日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dysregulation of the epigenetic landscape of normal aging in Alzheimer's disease

阿尔茨海默病中正常衰老表观遗传景观的失调

Raffaella Nativio, Greg Donahue, Amit Berson, Yemin Lan, Alexandre Amlie-Wolf, Ferit Tuzer, Jon B Toledo, Sager J Gosai, Brian D Gregory, Claudio Torres, John Q Trojanowski, Li-San Wang, F Brad Johnson, Nancy M Bonini, Shelley L Berger

HIV antiretroviral therapy drugs induce premature senescence and altered physiology in HUVECs

HIV 抗逆转录病毒治疗药物可诱发 HUVEC 过早衰老和生理改变

Justin Cohen, Luca D'Agostino, Ferit Tuzer, Claudio Torres

Astrocyte Senescence and Metabolic Changes in Response to HIV Antiretroviral Therapy Drugs

HIV 抗逆转录病毒治疗药物引起的星形胶质细胞衰老和代谢变化

Justin Cohen, Luca D'Agostino, Joel Wilson, Ferit Tuzer, Claudio Torres

Covalent conjugation of a peptide triazole to HIV-1 gp120 enables intramolecular binding site occupancy

肽三唑与 HIV-1 gp120 的共价结合可实现分子内结合位点占据

Ali Emileh, Caitlin Duffy, Andrew P Holmes, Arangassery Rosemary Bastian, Rachna Aneja, Ferit Tuzer, Srivats Rajagopal, Huiyuan Li, Cameron F Abrams, Irwin M Chaiken

Non-natural peptide triazole antagonists of HIV-1 envelope gp120

HIV-1 包膜 gp120 的非天然肽三唑拮抗剂

Kantharaju Kamanna, Rachna Aneja, Caitlin Duffy, Pamela Kubinski, Diogo Rodrigo Moreira, Lauren D Bailey, Karyn McFadden, Arne Schön, Andrew Holmes, Ferit Tuzer, Mark Contarino, Ernesto Freire, Irwin M Chaiken

HIV-1 Env gp120 structural determinants for peptide triazole dual receptor site antagonism

HIV-1 Env gp120 肽三唑双受体位点拮抗作用的结构决定因素

Ferit Tuzer, Navid Madani, Kantharaju Kamanna, Isaac Zentner, Judith LaLonde, Andrew Holmes, Elizabeth Upton, Srivats Rajagopal, Karyn McFadden, Mark Contarino, Joseph Sodroski, Irwin Chaiken

A model of peptide triazole entry inhibitor binding to HIV-1 gp120 and the mechanism of bridging sheet disruption

肽三唑进入抑制剂与HIV-1 gp120结合的模型及桥接片破坏机制

Ali Emileh, Ferit Tuzer, Herman Yeh, Muddegowda Umashankara, Diogo R M Moreira, Judith M Lalonde, Carole A Bewley, Cameron F Abrams, Irwin M Chaiken

The active core in a triazole peptide dual-site antagonist of HIV-1 gp120

HIV-1 gp120 三唑肽双位点拮抗剂的活性核心

Muddegowda Umashankara, Karyn McFadden, Isaac Zentner, Arne Schön, Srivats Rajagopal, Ferit Tuzer, Syna A Kuriakose, Mark Contarino, Judith Lalonde, Ernesto Freire, Irwin Chaiken

Introducing metallocene into a triazole peptide conjugate reduces its off-rate and enhances its affinity and antiviral potency for HIV-1 gp120

将茂金属引入三唑肽缀合物可降低其解离率并增强其对 HIV-1 gp120 的亲和力和抗病毒效力

Hosahudya Gopi, Simon Cocklin, Vanessa Pirrone, Karyn McFadden, Ferit Tuzer, Isaac Zentner, Sandya Ajith, Sabine Baxter, Navneet Jawanda, Fred C Krebs, Irwin M Chaiken

Structural determinants for affinity enhancement of a dual antagonist peptide entry inhibitor of human immunodeficiency virus type-1

人类免疫缺陷病毒 1 型双重拮抗肽进入抑制剂亲和力增强的结构决定因素

Hosahudya Gopi, M Umashankara, Vanessa Pirrone, Judith LaLonde, Navid Madani, Ferit Tuzer, Sabine Baxter, Isaac Zentner, Simon Cocklin, Navneet Jawanda, Shendra R Miller, Arne Schön, Jeffrey C Klein, Ernesto Freire, Fred C Krebs, Amos B Smith, Joseph Sodroski, Irwin Chaiken