日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Pan-TEAD Inhibitors That Disrupt YAP-TEAD Interaction as a Potential Therapy for Gastric Cancers and Mutant KRAS and EGFR Lung Cancers

发现可破坏YAP-TEAD相互作用的泛TEAD抑制剂,有望成为胃癌以及KRAS和EGFR突变型肺癌的潜在疗法

Kumar, Ramesh; Thian, Joanne; Toh, Joel D W; Farzana, Noorul; Sun, Jialin; Kang, CongBao; Low, Suet Mei Crystal; Wee, Sheena; Lim, Zijie; Gunaratne, Jayantha; Loh, Hui Mun; Kannan, Srinivasaraghavan; Verma, Chandra S; Chakraborty, Sayan; Hong, Wanjin

Author Correction: Design-rules for stapled peptides with in vivo activity and their application to Mdm2/X antagonists

作者更正:具有体内活性的肽链设计规则及其在 Mdm2/X 拮抗剂中的应用

Chandramohan, Arun; Josien, Hubert; Yuen, Tsz Ying; Duggal, Ruchia; Spiegelberg, Diana; Yan, Lin; Juang, Yu-Chi Angela; Ge, Lan; Aronica, Pietro G; Kaan, Hung Yi Kristal; Lim, Yee Hwee; Peier, Andrea; Sherborne, Brad; Hochman, Jerome; Lin, Songnian; Biswas, Kaustav; Nestor, Marika; Verma, Chandra S; Lane, David P; Sawyer, Tomi K; Garbaccio, Robert; Henry, Brian; Kannan, Srinivasaraghavan; Brown, Christopher J; Johannes, Charles W; Partridge, Anthony W

Conserved leucine-rich repeat proteins in the adhesive projectile slime of velvet worms

天鹅绒虫粘性喷射黏液中保守的富含亮氨酸重复序列蛋白

Hu, Zhaolong; Baer, Alexander; Hering, Lars; de Sena Oliveira, Ivo; Poulhazan, Alexandre; Browne, Darren C; Guo, Xue; Perrin, Quentin Moana; Sobota, Radoslaw M; Hoon, Shawn; Mayer, Georg; Kannan, Srinivasaraghavan; Verma, Chandra S; Harrington, Matthew J; Miserez, Ali

Responsiveness of different MET tumour alterations to type I and type II MET inhibitors.

不同MET肿瘤改变对I型和II型MET抑制剂的反应性

Murciano-Goroff Yonina R, Foglizzo Valentina, Chang Jason, Rekhtman Natasha, Sisk Ann Elizabeth, Gibson Jamie, Judka Lia, Clemens Kristen, Roa Paola, Ahmed Shaza Sayed, Bremer Nicole V, Binaco Courtney Lynn, Muzungu Sherifah Kemigisha, Rodriguez Estelamari, Merrill Madeline, Sgroe Erica, Repetto Matteo, Stadler Zsofia K, Berger Michael F, Yu Helena A, Toska Eneda, Kannan Srinivasaraghavan, Verma Chandra S, Drilon Alexander, Cocco Emiliano

Systematic benchmarking of 13 AI methods for predicting cyclic peptide membrane permeability

对 13 种预测环肽膜渗透性的 AI 方法进行系统基准测试

Liu, Wei; Li, Jianguo; Verma, Chandra S; Lee, Hwee Kuan

Exploring non-alcohol-based disinfectant: virucidal efficacy of arginine and Zinc chloride against feline calicivirus

探索非酒精类消毒剂:精氨酸和氯化锌对猫杯状病毒的杀病毒功效

Kong Li Ying, Marcella; Masirevic, Srdan; Tan, Yong Wah; Marzinek, Jan K; Fox, Stephen John; Verma, Chandra S; Bond, Peter J; Ishida, Yoshiki; Liu, Jiquan; Chua, Chun Song; Chu, Justin Jang Hann

Unravelling the dynamics of the maturation protein in MS2 bacteriophage via molecular simulations

通过分子模拟揭示MS2噬菌体成熟蛋白的动态变化

Masirevic, Srdan; Marzinek, Jan K; Liu, Jiquan; Maupin, C Mark; Fox, Stephen J; Verma, Chandra S; Bond, Peter J

Desmoplakin CSM models unravel mechanisms regulating the binding to intermediate filaments and putative therapeutics for cardiocutaneous diseases

桥粒蛋白CSM模型揭示了调控其与中间丝结合的机制,并为心皮肤疾病的治疗提供了潜在方法。

Badowski, Cedric; Benny, Paula; Verma, Chandra S; Lane, E Birgitte

Rarγ -Foxa1 signaling promotes luminal identity in prostate progenitors and is disrupted in prostate cancer

Rarγ-Foxa1信号通路促进前列腺祖细胞的管腔特性,并在前列腺癌中受到破坏。

Felice, Dario De; Alaimo, Alessandro; Bressan, Davide; Genovesi, Sacha; Marmocchi, Elisa; Annesi, Nicole; Beccaceci, Giulia; Dalfovo, Davide; Cutrupi, Federico; Foletto, Veronica; Lorenzoni, Marco; Gandolfi, Francesco; Kannan, Srinivasaraghavan; Verma, Chandra S; Vasciaveo, Alessandro; Shen, Michael M; Romanel, Alessandro; Chiacchiera, Fulvio; Cambuli, Francesco; Lunardi, Andrea

Stitched peptides as potential cell permeable inhibitors of oncogenic DAXX protein.

拼接肽作为致癌DAXX蛋白的潜在细胞渗透性抑制剂

Jelinska Clare, Kannan Srinivasaraghavan, Frosi Yuri, Ramlan Siti Radhiah, Winnerdy Fernaldo, Lakshminarayanan Rajamani, Johannes Charles W, Brown Christopher J, Phan Anh-Tuan, Rhodes Daniela, Verma Chandra S