日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A new therapeutic approach for Parkinson's disease: dual targeting of α-Synuclein aggregation and microglial function by the novel immunomodulator 3-Monothiopomalidomide

帕金森病的新疗法:新型免疫调节剂3-单硫代马来酸双重靶向α-突触核蛋白聚集和小胶质细胞功能

Palmas, Maria Francesca; Aminzadeh, Khosro; Runfola, Matteo; Parekh, Pathik; Porcedda, Clara; Tweedie, David; Casula, Luca; Cardia, Maria Cristina; Marongiu, Jacopo; Etzi, Michela; Lai, Francesco; Serra, Marcello; Pisanu, Augusta; Sogos, Valeria; De Simone, Alfonso; Kim, Dong Seok; Greig, Nigel H; Carta, Anna R

Host-directed treatments for tuberculous meningitis: A multi-platform approach across mouse and human models

针对结核性脑膜炎的宿主导向治疗:跨小鼠和人类模型的多平台方法

Jain, Sanjay; Gonzalez, Carlos Ruiz; Singh, Medha; Leon, Yuderleys Masias; Chen, Xueyi; Sarhan, Mona; Martinez-Martinez, Yazmin; Patel, Shruti; Shambles, Madelynn; Villabona-Rueda, Andres; Lissit, Kadia; Tweedie, David; Scerba, Michael; Bishai, William; Artemov, Dmitri; Xu, Jinchong; D'Alessio, Franco; Hafner, Richard; Greig, Nigel; Manion, Maura; Sereti, Irini

Anti-inflammatory and pro-proliferative effects of fasudil in human trisomy 21 neural progenitor cells

法舒地尔对人类21三体神经祖细胞的抗炎和促增殖作用

Baxter, Laura L; Lee, Sarah E; Fuentes, Kevin A; Mosley, Iman A; Raymond, Jonathan D; Guedj, Faycal; Zhou, Di; Slonim, Donna K; Glotfelty, Elliot J; Tweedie, David; Grieg, Nigel H; Bianchi, Diana W

Enhanced Bioavailability of a Thionated IMiD Derivative Nanosuspension for Parkinson's Disease Targeting α-Synuclein

硫代IMiD衍生物纳米悬浮液靶向α-突触核蛋白,增强其在帕金森病治疗中的生物利用度

Casula, Luca; Palmas, Maria Francesca; Cardia, Maria Cristina; Valenti, Donatella; Pini, Elena; Etzi, Michela; Marceddu, Salvatore; Sinico, Chiara; Tweedie, David; Greig, Nigel H; Kim, Dong Seok; Carta, Anna Rosa; Lai, Francesco

3-Monothiopomalidomide, a new immunomodulatory imide drug (IMiD), blunts inflammation and mitigates ischemic stroke in the rat.

3-单硫代马来度胺是一种新型免疫调节酰亚胺药物(IMiD),可减轻炎症并缓解大鼠缺血性中风

Chen Kai-Yun, Hsueh Shih-Chang, Parekh Pathik, Batsaikhan Buyandelger, Tweedie David, Luo Weiming, Patel Chirag, Chiang Yung-Hsiao, Bambakidis Nicholas, Hoffer Barry J, Huang Chi-Zong, Yu Seong-Jin, Wu Kuo-Jen, Wang Yun, Hong Eunji, Kim Dong Seok, Greig Nigel H

Correction: Batsaikhan et al. Post-Injury Neuroprotective Effects of the Thalidomide Analog 3,6'-Dithiothalidomide on Traumatic Brain Injury. Int. J. Mol. Sci. 2019, 20, 502

更正:Batsaikhan 等人,《沙利度胺类似物 3,6'-二硫代沙利度胺对创伤性脑损伤的损伤后神经保护作用》,《国际分子科学杂志》,2019 年,第 20 卷,第 502 页。

Batsaikhan, Buyandelger; Wang, Jing-Ya; Scerba, Michael T; Tweedie, David; Greig, Nigel H; Miller, Jonathan P; Hoffer, Barry J; Lin, Chih-Tung; Wang, Jia-Yi

Pharmacological characterization and preclinical evaluation of 11h: a novel, brain-penetrant PDE4 inhibitor for neurological disorders

11h 的药理学特性及临床前评价:一种新型的、可穿透血脑屏障的 PDE4 抑制剂,用于治疗神经系统疾病

Lackovic, Jacob; Dey, Sougata; Ward, Sara Jane; Greig, Nigel H; Tweedie, David; Beiranvand, Nassim; Saini, Uksha; Chatterjee, Dev; Varadhachary, Atul

Sitagliptin elevates plasma and CSF incretin levels following oral administration to nonhuman primates: relevance for neurodegenerative disorders

口服西格列汀后,非人灵长类动物血浆和脑脊液中的肠促胰岛素水平升高:与神经退行性疾病的相关性

Li, Yazhou; Vaughan, Kelli L; Wang, Yun; Yu, Seong-Jin; Bae, Eun-Kyung; Tamargo, Ian A; Kopp, Katherine O; Tweedie, David; Chiang, Cheng-Chuan; Schmidt, Keith T; Lahiri, Debomoy K; Tones, Michael A; Zaleska, Margaret M; Hoffer, Barry J; Mattison, Julie A; Greig, Nigel H

2-(Piperidin-3-yl)phthalimides reduce classical markers of cellular inflammation in LPS-challenged RAW 264.7 cells and also demonstrate potentially relevant sigma and serotonin receptor affinity in membrane preparations

2-(哌啶-3-基)邻苯二甲酰亚胺可降低LPS刺激的RAW 264.7细胞中经典的细胞炎症标志物,并且在膜制备物中也表现出潜在的相关σ受体和血清素受体亲和力。

Scerba, Michael T; Tweedie, David; Greig, Nigel H

A New Generation of IMiDs as Treatments for Neuroinflammatory and Neurodegenerative Disorders

新一代免疫调节剂作为神经炎症和神经退行性疾病的治疗药物

Kopp, Katherine O; Greer, Margaret E; Glotfelty, Elliot J; Hsueh, Shih-Chang; Tweedie, David; Kim, Dong Seok; Reale, Marcella; Vargesson, Neil; Greig, Nigel H