Targeting histone acetylation dynamics and oncogenic transcription by catalytic P300/CBP inhibition
通过抑制催化性P300/CBP来靶向组蛋白乙酰化动态和致癌转录
期刊:Molecular Cell
影响因子:14.5
doi:10.1016/j.molcel.2021.04.015
Simon J Hogg ,Olga Motorna ,Leonie A Cluse ,Timothy M Johanson ,Hannah D Coughlan ,Ramya Raviram ,Robert M Myers ,Matteo Costacurta ,Izabela Todorovski ,Lizzy Pijpers ,Stefan Bjelosevic ,Tobias Williams ,Shannon N Huskins ,Conor J Kearney ,Jennifer R Devlin ,Zheng Fan ,Jafar S Jabbari ,Ben P Martin ,Mohamed Fareh ,Madison J Kelly ,Daphné Dupéré-Richer ,Jarrod J Sandow ,Breon Feran ,Deborah Knight ,Tiffany Khong ,Andrew Spencer ,Simon J Harrison ,Gareth Gregory ,Vihandha O Wickramasinghe ,Andrew I Webb ,Phillippa C Taberlay ,Kenneth D Bromberg ,Albert Lai ,Anthony T Papenfuss ,Gordon K Smyth ,Rhys S Allan ,Jonathan D Licht ,Dan A Landau ,Omar Abdel-Wahab ,Jake Shortt ,Stephin J Vervoort ,Ricky W Johnstone