Asymmetric cycloadditions of o-quinone methides employing chiral ammonium fluoride precatalysts

利用手性氟化铵预催化剂的邻醌甲化物不对称环加成反应

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Abstract

The catalytic, enantioselective, [4 + 2] cycloaddition reaction of ortho-quinone methides with silyl ketene acetals is described. This mechanistically interesting reaction, initiated by a chiral cinchona alkaloid-derived ammonium fluoride "precatalyst" complex, affords a variety of alkyl- and aryl-substituted 3,4-dihydrocoumarin products in excellent yield and with good enantioselectivity.

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