日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small-molecule OPA1 inhibitors reverse mitochondrial adaptations to overcome therapy resistance in acute myeloid leukemia

小分子OPA1抑制剂逆转线粒体适应性,从而克服急性髓系白血病的治疗耐药性。

Sofia La Vecchia ,Saurav Doshi ,Petros Antonoglou ,Tanima Kundu ,Wafa Al Santli ,Kleopatra Avrampou ,Matthew T Witkowski ,Anna Pellattiero ,Federico Magrin ,Kristina Ames ,Amit Verma ,Kira Gritsman ,Xiaoyang Su ,Andrea Mattarei ,Iannis Aifantis ,Luca Scorrano ,Christina Glytsou

Small molecule OPA1 inhibitors amplify cytochrome c release and reverse cancer cells resistance to Bcl-2 inhibitors

小分子OPA1抑制剂可增强细胞色素c的释放,并逆转癌细胞对Bcl-2抑制剂的耐药性。

Anna Pellattiero,Charlotte Quirin,Federico Magrin,Mattia Sturlese,Alberto Fracasso,Nikolaos Biris,Stéphanie Herkenne,Laura Cendron,Evripidis Gavathiotis,Stefano Moro,Andrea Mattarei,Luca Scorrano

Selective inhibition of mitochondrial Kv1.3 prevents and alleviates multiple sclerosis in vivo

选择性抑制线粒体Kv1.3可预防和缓解体内多发性硬化症。

Beatrice Angi # ,Tatiana Varanita # ,Marco Puthenparampil ,Valentina Scattolini ,Michael Donadon ,Mitra Tavakoli ,Marta Favero ,Maguie El Boustani ,Matthias Soddemann ,Lucia Biasutto ,Diletta Arcidiacono ,Alberto Ongaro ,Andrea Mattarei ,Livio Trentin ,Gregory Wilson ,Erich Gulbins ,Paolo Gallo ,Ildiko Szabo

Drug-Drug Interaction Studies of Esmethadone (REL-1017) Involving CYP3A4- and CYP2D6-Mediated Metabolism

涉及 CYP3A4 和 CYP2D6 介导代谢的 Esmethadone (REL-1017) 药物相互作用研究

Nicola Ferri, Sara De Martin, James Stuart, Sergio Traversa, Franco Folli, Marco Pappagallo, Cedric O'Gorman, Clotilde Guidetti, Andrea Mattarei, Charles E Inturrisi, Paolo L Manfredi

The mitochondrial ATP-dependent potassium channel (mitoKATP) controls skeletal muscle structure and function

线粒体 ATP 依赖性钾通道 (mitoKATP) 控制骨骼肌的结构和功能

Giulia Di Marco #, Gaia Gherardi #, Agnese De Mario, Ilaria Piazza, Martina Baraldo, Andrea Mattarei, Bert Blaauw, Rosario Rizzuto, Diego De Stefani, Cristina Mammucari

Sphingosine is involved in PAPTP-induced death of pancreas cancer cells by interfering with mitochondrial functions

鞘氨醇通过干扰线粒体功能参与 PAPTP 诱导的胰腺癌细胞死亡

Sameer H Patel, Gregory C Wilson, Yuqing Wu, Simone Keitsch, Barbara Wilker, Andrea Mattarei, Syed A Ahmad, Ildiko Szabo, Erich Gulbins

Defective excitation-contraction coupling and mitochondrial respiration precede mitochondrial Ca2+ accumulation in spinobulbar muscular atrophy skeletal muscle

脊髓延髓肌萎缩症骨骼肌中,兴奋-收缩耦联缺陷和线粒体呼吸作用先于线粒体Ca2+积累。

Caterina Marchioretti # ,Giulia Zanetti # ,Marco Pirazzini # ,Gaia Gherardi ,Leonardo Nogara ,Roberta Andreotti ,Paolo Martini ,Lorenzo Marcucci ,Marta Canato ,Samir R Nath ,Emanuela Zuccaro ,Mathilde Chivet ,Cristina Mammucari ,Marco Pacifici ,Anna Raffaello ,Rosario Rizzuto ,Andrea Mattarei ,Maria A Desbats ,Leonardo Salviati ,Aram Megighian ,Gianni Sorarù ,Elena Pegoraro ,Elisa Belluzzi ,Assunta Pozzuoli ,Carlo Biz ,Pietro Ruggieri ,Chiara Romualdi ,Andrew P Lieberman ,Gopal J Babu ,Marco Sandri ,Bert Blaauw ,Manuela Basso ,Maria Pennuto

DA7R: A 7-Letter Zip Code to Target PDAC

DA7R:针对 PDAC 的 7 个字母邮政编码

Sofia Parrasia, Andrea Rossa, Nicola Roncaglia, Andrea Mattarei, Claudia Honisch, Ildikò Szabò, Paolo Ruzza, Lucia Biasutto

Pharmacological modulation of Kv1.3 potassium channel selectively triggers pathological B lymphocyte apoptosis in vivo in a genetic CLL model

药理学调节 Kv1.3 钾通道选择性地触发遗传性 CLL 模型中的体内病理性 B 淋巴细胞凋亡

Filippo Severin #, Andrea Urbani #, Tatiana Varanita #, Magdalena Bachmann, Michele Azzolini, Veronica Martini, Marco Pizzi, Angelo Paolo Dei Tos, Federica Frezzato, Andrea Mattarei, Paolo Ghia, Maria Teresa Sabrina Bertilaccio, Erich Gulbins, Cristina Paradisi, Mario Zoratti, Gianpietro Carlo Semen

Pharmacological targeting of the mitochondrial calcium-dependent potassium channel KCa3.1 triggers cell death and reduces tumor growth and metastasis in vivo

药物靶向线粒体钙依赖性钾通道 KCa3.1 可引发细胞死亡并减少体内肿瘤的生长和转移

Magdalena Bachmann, Andrea Rossa, Tatiana Varanita, Bernard Fioretti, Lucia Biasutto, Stefan Milenkovic, Vanessa Checchetto, Roberta Peruzzo, Syed A Ahmad, Sameer H Patel, Robert Lukowski, Michael J Edwards, Matteo Ceccarelli, Erich Gulbins, Mario Zoratti, Andrea Mattarei, Ildiko Szabo