日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

AI-driven discovery of synergistic drug combinations against pancreatic cancer.

利用人工智能发现对抗胰腺癌的协同药物组合

Pourmousa Mohsen, Jain Sankalp, Barnaeva Elena, Jin Wengong, Hochuli Joshua, Itkin Zina, Maxfield Travis, Melo-Filho Cleber, Thieme Andrew, Wilson Kelli, Klumpp-Thomas Carleen, Michael Sam, Southall Noel, Jaakkola Tommi, Muratov Eugene N, Barzilay Regina, Tropsha Alexander, Ferrer Marc, Zakharov Alexey V

A defined roadmap of radial glia and astrocyte differentiation from human pluripotent stem cells

人类多能干细胞向放射状胶质细胞和星形胶质细胞分化的明确路线图

Vukasin M Jovanovic, Claire Weber, Jaroslav Slamecka, Seungmi Ryu, Pei-Hsuan Chu, Chaitali Sen, Jason Inman, Juliana Ferreira De Sousa, Elena Barnaeva, Marissa Hirst, David Galbraith, Pinar Ormanoglu, Yogita Jethmalani, Jennifer Colon Mercado, Sam Michael, Michael E Ward, Anton Simeonov, Ty C Voss, 

Discovery of a functionally selective ghrelin receptor (GHSR(1a)) ligand for modulating brain dopamine

发现一种功能选择性生长素释放肽受体(GHSR(1a))配体,用于调节脑多巴胺

Gross, J D; Kim, D W; Zhou, Y; Jansen, D; Slosky, L M; Clark, N B; Ray, C R; Hu, X; Southall, N; Wang, A; Xu, X; Barnaeva, E; Wetsel, W C; Ferrer, M; Marugan, J J; Caron, M G; Barak, L S; Toth, K

Discovery of small molecule agonists of the Relaxin Family Peptide Receptor 2

发现松弛素家族肽受体 2 的小分子激动剂

Maria Esteban-Lopez, Kenneth J Wilson, Courtney Myhr, Elena M Kaftanovskaya, Mark J Henderson, Noel T Southall, Xin Xu, Amy Wang, Xin Hu, Elena Barnaeva, Wenjuan Ye, Emmett R George, John T Sherrill, Marc Ferrer, Roy Morello, Irina U Agoulnik, Juan J Marugan, Alexander I Agoulnik

Discovery of small molecule inhibitors that effectively disrupt IQGAP1-Cdc42 interaction in breast cancer cells

发现可有效破坏乳腺癌细胞中 IQGAP1-Cdc42 相互作用的小分子抑制剂

Samar Sayedyahossein, Jessica Smith, Elena Barnaeva, Zhigang Li, Jun Choe, Michael Ronzetti, Christopher Dextras, Xin Hu, Juan Marugan, Noel Southall, Bolormaa Baljinnyam, Louise Thines, Andy D Tran, Marc Ferrer, David B Sacks

Robotic high-throughput biomanufacturing and functional differentiation of human pluripotent stem cells

机器人高通量生物制造和人类多能干细胞的功能分化

Carlos A Tristan, Pinar Ormanoglu, Jaroslav Slamecka, Claire Malley, Pei-Hsuan Chu, Vukasin M Jovanovic, Yeliz Gedik, Yogita Jethmalani, Charles Bonney, Elena Barnaeva, John Braisted, Sunil K Mallanna, Dorjbal Dorjsuren, Michael J Iannotti, Ty C Voss, Sam Michael, Anton Simeonov, Ilyas Singeç

Identification of a Small-Molecule Inhibitor That Disrupts the SIX1/EYA2 Complex, EMT, and Metastasis

鉴定一种可破坏 SIX1/EYA2 复合物、EMT 和转移的小分子抑制剂

Hengbo Zhou ,Melanie A Blevins ,Jessica Y Hsu ,Deguang Kong ,Matthew D Galbraith ,Andrew Goodspeed ,Rachel Culp-Hill ,Michael U J Oliphant ,Dominique Ramirez ,Lingdi Zhang ,Jennyvette Trinidad-Pineiro ,Lesley Mathews Griner ,Rebecca King ,Elena Barnaeva ,Xin Hu ,Noel T Southall ,Marc Ferrer ,Daniel L Gustafson ,Daniel P Regan ,Angelo D'Alessandro ,James C Costello ,Samarjit Patnaik ,Juan Marugan ,Rui Zhao ,Heide L Ford

Robotic High-Throughput Biomanufacturing and Functional Differentiation of Human Pluripotent Stem Cells

机器人高通量生物制造和人类多能干细胞的功能分化

Carlos A Tristan, Pinar Ormanoglu, Jaroslav Slamecka, Claire Malley, Pei-Hsuan Chu, Vukasin M Jovanovic, Yeliz Gedik, Charles Bonney, Elena Barnaeva, John Braisted, Sunil K Mallanna, Dorjbal Dorjsuren, Michael J Iannotti, Ty C Voss, Sam Michael, Anton Simeonov, Ilyas Singeç

Identification of Chemotype Agonists for Human Resolvin D1 Receptor DRV1 with Pro-Resolving Functions

具有促分解功能的人类 Resolvin D1 受体 DRV1 化学型激动剂的鉴定

Nan Chiang, Elena Barnaeva, Xin Hu, Juan Marugan, Noel Southall, Marc Ferrer, Charles N Serhan

A large scale high-throughput screen identifies chemical inhibitors of phosphatidylinositol 4-kinase type II alpha

大规模高通量筛选鉴定了磷脂酰肌醇 4-激酶 II 型 α 的化学抑制剂

Nivedita Sengupta, Marko Jović, Elena Barnaeva, David W Kim, Xin Hu, Noel Southall, Milan Dejmek, Ivana Mejdrova, Radim Nencka, Adriana Baumlova, Dominika Chalupska, Evzen Boura, Marc Ferrer, Juan Marugan, Tamas Balla