日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A general assay platform to study protein pharmacology using ligand-dependent structural dynamics.

利用配体依赖性结构动力学研究蛋白质药理学的通用检测平台

Ciulla Daniel A, Dranchak Patricia K, Aitha Mahesh, van Neer Renier H P, Shah Divia, Tharakan Ravi, Wilson Kelli M, Wang Yuhong, Braisted John C, Inglese James

AI-driven discovery of synergistic drug combinations against pancreatic cancer.

利用人工智能发现对抗胰腺癌的协同药物组合

Pourmousa Mohsen, Jain Sankalp, Barnaeva Elena, Jin Wengong, Hochuli Joshua, Itkin Zina, Maxfield Travis, Melo-Filho Cleber, Thieme Andrew, Wilson Kelli, Klumpp-Thomas Carleen, Michael Sam, Southall Noel, Jaakkola Tommi, Muratov Eugene N, Barzilay Regina, Tropsha Alexander, Ferrer Marc, Zakharov Alexey V

A review of diffuse hemispheric glioma, H3 G34-mutant disease development, DNA repair, microenvironment, and treatments on the horizon

弥漫性半球胶质瘤、H3 G34突变疾病发展、DNA修复、微环境及未来治疗进展综述

Crowell, Cameron; Zhu, Ziwen; Li, Yingxiang; Varela, Maria L; Ostrom, Quinn; Cimino, Patrick J; Patel, Sohil H; Baker, Suzanne J; Bettegowda, Chetan; Noushmehr, Houtan; Kleinman, Claudia L; Canty, Laura; Cruzeiro, Gustavo Alencastro Veiga; Nellan, Anandani; Becher, Oren; Davidson, Tom B; Hambardzumyan, Dolores; Green, Adam; Thorne, Robert; Wilson, Kelli; Theeler, Brett; Gregory, Jason; Mathen, Peter; Biassou, Nadia; McThenia, Sheila; Erker, Craig; Galvin, Robert; Soldatos, Ariane; Lowenstein, Pedro R; Castro, Maria G; Jackson, Sadhana

Large-scale human myeloma cell line small molecule compound screen dataset

大规模人类骨髓瘤细胞系小分子化合物筛选数据集

Hughitt, V Keith; Simmons, John K; Gorjifard, Sayeh; Michalowski, Aleksandra; Wilson, Kelli; Zhang, Xiaohu; Shinn, Paul; Klumpp-Thomas, Carleen; McKnight, Crystal; Itkin, Zina; Chen, Lu; Michael, Sam; Keats, Jonathan; Thomas, Craig; Mock, Beverly A

Targeting NAD+ Metabolism Vulnerability in FH-Deficient Hereditary Leiomyomatosis and Renal Cell Carcinoma with the Novel NAMPT Inhibitor OT-82.

利用新型 NAMPT 抑制剂 OT-82 靶向 FH 缺陷型遗传性平滑肌瘤病和肾细胞癌中的 NAD+ 代谢脆弱性

Najera Susana S, Ricketts Christopher J, Schmidt Laura S, Medina Julia I, Saito Keita, Ileva Lilia, Brender Jeffrey R, James Amy M, Peer Cody J, Gouker Brad, Karim Baktiar O, Chernova Olga, Wells Catherine, Wei Ming-Hui, Yang Youfeng, Zhang Xiaohu, Klumpp-Thomas Carleen, Travers Jameson, Chen Lu, Wilson Kelli M, Issaq Sameer H, Figg William D, Difilippantonio Simone, Kalen Joseph D, Krishna Murali C, Thomas Craig J, Ceribelli Michele, Heske Christine M, Crooks Daniel R, Meier Jordan L

The Kinase Inhibitor GNF-7 Is Synthetically Lethal in Topoisomerase 1-Deficient Ewing Sarcoma.

激酶抑制剂 GNF-7 在拓扑异构酶 1 缺陷型尤文氏肉瘤中具有合成致死性

Sayers Carly M, Carter Morgan B, Lei Haiyan, Mendoza Arnulfo, Shema Steven, Zhang Xiaohu, Wilson Kelli, Chen Lu, Klumpp-Thomas Carleen, Thomas Craig J, Heske Christine M, Shern Jack F

An Assessment of Kinase Selectivity, Enzyme Inhibition Kinetics and in Vitro Activity for Several Bruton Tyrosine Kinase (BTK) Inhibitors

对几种布鲁顿酪氨酸激酶(BTK)抑制剂的激酶选择性、酶抑制动力学和体外活性进行评估

Corrionero, Ana; Zhang, Xiaohu; Alfonso, Patricia; Morris, Patrick J; Klumpp-Thomas, Carleen; Melani, Christopher; McKnight, Crystal; Phelan, James D; Holland, David; Wilson, Kelli; Hoyt, Scott B; Roschewski, Mark; Tonge, Peter J; Wilson, Wyndham; Ceribelli, Michele; Staudt, Louis M; Thomas, Craig J

Direct Co-Targeting of Bcl-xL and Mcl-1 Exhibits Synergistic Effects in AR-V7-Expressing CRPC Models.

Bcl-xL 和 Mcl-1 的直接共同靶向在 AR-V7 表达的 CRPC 模型中表现出协同效应

Brim Benjamin C, Leon Andres F, Beatson Erica L, Kindrick Jessica D, Bhadresha Kinjal, Zhang Xiaohu, Napoli Giulia C, Risdon Emily N, Schmidt Keith T, Wilson Kelli M, McKnight Crystal, Beck Erin, Klumpp-Thomas Carleen, Ceribelli Michele, Yin JuanJuan, Sowalsky Adam G, Price Douglas K, Chau Cindy H, Thomas Craig J, Figg William D

A High-Throughput Screening Pipeline to Identify Methyltransferase and Exonuclease Inhibitors of SARS-CoV-2 NSP14

用于鉴定 SARS-CoV-2 NSP14 甲基转移酶和核酸外切酶抑制剂的高通量筛选流程

Hanson, Quinlin; Hu, Xin; Pal, Sourav; Recabo, Katlin; Ye, Lin; Poon, Ivy; Denson, John-Paul; Messing, Simon; Shen, Min; Wilson, Kelli M; Zakharov, Alexey; Esposito, Dominic; Martinez, Natalia J

A machine learning-based analysis method for small molecule high content screening of three-dimensional cancer spheroid morphology.

基于机器学习的小分子高内涵筛选三维癌球体形态的分析方法。

Goyal Vishakha, Blivis Dvir, Titus Steven A, Itkin Misha, Zakharov Alexey, Wilson Kelli, Martinez Natalia J, Voss Ty C