日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Allosteric modulation and G-protein selectivity of the Ca(2+)-sensing receptor.

Ca(2+)敏感受体的变构调节和G蛋白选择性

He Feng, Wu Cheng-Guo, Gao Yang, Rahman Sabrina N, Zaoralová Magda, Papasergi-Scott Makaía M, Gu Ting-Jia, Robertson Michael J, Seven Alpay B, Li Lingjun, Mathiesen Jesper M, Skiniotis Georgios

Insights into distinct signaling profiles of the µOR activated by diverse agonists

深入了解不同激动剂激活的µOR的不同信号传导特征

Qianhui Qu #, Weijiao Huang #, Deniz Aydin #, Joseph M Paggi #, Alpay B Seven #, Haoqing Wang, Soumen Chakraborty, Tao Che, Jeffrey F DiBerto, Michael J Robertson, Asuka Inoue, Carl-Mikael Suomivuori, Bryan L Roth, Susruta Majumdar, Ron O Dror, Brian K Kobilka, Georgios Skiniotis9

Time-resolved cryo-EM of G protein activation by a GPCR

利用时间分辨冷冻电镜观察G蛋白受体激活G蛋白的过程

Papasergi-Scott, Makaía M; Pérez-Hernández, Guillermo; Batebi, Hossein; Gao, Yang; Eskici, Gözde; Seven, Alpay B; Panova, Ouliana; Hilger, Daniel; Casiraghi, Marina; He, Feng; Maul, Luis; Gmeiner, Peter; Kobilka, Brian K; Hildebrand, Peter W; Skiniotis, Georgios

Bespoke library docking for 5-HT2A receptor agonists with antidepressant activity

针对具有抗抑郁活性的5-HT2A受体激动剂的定制化化合物库对接

Anat Levit Kaplan #,Danielle N Confair #,Kuglae Kim #,Ximena Barros-Álvarez #,Ramona M Rodriguiz,Ying Yang,Oh Sang Kweon,Tao Che,John D McCorvy,David N Kamber,James P Phelan,Luan Carvalho Martins,Vladimir M Pogorelov,Jeffrey F DiBerto,Samuel T Slocum,Xi-Ping Huang,Jain Manish Kumar,Michael J Robertson,Ouliana Panova,Alpay B Seven,Autumn Q Wetsel,William C Wetsel,John J Irwin,Georgios Skiniotis,Brian K Shoichet,Bryan L Roth,Jonathan A Ellman

The tethered peptide activation mechanism of adhesion GPCRs

粘附性GPCR的系链肽激活机制

Ximena Barros-Álvarez #,Robert M Nwokonko #,Alexander Vizurraga #,Donna Matzov #,Feng He,Makaía M Papasergi-Scott,Michael J Robertson,Ouliana Panova,Eliane Hadas Yardeni,Alpay B Seven,Frank E Kwarcinski,Hongyu Su,Maria Claudia Peroto,Justin G Meyerowitz,Moran Shalev-Benami,Gregory G Tall,Georgios Skiniotis

Signaling snapshots of a serotonin receptor activated by the prototypical psychedelic LSD

典型迷幻剂LSD激活血清素受体的信号快照

Can Cao,Ximena Barros-Álvarez,Shicheng Zhang,Kuglae Kim,Marc A Dämgen,Ouliana Panova,Carl-Mikael Suomivuori,Jonathan F Fay,Xiaofang Zhong,Brian E Krumm,Ryan H Gumpper,Alpay B Seven,Michael J Robertson,Nevan J Krogan,Ruth Hüttenhain,David E Nichols,Ron O Dror,Georgios Skiniotis,Bryan L Roth

Structure determination of inactive-state GPCRs with a universal nanobody.

利用通用纳米抗体测定非活性状态GPCR的结构

Robertson Michael J, Papasergi-Scott Makaía M, He Feng, Seven Alpay B, Meyerowitz Justin G, Panova Ouliana, Peroto Maria Claudia, Che Tao, Skiniotis Georgios

G-protein activation by a metabotropic glutamate receptor

代谢型谷氨酸受体激活 G 蛋白

Alpay B Seven, Ximena Barros-Álvarez, Marine de Lapeyrière, Makaía M Papasergi-Scott, Michael J Robertson, Chensong Zhang, Robert M Nwokonko, Yang Gao, Justin G Meyerowitz, Jean-Philippe Rocher, Dominik Schelshorn, Brian K Kobilka, Jesper M Mathiesen, Georgios Skiniotis

Asymmetric activation of the calcium-sensing receptor homodimer

钙敏感受体同型二聚体的不对称激活

Yang Gao, Michael J Robertson, Sabrina N Rahman, Alpay B Seven, Chensong Zhang, Justin G Meyerowitz, Ouliana Panova, Fadil M Hannan, Rajesh V Thakker, Hans Bräuner-Osborne, Jesper M Mathiesen, Georgios Skiniotis

Structures of metabotropic GABAB receptor

代谢型 GABAB 受体的结构

Makaía M Papasergi-Scott #, Michael J Robertson #, Alpay B Seven, Ouliana Panova, Jesper M Mathiesen, Georgios Skiniotis