizio; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Vignaroli, Carla; Sabatini, Stefano

New Pyridobenothiazolone Derivatives Display Nanomolar Pan-Serotype Anti-Dengue Virus Activity.

新型吡啶并噻唑啉酮衍生物显示出纳摩尔级泛血清型抗登革病毒活性

Felicetti Tommaso, Gwee Chin Piaw, Chan Kitti Wing Ki, Pepe Giacomo, Milite Ciro, Campiglia Pietro, Watanabe Satoru, Mazlan Muhammad Danial Bin Mohd, Sabatini Stefano, Massari Serena, Tabarrini Oriana, Sbardella Gianluca, Vasudevan Subhash G, Manfroni Giuseppe

New anti-ovarian cancer quinolone derivatives acting by modulating microRNA processing machinery

通过调节 microRNA 加工机制发挥作用的新型抗卵巢癌喹诺酮衍生物

Tommaso Felicetti, Nicola Di Iacovo, Maria Agnese Della Fazia, Danilo Piobbico, Stefania Pieroni, Martina Pacetti, Jialing Yu, Yilun Sun, Serena Massari, Maria Letizia Barreca, Stefano Sabatini, Oriana Tabarrini, Violetta Cecchetti, Fei Wang, Yves Pommier, Mariangela Morlando, Giuseppe Servillo, Giu

New anti-ovarian cancer quinolone derivatives acting by modulating microRNA processing machinery

新型抗卵巢癌喹诺酮衍生物通过调节microRNA加工机制发挥作用

Tommaso Felicetti,Nicola Di Iacovo,Maria Agnese Della Fazia,Danilo Piobbico,Stefania Pieroni,Martina Pacetti,Jialing Yu,Yilun Sun,Serena Massari,Maria Letizia Barreca,Stefano Sabatini,Oriana Tabarrini,Violetta Cecchetti,Fei Wang,Yves Pommier,Mariangela Morlando,Giuseppe Servillo,Giuseppe Manfroni

Synthetically accessible de novo design using reaction vectors: Application to PARP1 inhibitors

利用反应载体进行合成可及的从头设计:应用于PARP1抑制剂

Ghiandoni, Gian Marco; Flanagan, Stuart R; Bodkin, Michael J; Nizi, Maria Giulia; Galera-Prat, Albert; Brai, Annalaura; Chen, Beining; Wallace, James E A; Hristozov, Dimitar; Webster, James; Manfroni, Giuseppe; Lehtiö, Lari; Tabarrini, Oriana; Gillet, Valerie J

[1,2,4]Triazolo[3,4- b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes

[1,2,4]三唑并[3,4-b]苯并噻唑支架作为多功能烟酰胺模拟物,可对不同的 PARP 酶进行纳摩尔级抑制

Sudarshan Murthy, Maria Giulia Nizi, Mirko M Maksimainen, Serena Massari, Juho Alaviuhkola, Barbara E Lippok, Chiara Vagaggini, Sven T Sowa, Albert Galera-Prat, Yashwanth Ashok, Harikanth Venkannagari, Renata Prunskaite-Hyyryläinen, Elena Dreassi, Bernhard Lüscher, Patricia Korn, Oriana Tabarrini, L

Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules

从药物化学角度探讨小分子靶向单ADP核糖基化PARP的策略

Nizi, Maria Giulia; Maksimainen, Mirko M; Lehtiö, Lari; Tabarrini, Oriana