日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advances in Therapeutic Antibody Discovery and Development Targeting G Protein-Coupled Receptors

靶向G蛋白偶联受体的治疗性抗体发现与开发进展

Hutchings, Catherine J; Ünsal, Serbülent; Rappas, Mathieu; Barnes, Matthew; Waldhoer, Maria; Holland, Ben; Culka, Martin

A GLP-1 analogue optimized for cAMP-biased signaling improves weight loss in obese mice.

针对 cAMP 偏向信号传导优化的 GLP-1 类似物可改善肥胖小鼠的体重减轻

Douros Jonathan D, Novikoff Aaron, DuBois Barent, Rohlfs Rebecca, Mokrosinski Jacek, Hogendorf Wouter F J, Augustin Robert, Merkestein Myrte, Egaa Martini Lene Brandt, Linderoth Lars, Gerrard Elliot, Kodra Janos Tibor, Norlin Jenny, Roed Nikolaj Kulahin, Oldenburger Anouk, Mowery Stephanie A, Waldhoer Maria, Perez-Tilve Diego, Finan Brian, Reedtz-Runge Steffen, Müller Timo D, Knerr Patrick J

Reply to: How carvedilol does not activate β(2)-adrenoceptors

回复:卡维地洛为何不激活β(2)-肾上腺素受体

Kostenis, Evi; Gomeza, Jesus; Miess-Tanneberg, Elke; Blum, Nina Kathleen; Benkel, Tobias; Chevigné, Andy; Hoffmann, Carsten; Kolb, Peter; Nikolaev, Viacheslav; Waldhoer, Maria; Szpakowska, Martyna; Inoue, Asuka; Schulz, Stefan

The European Research Network on Signal Transduction (ERNEST): Toward a Multidimensional Holistic Understanding of G Protein-Coupled Receptor Signaling

欧洲信号转导研究网络(ERNEST):迈向对G蛋白偶联受体信号传导的多维整体理解

Sommer, Martha E; Selent, Jana; Carlsson, Jens; De Graaf, Chris; Gloriam, David E; Keseru, Gyorgy M; Kosloff, Mickey; Mordalski, Stefan; Rizk, Aurelien; Rosenkilde, Mette M; Sotelo, Eddy; Tiemann, Johanna K S; Tobin, Andrew; Vardjan, Nina; Waldhoer, Maria; Kolb, Peter

A Focus on Unusual ECL2 Interactions Yields β(2) -Adrenergic Receptor Antagonists with Unprecedented Scaffolds

聚焦于不寻常的ECL2相互作用,获得了具有前所未有的骨架结构的β(2)-肾上腺素能受体拮抗剂

Scharf, Magdalena M; Zimmermann, Mirjam; Wilhelm, Florian; Stroe, Raimond; Waldhoer, Maria; Kolb, Peter

Gα13 mediates human cytomegalovirus-encoded chemokine receptor US28-induced cell death in melanoma

Gα13介导人巨细胞病毒编码的趋化因子受体US28诱导的黑色素瘤细胞死亡

Joshi, Shripad; Wels, Christian; Beham-Schmid, Christine; Fukunaga-Kalabis, Mizuho; Holmen, Sheri L; Otte, Marcus; Herlyn, Meenhard; Waldhoer, Maria; Schaider, Helmut

Functional consequences of glucagon-like peptide-1 receptor cross-talk and trafficking

胰高血糖素样肽-1受体串扰和转运的功能后果

Roed, Sarah Noerklit; Nøhr, Anne Cathrine; Wismann, Pernille; Iversen, Helle; Bräuner-Osborne, Hans; Knudsen, Sanne Moeller; Waldhoer, Maria

Minireview: recent developments in the physiology and pathology of the lysophosphatidylinositol-sensitive receptor GPR55

小综述:溶血磷脂酰肌醇敏感受体GPR55的生理学和病理学最新进展

Henstridge, Christopher M; Balenga, Nariman A B; Kargl, Julia; Andradas, Clara; Brown, Andrew J; Irving, Andrew; Sanchez, Cristina; Waldhoer, Maria

Opioid-receptor-heteromer-specific trafficking and pharmacology

阿片受体异源体特异性转运和药理学

van Rijn, Richard M; Whistler, Jennifer L; Waldhoer, Maria

G protein-coupled receptor-associated sorting protein 1 regulates the postendocytic sorting of seven-transmembrane-spanning G protein-coupled receptors

G蛋白偶联受体相关分选蛋白1调节七次跨膜G蛋白偶联受体的内吞后分选

Moser, Elisabeth; Kargl, Julia; Whistler, Jennifer L; Waldhoer, Maria; Tschische, Pia