日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dual targeting of RET and SRC synergizes in RET fusion-positive cancer cells

RET 和 SRC 双重靶向治疗对 RET 融合阳性癌细胞具有协同作用。

Son, Juhyeon; Remsing Rix, Lily L; Fang, Bin; Welsh, Eric A; Bremer, Nicole V; Foglizzo, Valentina; Roa, Paola; Sigcha-Coello, Nickole; Liao, Yi; Haura, Eric B; Drilon, Alexander; Koomen, John M; Cocco, Emiliano; Rix, Uwe

High-throughput discovery and characterisation of pentafluorobenzene sulfonamide modifiers of Aurora A kinase

利用高通量方法发现和表征Aurora A激酶的五氟苯磺酰胺修饰剂

Chesti, Julian; Miles, Jennifer A; Collins, Lawrence J; McCallum, Hamish A; Foglizzo, Martina; Ahangar, Mohd Syed; Zeqiraj, Elton; Bayliss, Richard; Warriner, Stuart L; Wright, Megan H; Nelson, Adam

A programmed decline in ribosome levels governs human early neurodevelopment

核糖体水平的程序性下降控制着人类早期神经发育。

Chunyang Ni # ,Yudong Wei # ,Barbara Vona # ,Dayea Park ,Yulei Wei ,Daniel A Schmitz ,Yi Ding ,Masahiro Sakurai ,Emily Ballard ,Leijie Li ,Yan Liu ,Ashwani Kumar ,Chao Xing ,Shenlu Qin ,Sangin Kim ,Martina Foglizzo ,Jianchao Zhao ,Hyung-Goo Kim ,Cumhur Ekmekci ,Ehsan Ghayoor Karimiani ,Shima Imannezhad ,Fatemeh Eghbal ,Reza Shervin Badv ,Eva Maria Christina Schwaibold ,Mohammadreza Dehghani ,Mohammad Yahya Vahidi Mehrjardi ,Zahra Metanat ,Hosein Eslamiyeh ,Ebtissal Khouj ,Saleh Mohammed Nasser Alhajj ,Aziza Chedrawi ,Khushnooda Ramzan ,Jamil A Hashmi ,Majed M Alluqmani ,Sulman Basit ,Danai Veltra ,Nikolaos M Marinakis ,Georgios Niotakis ,Pelagia Vorgia ,Christalena Sofocleous ,Hane Lee ,Won Chan Jeong ,Muhammad Umair ,Muhammad Bilal ,César Augusto Pinheiro Ferreira Alves ,Matthew Sieber ,Michael Kruer ,Henry Houlden ,Fowzan S Alkuraya ,Elton Zeqiraj ,Roger A Greenberg ,Can Cenik ,Leqian Yu ,Reza Maroofian ,Jun Wu ,Michael Buszczak

Molecular glues that inhibit deubiquitylase activity and inflammatory signaling.

抑制去泛素化酶活性和炎症信号的分子胶

Chandler Francesca, Reddy Poli Adi Narayana, Bhutda Smita, Ross Rebecca L, Datta Arindam, Walden Miriam, Walker Kieran, Di Donato Stefano, Cassel Joel A, Prakesch Michael A, Aman Ahmed, Datti Alessandro, Campbell Lisa J, Foglizzo Martina, Bell Lillie, Stein Daniel N, Ault James R, Al-Awar Rima S, Calabrese Antonio N, Sicheri Frank, Del Galdo Francesco, Salvino Joseph M, Greenberg Roger A, Zeqiraj Elton

Responsiveness of different MET tumour alterations to type I and type II MET inhibitors.

不同MET肿瘤改变对I型和II型MET抑制剂的反应性

Murciano-Goroff Yonina R, Foglizzo Valentina, Chang Jason, Rekhtman Natasha, Sisk Ann Elizabeth, Gibson Jamie, Judka Lia, Clemens Kristen, Roa Paola, Ahmed Shaza Sayed, Bremer Nicole V, Binaco Courtney Lynn, Muzungu Sherifah Kemigisha, Rodriguez Estelamari, Merrill Madeline, Sgroe Erica, Repetto Matteo, Stadler Zsofia K, Berger Michael F, Yu Helena A, Toska Eneda, Kannan Srinivasaraghavan, Verma Chandra S, Drilon Alexander, Cocco Emiliano

The UFM1 E3 ligase recognizes and releases 60S ribosomes from ER translocons

UFM1 E3 连接酶识别并从 ER 转运子中释放 60S 核糖体

Linda Makhlouf #, Joshua J Peter #, Helge M Magnussen #, Rohan Thakur, David Millrine, Thomas C Minshull, Grace Harrison, Joby Varghese, Frederic Lamoliatte, Martina Foglizzo, Thomas Macartney, Antonio N Calabrese, Elton Zeqiraj, Yogesh Kulathu

The SPATA5-SPATA5L1 ATPase complex directs replisome proteostasis to ensure genome integrity

SPATA5-SPATA5L1 ATPase复合物指导复制体蛋白稳态以确保基因组完整性

Vidhya Krishnamoorthy, Martina Foglizzo, Robert L Dilley, Angela Wu, Arindam Datta, Parul Dutta, Lisa J Campbell, Oksana Degtjarik, Laura J Musgrove, Antonio N Calabrese, Elton Zeqiraj, Roger A Greenberg

Zurletrectinib is a next-generation TRK inhibitor with strong intracranial activity against NTRK fusion-positive tumours with on-target resistance to first-generation agents

Zurletrectinib 是一种新一代 TRK 抑制剂,对具有靶向耐药性的 NTRK 融合阳性肿瘤具有强大的颅内活性。

Roa, Paola; Foglizzo, Valentina; Harada, Guilherme; Repetto, Matteo; Kulick, Amanda; de Stanchina, Elisa; de Marchena, Michelle; Auwardt, Supipi; Sayed Ahmed, Shaza; Bremer, Nicole Virginia; Yang, Soo-Ryum; Feng, Yangbo; Zhou, Chao; Kong, Norman; Liang, Ruixia; Xu, Haipeng; Zhang, Bin; Bardelli, Alberto; Toska, Eneda; Ventura, Andrea; Drilon, Alexander; Cocco, Emiliano

Mutations in the Serine/Threonine Kinase BRAF: Oncogenic Drivers in Solid Tumors

丝氨酸/苏氨酸激酶BRAF的突变:实体瘤的致癌驱动因素

Roa, Paola; Bremer, Nicole Virginia; Foglizzo, Valentina; Cocco, Emiliano

Molecular glues that inhibit specific Zn2+-dependent DUB activity and inflammation

抑制特定 Zn2+ 依赖性 DUB 活性和炎症的分子胶

Francesca Chandler, Poli Adi Narayana Reddy, Smita Bhutda, Rebecca L Ross, Miriam Walden, Kieran Walker, Stefano Di Donato, Joel A Cassel, Michael A Prakesch, Ahmed Aman, Alessandro Datti, Lisa J Campbell, Martina Foglizzo, Lillie Bell, Daniel N Stein, James R Ault, Rima S Al-Awar, Antonio N Calabre