日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Cyclin-Dependent Kinase 8 Inhibitor E966-0530-45418 Attenuates Pulmonary Fibrosis In Vitro and In Vivo

细胞周期蛋白依赖性激酶8抑制剂E966-0530-45418在体外和体内均能减轻肺纤维化

Ching-Hsuan Chou,Wei-Jan Huang,Kai-Cheng Hsu,Jui-Yi Hsu,Tony Eight Lin,Chia-Ron Yang

A novel HDAC8 inhibitor H7E exerts retinoprotective effects against glaucomatous injury via ameliorating aberrant Müller glia activation and oxidative stress

新型 HDAC8 抑制剂 H7E 通过改善异常 Müller 胶质细胞活化和氧化应激发挥对青光眼损伤的视网膜保护作用

Liang-Huan Wu, Yu-Wen Cheng, Fan-Li Lin, Kai-Cheng Hsu, Mong-Heng Wang, Jing-Lun Yen, Tsung-Jen Wang, Tony Eight Lin, Yi-Chien Liu, Wei-Jan Huang, George Hsiao

Discovering a novel dual specificity tyrosine-phosphorylation-regulated kinase 1A (DYRK1A) inhibitor and its impact on tau phosphorylation and amyloid-β formation

发现一种新型双特异性酪氨酸磷酸化调节激酶1A (DYRK1A) 抑制剂及其对tau蛋白磷酸化和β-淀粉样蛋白形成的影响

Huang-Ju Tu ,Min-Wu Chao ,Cheng-Chung Lee ,Chao-Shiang Peng ,Yi-Wen Wu ,Tony Eight Lin ,Yu-Wei Chang ,Shih-Chung Yen ,Kai-Cheng Hsu ,Shiow-Lin Pan ,Wei-Chun HuangFu

Synthesis and biological evaluation of ortho-phenyl phenylhydroxamic acids containing phenothiazine with improved selectivity for class IIa histone deacetylases

含吩噻嗪的邻苯基苯异羟肟酸的合成及生物学评价,以提高对 IIa 类组蛋白去乙酰化酶的选择性

Kai-Cheng Hsu, Yun-Yi Huang, Jung-Chun Chu, Yu-Wen Huang, Jing-Lan Hu, Tony Eight Lin, Shih-Chung Yen, Jing-Ru Weng, Wei-Jan Huang

From Sea to Science: Coral Aquaculture for Sustainable Anticancer Drug Development

从海洋到科学:珊瑚养殖助力可持续抗癌药物开发

Hung-Yu Lin, Tsen-Ni Tsai, Kai-Cheng Hsu, Yu-Ming Hsu, Lin-Chien Chiang, Mohamed El-Shazly, Ken-Ming Chang, Yu-Hsuan Lin, Shang-Yi Tu, Tony Eight Lin, Ying-Chi Du, Yi-Chang Liu, Mei-Chin Lu

In silico identification of a novel Cdc2-like kinase 2 (CLK2) inhibitor in triple negative breast cancer

通过计算机模拟鉴定三阴性乳腺癌中新型 Cdc2 样激酶 2 (CLK2) 抑制剂

Cheng-Chiao Huang, Chia-Ming Hsu, Min-Wu Chao, Kai-Cheng Hsu, Tony Eight Lin, Shih-Chung Yen, Huang-Ju Tu, Shiow-Lin Pan

Targeting formyl peptide receptor 1 with anteiso-C13-surfactin for neutrophil-dominant acute respiratory distress syndrome

以反异-C13-表面活性素为靶点,治疗中性粒细胞为主的急性呼吸窘迫综合征

Shun-Chin Yang, Yi-Hsuan Wang, Chiu-Ming Ho, Yung-Fong Tsai, Ping-Jyun Sung, Tony Eight Lin, Tsong-Long Hwang

Design, synthesis, and biological activity of dual monoamine oxidase A and heat shock protein 90 inhibitors, N-Methylpropargylamine-conjugated 4-isopropylresorcinol for glioblastoma

针对胶质母细胞瘤的双单胺氧化酶 A 和热休克蛋白 90 抑制剂 N-甲基炔丙基胺结合的 4-异丙基间苯二酚的设计、合成和生物活性

Hui-Ju Tseng, Suddhasatwa Banerjee, Bin Qian, Mei-Jung Lai, Tung-Yun Wu, Tsung-I Hsu, Tony Eight Lin, Kai-Cheng Hsu, Kuo-Hsiang Chuang, Jing-Ping Liou, Jean C Shih

Urolithin A exhibits a neuroprotective effect against Alzheimer's disease by inhibiting DYRK1A activity

尿石素 A 通过抑制 DYRK1A 活性发挥对阿尔茨海默病的神经保护作用

Huang-Ju Tu, Chih-Jou Su, Chao-Shiang Peng, Tony Eight Lin, Wei-Chun HuangFu, Kai-Cheng Hsu, Tsong-Long Hwang, Shiow-Lin Pan

Pragmatic recruitment of memantine as the capping group for the design of HDAC inhibitors: A preliminary attempt to unravel the enigma of glioblastoma

务实地招募美金刚作为 HDAC 抑制剂设计的封端基团:初步尝试解开胶质母细胞瘤之谜

Kunal Nepali, Tsung-I Hsu, Chien-Ming Hsieh, Wei-Lun Lo, Mei-Jung Lai, Kai-Cheng Hsu, Tony Eight Lin, Jian-Ying Chuang, Jing-Ping Liou