日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Retraction Note: Kinase profiling of liposarcomas using RNAi and drug screening assays identified druggable targets

撤稿声明:利用RNAi和药物筛选方法对脂肪肉瘤进行激酶谱分析,鉴定出可成药靶点。

Kanojia, Deepika; Garg, Manoj; Martinez, Jacqueline; M T, Anand; B Luty, Samuel; B Doan, Ngan; W Said, Jonathan; Forscher, Charles; W Tyner, Jeffrey; Koeffler, H Phillip

Mapping the proteogenomic landscape enables prediction of drug response in acute myeloid leukemia

绘制蛋白质组学图谱可预测急性髓系白血病的药物反应

James C Pino, Camilo Posso, Sunil K Joshi, Michael Nestor, Jamie Moon, Joshua R Hansen, Chelsea Hutchinson-Bunch, Marina A Gritsenko, Karl K Weitz, Kevin Watanabe-Smith, Nicola Long, Jason E McDermott, Brian J Druker, Tao Liu, Jeffrey W Tyner, Anupriya Agarwal, Elie Traer, Paul D Piehowski, Cristina

Ubiquitin-specific protease 7 inhibitors reveal a differentiated mechanism of p53-driven anti-cancer activity

泛素特异性蛋白酶 7 抑制剂揭示 p53 驱动抗癌活性的差异化机制

Alan S Futran, Tao Lu, Katherine Amberg-Johnson, Jiayi Xu, Xiaoxiao Yang, Saidi He, Sarah Boyce, Jeffrey A Bell, Robert Pelletier, Takao Suzuki, Xianhai Huang, Heng Qian, Liping Fang, Li Xing, Zhaowu Xu, Stephen E Kurtz, Jeffrey W Tyner, Wayne Tang, Tao Guo, Karen Akinsanya, David Madge, Kristian K

Disruption of the MYC Superenhancer Complex by Dual Targeting of FLT3 and LSD1 in Acute Myeloid Leukemia

急性髓系白血病中FLT3和LSD1双重靶向破坏MYC超级增强子复合物

William M Yashar # ,Brittany M Curtiss #,Daniel J Coleman,Jake VanCampen,Garth Kong,Jommel Macaraeg,Joseph Estabrook,Emek Demir ,Nicola Long,Daniel Bottomly,Shannon K McWeeney,Jeffrey W Tyner ,Brian J Druker ,Julia E Maxson,Theodore P Braun

Treatment for ovarian clear cell carcinoma with combined inhibition of WEE1 and ATR

联合抑制 WEE1 和 ATR 治疗卵巢透明细胞癌

Wenwen Chien, Jeffrey W Tyner, Sigal Gery, Yueyuan Zheng, Li-Yan Li, Mohan Shankar Gopinatha Pillai, Chehyun Nam, Neil A Bhowmick, De-Chen Lin, H Phillip Koeffler

Tuft cells mediate commensal remodeling of the small intestinal antimicrobial landscape

簇细胞介导小肠抗菌景观的共生重塑

Connie Fung, Lisa M Fraser, Gabriel M Barrón, Matthew B Gologorsky, Samantha N Atkinson, Elias R Gerrick, Michael Hayward, Jennifer Ziegelbauer, Jessica A Li, Katherine F Nico, Miles D W Tyner, Leila B DeSchepper, Amy Pan, Nita H Salzman, Michael R Howitt

Integrative analysis of drug response and clinical outcome in acute myeloid leukemia

急性髓系白血病药物反应与临床结果的综合分析

Daniel Bottomly ,Nicola Long ,Anna Reister Schultz ,Stephen E Kurtz ,Cristina E Tognon ,Kara Johnson ,Melissa Abel ,Anupriya Agarwal ,Sammantha Avaylon ,Erik Benton ,Aurora Blucher ,Uma Borate ,Theodore P Braun ,Jordana Brown ,Jade Bryant ,Russell Burke ,Amy Carlos ,Bill H Chang ,Hyun Jun Cho ,Stephen Christy ,Cody Coblentz ,Aaron M Cohen ,Amanda d'Almeida ,Rachel Cook ,Alexey Danilov ,Kim-Hien T Dao ,Michie Degnin ,James Dibb ,Christopher A Eide ,Isabel English ,Stuart Hagler ,Heath Harrelson ,Rachel Henson ,Hibery Ho ,Sunil K Joshi ,Brian Junio ,Andy Kaempf ,Yoko Kosaka ,Ted Laderas ,Matt Lawhead ,Hyunjung Lee ,Jessica T Leonard ,Chenwei Lin ,Evan F Lind ,Selina Qiuying Liu ,Pierrette Lo ,Marc M Loriaux ,Samuel Luty ,Julia E Maxson ,Tara Macey ,Jacqueline Martinez ,Jessica Minnier ,Andrea Monteblanco ,Motomi Mori ,Quinlan Morrow ,Dylan Nelson ,Justin Ramsdill ,Angela Rofelty ,Alexandra Rogers ,Kyle A Romine ,Peter Ryabinin ,Jennifer N Saultz ,David A Sampson ,Samantha L Savage ,Robert Schuff ,Robert Searles ,Rebecca L Smith ,Stephen E Spurgeon ,Tyler Sweeney ,Ronan T Swords ,Aashis Thapa ,Karina Thiel-Klare ,Elie Traer ,Jake Wagner ,Beth Wilmot ,Joelle Wolf ,Guanming Wu ,Amy Yates ,Haijiao Zhang ,Christopher R Cogle ,Robert H Collins ,Michael W Deininger ,Christopher S Hourigan ,Craig T Jordan ,Tara L Lin ,Micaela E Martinez ,Rachel R Pallapati ,Daniel A Pollyea ,Anthony D Pomicter ,Justin M Watts ,Scott J Weir ,Brian J Druker ,Shannon K McWeeney ,Jeffrey W Tyner

Genome-wide CRISPR screen identifies regulators of MAPK and MTOR pathways mediating sorafenib resistance in acute myeloid leukemia

全基因组 CRISPR 筛选可识别出介导急性髓系白血病索拉非尼耐药性的 MAPK 和 MTOR 通路调节剂

Alisa Damnernsawad, Daniel Bottomly, Stephen E Kurtz, Christopher A Eide, Shannon K McWeeney, Jeffrey W Tyner, Tamilla Nechiporuk

Luxeptinib (CG-806) Targets FLT3 and Clusters of Kinases Operative in Acute Myeloid Leukemia

Luxeptinib (CG-806) 靶向作用于急性髓系白血病的 FLT3 和激酶簇

William G Rice, Stephen B Howell, Hongying Zhang, Nasrin Rastgoo, Andrea Local, Stephen E Kurtz, Pierrette Lo, Daniel Bottomly, Beth Wilmot, Shannon K McWeeney, Brian J Druker, Jeffrey W Tyner

Functional proteomics of patient derived head and neck squamous cell carcinoma cells reveal novel applications of trametinib

患者来源的头颈部鳞状细胞癌细胞的功能蛋白质组学揭示了曲美替尼的新应用

Myles Vigoda, Chase Mathieson, Nathaniel Evans, Carolyn Hale, Jennifer Jennings, Olivia Lucero, Sophia Jeng, Daniel Bottomly, Daniel Clayburgh, Peter Andersen, Ryan Li, Daniel Petrisor, Jeffrey W Tyner, Shannon McWeeney, Molly Kulesz-Martin