日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New series of pentamidine-based 1,2,3-triazole-diaryl-hydrazones: design, synthesis, and evaluation of their leishmanicidal activity and mechanism of action against Leishmania (L.) amazonensis

新型戊烷脒基1,2,3-三唑二芳基腙类化合物的设计、合成及其对亚马逊利什曼原虫(Leishmania (L.) amazonensis)的杀利什曼原虫活性和作用机制评价

Espuri Sepini, Patrícia F; Gontijo, Vanessa Silva; Tavares, Laiane Mota; Souza, Leonardo Maciel; Souza, Thalles H F; Couto, Dyecika S; Nunes, Juliana B; Ribeiro, Catarina Azevedo; da Silva Cravo, Sara M Mendonça; Zavan, Bruno; Alves, Marina A; Souza, Hygor M R; Ionta, Marisa; Sousa, Maria Emília; Peloso, Eduardo F; Marques, Marcos J; Viegas, Claudio Jr

Monoamine Oxidase Inhibitors in Drug Discovery Against Parkinson's Disease: An Update

单胺氧化酶抑制剂在帕金森病药物研发中的应用:最新进展

Ribeiro, Luana Vergueiro; Massuda, Larissa Emika; Gontijo, Vanessa Silva; Viegas, Claudio Jr

Novel Multifunctional Cannabidiol-Based Analogues with In Silico, In Vitro, and In Vivo Anti-SARS-CoV-2 Effect

新型多功能大麻二酚类似物在计算机模拟、体外和体内均显示出抗SARS-CoV-2活性

Franco, Graziella Dos Reis Rosa; Gontijo, Vanessa Silva; Viegas, Flávia Pereira Dias; Silva, Matheus de Freitas; Ortiz, Cindy Juliet Cristancho; Damásio, Caio Miranda; Silva, Isabella Marie Fernandes; Campos, Thâmara Gaspar; Reis, Erik Vinicius de Sousa; Clarindo, Felipe Alves; Moraes, Thaís de Fátima Silva; Silva, Matheus Müller Pereira da; França, Patrícia Ribeiro de Carvalho; Guedes, Isabella Alvim; Dardenne, Laurent Emmanuel; Reis, Jordana Grazziela Alves Coelho Dos; Fernandes, Patrícia Dias; Viegas, Claudio Jr

Design, Synthesis, and Evaluation of Antinociceptive Properties of Novel CBD-Based Terpene-Cinnamoyl-Acyl-Hydrazone Analogues.

新型CBD基萜烯-肉桂酰-酰基-腙类似物的设计、合成及镇痛性能评价

de Souza Mikaela Lucinda, de Paiva João Pedro Barros, Franco Graziella Dos Reis Rosa, Gontijo Vanessa Silva, Alves Marina Amaral, de Souza Hygor Marcos Ribeiro, Lontra Anna Carolina Pereira, de Oliveira Eduardo Araújo, Giorno Thaís Biondino Sardella, Guedes Isabella Alvim, Dardenne Laurent Emmanuel, Fernandes Patrícia Dias, Viegas Claudio Jr

Curcumin-like Compound Inhibits Proliferation of Adenocarcinoma Cells by Inducing Cell Cycle Arrest and Senescence.

姜黄素样化合物通过诱导细胞周期停滞和衰老来抑制腺癌细胞的增殖

Fonseca Rafael, Louzano Yasmin Dos Santos, Ortiz Cindy Juliet Cristancho, Silva Matheus de Freitas, Felix Maria Luiza Vieira, Ferreira-Silva Guilherme Álvaro, Caixeta Ester Siqueira, Zavan Bruno, Viegas Claudio Jr, Ionta Marisa

Simarouba berteroana Krug & Urb. Extracts and Fractions Possess Anthelmintic Activity Against Eggs and Larvae of Multidrug-Resistant Haemonchus contortus

Simarouba berteroana Krug & Urb. 提取物和组分对多重耐药性捻转血矛线虫的卵和幼虫具有驱虫活性

Espino Ureña, Marcos Javier; Katchborian-Neto, Albert; Garcez Neto, José Ribamar; da Silva Lopes, Francisco Flávio; de Morais, Selene Maia; Narciso Dos Reis, Vitor Eduardo; Cardoso, Carmen Lúcia; Beserra de Oliveira, Lorena Mayana; Viegas, Claudio Jr; Marques, Marcos José; Correia Ribeiro, Wesley Lyeverton

Potential Impact of the Multi-Target Drug Approach in the Treatment of Some Complex Diseases

多靶点药物疗法在某些复杂疾病治疗中的潜在影响

Makhoba, Xolani H; Viegas, Claudio Jr; Mosa, Rebamang A; Viegas, Flávia P D; Pooe, Ofentse J

Editorial: Oxidative Stress: How Has It Been Considered in the Design of New Drug Candidates for Neurodegenerative Diseases?

社论:氧化应激:在设计治疗神经退行性疾病的新药候选药物时,如何考虑氧化应激?

Viegas, Claudio Jr; Fraga, Carlos A Manssour; Sousa, Maria Emilia; Tarozzi, Andrea

PQM130, a Novel Feruloyl-Donepezil Hybrid Compound, Effectively Ameliorates the Cognitive Impairments and Pathology in a Mouse Model of Alzheimer's Disease

PQM130,一种新型的阿魏酰-多奈哌齐杂合化合物,能有效改善阿尔茨海默病小鼠模型的认知障碍和病理变化。

Morroni, Fabiana; Sita, Giulia; Graziosi, Agnese; Ravegnini, Gloria; Molteni, Raffaella; Paladini, Maria Serena; Dias, Kris Simone Tranches; Dos Santos, Ariele Faria; Viegas, Claudio Jr; Camps, Ihosvany; Pruccoli, Letizia; Tarozzi, Andrea; Hrelia, Patrizia

Multi-Target Directed Drugs: A Modern Approach for Design of New Drugs for the treatment of Alzheimer's Disease

多靶点靶向药物:治疗阿尔茨海默病新药设计的现代方法

Dias, Kris Simone Tranches; Viegas, Claudio Jr