日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Expanding the toolbox to develop IAP-based degraders of TEAD transcription factors.

扩展工具箱,开发基于 IAP 的 TEAD 转录因子降解剂。

Gupta Nishma, Trainor Nicole, Radwan Mona, Nguyen Stephanie, Duncan Luke, Tang Andrew X, Beveridge Julia, Silke Natasha, Yousef Jumana, Bilgilier Ceren, Wachter Johannes, Greb Peter, Jandova Zuzana, Eliaš Ján, Kopf Sara, Gerstberger Thomas, Stolt-Bergner Peggy, Braun Nina, Weinstabl Harald, McConnell Darryl B, Mauri Federico, Lucet Isabelle S, Silke John, Chessum Nicola E A, Roy Michael J

Frustration in the protein-protein interface plays a central role in the cooperativity of PROTAC ternary complexes

蛋白质-蛋白质界面处的相互作用受阻在PROTAC三元复合物的协同作用中起着核心作用。

Ma, Ning; Bhattacharya, Supriyo; Muk, Sanychen; Jandova, Zuzana; Schmalhorst, Philipp S; Ghosh, Soumadwip; Le, Keith; Diers, Emelyne; Trainor, Nicole; Farnaby, William; Roy, Michael J; Kofink, Christiane; Greb, Peter; Weinstabl, Harald; Ciulli, Alessio; Bader, Gerd; Sankar, Kyra; Bergner, Andreas; Vaidehi, Nagarajan

Drugit: crowd-sourcing molecular design of non-peptidic VHL binders

Drugit:众包非肽类VHL结合剂的分子设计

Scott, Thomas; Smethurst, Christian Alan Paul; Westermaier, Yvonne; Mayer, Moriz; Greb, Peter; Kousek, Roland; Biberger, Tobias; Bader, Gerd; Jandova, Zuzana; Schmalhorst, Philipp S; Fuchs, Julian E; Magarkar, Aniket; Hoenke, Christoph; Gerstberger, Thomas; Combs, Steven A; Pape, Richard; Phul, Saksham; Kothiwale, Sandeepkumar; Bergner, Andreas; Waterson, Alex G; Weinstabl, Harald; McConnell, Darryl B; Meiler, Jens; Böttcher, Jark; Moretti, Rocco

At the Nexus Between Epigenetics and Senescence: The Effects of Senolytic (BI01) Administration on DNA Methylation Clock Age and the Methylome in Aged and Regenerated Skeletal Muscle.

表观遗传学与衰老之间的联系:衰老细胞清除剂 (BI01) 给药对衰老和再生骨骼肌中 DNA 甲基化时钟年龄和甲基化组的影响

Chambers Toby L, Wells Jaden, Koopmans Pieter Jan, Morena Francielly, Malik Zain B, Greene Nicholas P, Filareto Antonio, Franti Michael, Sini Patrizia, Weinstabl Harald, Brooke Robert T, Milčiūtė Milda, Gordevičius Juozas, Horvath Steve, Wen Yuan, Dungan Cory M, Murach Kevin A

Synthesis of Complex Tetracyclic Fused Scaffolds Enabled by (3 + 2) Cycloaddition

利用 (3 + 2) 环加成反应合成复杂的四环稠合骨架

Porte, Vincent; van Veen, Branca C; Zhang, Haoqi; Piacentini, Paolo; Matheu, Sergio Armentia; Woolford, Sophie; Sokol, Kevin R; Shaaban, Saad; Weinstabl, Harald; Maulide, Nuno

Synthesis of a (13)C-methylene-labeled isoleucine precursor as a useful tool for studying protein side-chain interactions and dynamics

合成(13)C-亚甲基标记的异亮氨酸前体作为研究蛋白质侧链相互作用和动力学的有用工具

Höfurthner, Theresa; Toscano, Giorgia; Kontaxis, Georg; Beier, Andreas; Mayer, Moriz; Geist, Leonhard; McConnell, Darryl B; Weinstabl, Harald; Lichtenecker, Roman; Konrat, Robert

Electrochemical Umpolung C-H Functionalization of Oxindoles

氧吲哚的电化学极性反转CH官能化

Pastor, Miryam; Vayer, Marie; Weinstabl, Harald; Maulide, Nuno

Targeted Synthesis of Complex Spiro[3H-indole-3,2'-pyrrolidin]-2(1H)-ones by Intramolecular Cyclization of Azomethine Ylides: Highly Potent MDM2-p53 Inhibitors

通过亚胺叶立德的分子内环化靶向合成复杂的螺[3H-吲哚-3,2'-吡咯烷]-2(1H)-酮:高效的MDM2-p53抑制剂

Gollner, Andreas; Weinstabl, Harald; Fuchs, Julian E; Rudolph, Dorothea; Garavel, Geraldine; Hofbauer, Karin S; Karolyi-Oezguer, Jale; Gmaschitz, Gerhard; Hela, Wolfgang; Kerres, Nina; Grondal, Elisabeth; Werni, Patrick; Ramharter, Juergen; Broeker, Joachim; McConnell, Darryl B

Total synthesis of (+)-linoxepin by utilizing the Catellani reaction

利用卡特拉尼反应全合成(+)-利诺昔平

Weinstabl, Harald; Suhartono, Marcel; Qureshi, Zafar; Lautens, Mark