日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hsc70 promotes anti-tumor immunity by targeting PD-L1 for lysosomal degradation

Hsc70通过靶向PD-L1使其溶酶体降解,从而促进抗肿瘤免疫。

Xiaoyan Xu # ,Tingxue Xie # ,Mengxin Zhou # ,Yaqin Sun # ,Fengqi Wang # ,Yanan Tian ,Ziyan Chen ,Yanqi Xie ,Ronghai Wu ,Xufeng Cen ,Jichun Zhou ,Tingjun Hou ,Lei Zhang ,Chaoyang Huang ,Qingwei Zhao ,Dongrui Wang ,Hongguang Xia

Myofascial edema of gastrocnemius: A prominent MRI characteristic in dermatomyositis patients with anti-transcriptional intermediate factor 1-γ antibody

腓肠肌肌筋膜水肿:抗转录中间因子1-γ抗体阳性皮肌炎患者的显著MRI特征

Zhen, Chao; Zhao, Bing; He, Jingzhen; Wei, Li; Yan, Chuanzhu; Dai, Tingjun; Hou, Ying

Discovery of Novel Anti-Resistance AR Antagonists Guided by Funnel Metadynamics Simulation

漏斗元动力学模拟指导新型抗耐药 AR 拮抗剂的发现

Haiyi Chen, Yuxin Zhou, Xinyue Wang, Xin Chai, Zhe Wang, Ercheng Wang, Lei Xu, Tingjun Hou, Dan Li, Mojie Duan

A small molecule inhibitor of the UBE2F-CRL5 axis induces apoptosis and radiosensitization in lung cancer

UBE2F-CRL5 轴的小分子抑制剂诱导肺癌细胞凋亡和放射增敏

Tiantian Xu #, Qisheng Ma #, Yanan Li, Qing Yu, Peichen Pan, Yawen Zheng, Zhijian Li, Xiufang Xiong, Tingjun Hou, Bin Yu, Hongmin Liu, Yi Sun

Structure-guided and phage-assisted evolution of a therapeutic anti-EGFR antibody to reverse acquired resistance

结构引导和噬菌体辅助进化治疗性抗 EGFR 抗体以逆转获得性耐药性

Xinlei Zhuang #, Zhe Wang #, Jiansheng Fan, Xuefei Bai, Yingchun Xu, James J Chou, Tingjun Hou, Shuqing Chen, Liqiang Pan

High-throughput glycolytic inhibitor discovery targeting glioblastoma by graphite dots-assisted LDI mass spectrometry

通过石墨点辅助 LDI 质谱法发现针对胶质母细胞瘤的高通量糖酵解抑制剂

Rui Shi, Peichen Pan, Rui Lv, Chongqing Ma, Enhui Wu, Ruochen Guo, Zhihao Zhao, Hexing Song, Joe Zhou, Yang Liu, Guoqiang Xu, Tingjun Hou, Zhenhui Kang, Jian Liu

Discovery and Optimization of N-Acyl-6-sulfonamide-tetrahydroquinoline Derivatives as Novel Non-Steroidal Selective Glucocorticoid Receptor Modulators

发现和优化 N-酰基-6-磺酰胺-四氢喹啉衍生物作为新型非甾体选择性糖皮质激素受体调节剂

Dan Li, Xiaodong Bao, Jinping Pang, Xueping Hu, Longling Wang, Jiajia Wang, Zhaoxu Yang, Lei Xu, Siyu Wang, Qinjie Weng, Sunliang Cui, Tingjun Hou

Discovery of novel non-steroidal selective glucocorticoid receptor modulators by structure- and IGN-based virtual screening, structural optimization, and biological evaluation

通过基于结构和 IGN 的虚拟筛选、结构优化和生物学评价发现新型非甾体选择性糖皮质激素受体调节剂

Xueping Hu, Jinping Pang, Changwei Chen, Dejun Jiang, Chao Shen, Xin Chai, Liu Yang, Xujun Zhang, Lei Xu, Sunliang Cui, Tingjun Hou, Dan Li

Multi-Channel Metabolomics Analysis Identifies Novel Metabolite Biomarkers for the Early Detection of Fatty Liver Disease in Dairy Cows

多通道代谢组学分析鉴定出用于奶牛脂肪肝疾病早期检测的新型代谢物生物标志物

Zhang, Xuan; Liu, Tingjun; Hou, Xianpeng; Hu, Chengzhang; Zhang, Letian; Wang, Shengxuan; Zhang, Qin; Shi, Kerong

Discovery of Novel GR Ligands toward Druggable GR Antagonist Conformations Identified by MD Simulations and Markov State Model Analysis

通过 MD 模拟和马尔可夫状态模型分析确定新型 GR 配体与可用于药物的 GR 拮抗剂构象的发现

Xueping Hu, Jinping Pang, Jintu Zhang, Chao Shen, Xin Chai, Ercheng Wang, Haiyi Chen, Xuwen Wang, Mojie Duan, Weitao Fu, Lei Xu, Yu Kang, Dan Li, Hongguang Xia, Tingjun Hou